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CL2008001176A1 - Combinacion farmaceutica que comprende pregabalina y 1-(2-etoxietil)-5-[etil(metil)amino]-n-mesil-7-[(4-metil-2-piridil)amino]-1h-pirazol[4,3-d]pirimidina-3-carboxamida; composicion farmaceutica; y uso de la combinacion para el tratamiento del dolor. - Google Patents

Combinacion farmaceutica que comprende pregabalina y 1-(2-etoxietil)-5-[etil(metil)amino]-n-mesil-7-[(4-metil-2-piridil)amino]-1h-pirazol[4,3-d]pirimidina-3-carboxamida; composicion farmaceutica; y uso de la combinacion para el tratamiento del dolor.

Info

Publication number
CL2008001176A1
CL2008001176A1 CL2008001176A CL2008001176A CL2008001176A1 CL 2008001176 A1 CL2008001176 A1 CL 2008001176A1 CL 2008001176 A CL2008001176 A CL 2008001176A CL 2008001176 A CL2008001176 A CL 2008001176A CL 2008001176 A1 CL2008001176 A1 CL 2008001176A1
Authority
CL
Chile
Prior art keywords
amino
methyl
combination
mesyl
ethoxyethyl
Prior art date
Application number
CL2008001176A
Other languages
English (en)
Inventor
Paul Gunn Kevin
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39684397&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2008001176(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of CL2008001176A1 publication Critical patent/CL2008001176A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Composición farmacéutica que incluye pregabalina o una sal o solvato del mismo y 1-(2-etoxietil)-5-[etil(metil)amino]-n-mesil-7-[(4-metil-2-piridil)amino]-1h-pirazolo[4,3-d]pirimidina-3-carboxamida o un tautomero, un sal farmacéuticamente aceptable de la misma; y uso de la composición para el tratamiento del dolor.
CL2008001176A 2007-05-01 2008-04-23 Combinacion farmaceutica que comprende pregabalina y 1-(2-etoxietil)-5-[etil(metil)amino]-n-mesil-7-[(4-metil-2-piridil)amino]-1h-pirazol[4,3-d]pirimidina-3-carboxamida; composicion farmaceutica; y uso de la combinacion para el tratamiento del dolor. CL2008001176A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US91517407P 2007-05-01 2007-05-01

Publications (1)

Publication Number Publication Date
CL2008001176A1 true CL2008001176A1 (es) 2008-11-07

Family

ID=39684397

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2008001176A CL2008001176A1 (es) 2007-05-01 2008-04-23 Combinacion farmaceutica que comprende pregabalina y 1-(2-etoxietil)-5-[etil(metil)amino]-n-mesil-7-[(4-metil-2-piridil)amino]-1h-pirazol[4,3-d]pirimidina-3-carboxamida; composicion farmaceutica; y uso de la combinacion para el tratamiento del dolor.

Country Status (8)

Country Link
US (1) US20080293746A1 (es)
AR (1) AR066362A1 (es)
CL (1) CL2008001176A1 (es)
PA (1) PA8778901A1 (es)
PE (1) PE20090224A1 (es)
TW (1) TW200904401A (es)
UY (1) UY31062A1 (es)
WO (1) WO2008132589A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0934061B3 (en) 1996-07-24 2015-01-21 Warner-Lambert Company LLC Isobutylgaba and its derivatives for the treatment of pain

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0219024D0 (en) * 2002-08-15 2002-09-25 Pfizer Ltd Synergistic combinations
GB0327319D0 (en) * 2003-11-24 2003-12-24 Pfizer Ltd Novel pharmaceuticals

Also Published As

Publication number Publication date
AR066362A1 (es) 2009-08-12
UY31062A1 (es) 2008-11-28
WO2008132589A1 (en) 2008-11-06
US20080293746A1 (en) 2008-11-27
TW200904401A (en) 2009-02-01
PE20090224A1 (es) 2009-03-13
PA8778901A1 (es) 2008-12-18

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