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MX2018002538A - Derivados de espinosina. - Google Patents

Derivados de espinosina.

Info

Publication number
MX2018002538A
MX2018002538A MX2018002538A MX2018002538A MX2018002538A MX 2018002538 A MX2018002538 A MX 2018002538A MX 2018002538 A MX2018002538 A MX 2018002538A MX 2018002538 A MX2018002538 A MX 2018002538A MX 2018002538 A MX2018002538 A MX 2018002538A
Authority
MX
Mexico
Prior art keywords
derivatives
spinosyn
insecticides
spinosyn derivatives
spinosyns
Prior art date
Application number
MX2018002538A
Other languages
English (en)
Inventor
Calabrese Andrew
Original Assignee
Agrimetis Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agrimetis Llc filed Critical Agrimetis Llc
Publication of MX2018002538A publication Critical patent/MX2018002538A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/22Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N45/00Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring
    • A01N45/02Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring having three carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D313/00Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N2300/00Combinations or mixtures of active ingredients covered by classes A01N27/00 - A01N65/48 with other active or formulation relevant ingredients, e.g. specific carrier materials or surfactants, covered by classes A01N25/00 - A01N65/48

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dermatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicinal Preparation (AREA)

Abstract

Se proveen composiciones que incluyen derivados de espinosinas y métodos de producción de derivados de espinosinas. Los derivados de espinosina descriptos en la presente incluyen derivados de espinosina funcionalizados en el doble enlace C5-C6 de la espinosina A para proveer un sistema de anillo adicional. El método produce derivados de espinosina que exhiben actividad hacia insectos, arácnidos, y/o nemátodos y que resultan de utilidad en los mercados agrícola y de la salud animal.
MX2018002538A 2015-09-03 2016-09-01 Derivados de espinosina. MX2018002538A (es)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US201562214083P 2015-09-03 2015-09-03
US201662290676P 2016-02-03 2016-02-03
US201662303015P 2016-03-03 2016-03-03
US201662303078P 2016-03-03 2016-03-03
US201662380664P 2016-08-29 2016-08-29
PCT/US2016/049870 WO2017040763A1 (en) 2015-09-03 2016-09-01 Spinosyn derivatives as insecticides

Publications (1)

Publication Number Publication Date
MX2018002538A true MX2018002538A (es) 2018-08-14

Family

ID=56940400

Family Applications (3)

Application Number Title Priority Date Filing Date
MX2018002540A MX2018002540A (es) 2015-09-03 2016-09-01 Derivados de espinosina y metodos de preparacion.
MX2018002538A MX2018002538A (es) 2015-09-03 2016-09-01 Derivados de espinosina.
MX2018002539A MX2018002539A (es) 2015-09-03 2016-09-02 Derivados de espinosina y metodos de preparacion.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
MX2018002540A MX2018002540A (es) 2015-09-03 2016-09-01 Derivados de espinosina y metodos de preparacion.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2018002539A MX2018002539A (es) 2015-09-03 2016-09-02 Derivados de espinosina y metodos de preparacion.

Country Status (12)

Country Link
US (3) US10570166B2 (es)
EP (3) EP3344611B1 (es)
JP (3) JP2018532708A (es)
KR (3) KR20180048871A (es)
CN (3) CN108137529A (es)
AU (3) AU2016317854A1 (es)
BR (2) BR112018004310A2 (es)
CA (3) CA2997540A1 (es)
CL (2) CL2018000527A1 (es)
IL (2) IL257760A (es)
MX (3) MX2018002540A (es)
WO (4) WO2017040763A1 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10570166B2 (en) 2015-09-03 2020-02-25 Agrimetis, Llc Spinosyn derivatives as insecticides
JP2020506891A (ja) 2017-01-13 2020-03-05 アグリメティス,エルエルシー アジリジンスピノシン誘導体および製造方法
CN119157876A (zh) * 2017-12-15 2024-12-20 塔苏斯制药有限公司 用于治疗睑炎的异恶唑啉驱虫剂制剂和方法
AR116524A1 (es) * 2018-10-04 2021-05-19 Elanco Tiergesundheit Ag Potenciación de tratamiento de helmintos
US12502377B2 (en) 2019-04-04 2025-12-23 Tarsus Pharmaceuticals, Inc. Method of eradicating ticks that attach to humans using lotilaner formulations
BR112023021924A2 (pt) 2021-04-23 2024-01-16 Acies Bio D O O Composto, composição, uso de um composto, e, métodos para controlar uma praga e para proteger uma planta contra uma praga de plantas
EP4079744B1 (en) 2021-04-23 2025-08-06 Acies Bio d.o.o. Novel spinosyn compounds and their use as a pesticide
EP4101858A1 (en) 2021-06-08 2022-12-14 Acies Bio d.o.o. Novel spinosyn compounds

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CZ296136B6 (cs) 1998-07-02 2006-01-11 Eli Lilly And Company Prostredek pro péci o vlasy
EP1207757B1 (en) 1999-08-12 2005-02-23 Eli Lilly And Company Ectoparasiticidal aqueous suspension formulations of spinosyns
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EP2445506B1 (en) 2009-06-24 2014-12-31 Entarco SA The use of spinosyns and spinosyn compositions against diseases caused by protozoans, viral infections and cancer
KR20120098930A (ko) 2010-01-25 2012-09-05 일라이 릴리 앤드 캄파니 말과 말파리 유충을 내부적으로 억제 또는 처리하기 위한 방법
JP2013542737A (ja) 2010-11-05 2013-11-28 イーライ リリー アンド カンパニー 昆虫侵入を阻害するための方法
EP2654757A1 (en) 2010-12-22 2013-10-30 Entarco SA The use of spinosyns and spinosyn compositions as local anesthetics and as antiarrhythmic agents
KR101960110B1 (ko) 2010-12-29 2019-03-19 다우 아그로사이언시즈 엘엘씨 곤충 방제 방법
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US10570166B2 (en) 2015-09-03 2020-02-25 Agrimetis, Llc Spinosyn derivatives as insecticides

Also Published As

Publication number Publication date
EP3344611B1 (en) 2020-11-04
EP3344612A1 (en) 2018-07-11
IL257759A (en) 2018-04-30
JP2018532708A (ja) 2018-11-08
US10570166B2 (en) 2020-02-25
US10711026B2 (en) 2020-07-14
AU2016317854A1 (en) 2018-03-15
KR20180041755A (ko) 2018-04-24
EP3344610B1 (en) 2020-05-06
KR20180048871A (ko) 2018-05-10
AU2016315860A1 (en) 2018-03-15
US20180251487A1 (en) 2018-09-06
BR112018004310A2 (pt) 2018-10-09
WO2017040769A1 (en) 2017-03-09
CN108026063A (zh) 2018-05-11
WO2017040882A1 (en) 2017-03-09
CL2018000525A1 (es) 2018-07-13
WO2017040763A1 (en) 2017-03-09
AU2016317848A1 (en) 2018-03-15
EP3344610A1 (en) 2018-07-11
IL257760A (en) 2018-04-30
US20190071464A1 (en) 2019-03-07
MX2018002539A (es) 2018-08-14
CN108137529A (zh) 2018-06-08
CA2997639A1 (en) 2017-03-09
EP3344612B1 (en) 2020-06-17
BR112018004313A2 (pt) 2018-10-09
MX2018002540A (es) 2018-08-14
CA2997499A1 (en) 2017-03-09
CL2018000527A1 (es) 2018-07-13
US20190309007A1 (en) 2019-10-10
KR20180050340A (ko) 2018-05-14
JP2018531912A (ja) 2018-11-01
EP3344611A1 (en) 2018-07-11
US10717756B2 (en) 2020-07-21
WO2017040878A1 (en) 2017-03-09
CN108137528A (zh) 2018-06-08
CA2997540A1 (en) 2017-03-09
JP2018532707A (ja) 2018-11-08

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