CL2008000491A1 -
COMPOUNDS DERIVED FROM 1,1-DIOXO-1-TIA-DIAZA-DIBENZO CICLOHEPTENO; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; PROCESS FOR THE PREPARATION OF SUCH COMPOUNDS; AND ITS USE TO TREAT HEPATITIS C.
- Google Patents
COMPOUNDS DERIVED FROM 1,1-DIOXO-1-TIA-DIAZA-DIBENZO CICLOHEPTENO; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; PROCESS FOR THE PREPARATION OF SUCH COMPOUNDS; AND ITS USE TO TREAT HEPATITIS C.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tibotec Pharm LtdfiledCriticalTibotec Pharm Ltd
Publication of CL2008000491A1publicationCriticalpatent/CL2008000491A1/en
C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
C07D495/04—Ortho-condensed systems
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
A61P31/12—Antivirals
A—HUMAN NECESSITIES
A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines
(AREA)
Plural Heterocyclic Compounds
(AREA)
CL200800491A2007-02-162008-02-15
COMPOUNDS DERIVED FROM 1,1-DIOXO-1-TIA-DIAZA-DIBENZO CICLOHEPTENO; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; PROCESS FOR THE PREPARATION OF SUCH COMPOUNDS; AND ITS USE TO TREAT HEPATITIS C.
CL2008000491A1
(en)
COMPOUNDS DERIVED FROM 1,1-DIOXO-1-TIA-DIAZA-DIBENZO CICLOHEPTENO; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; PROCESS FOR THE PREPARATION OF SUCH COMPOUNDS; AND ITS USE TO TREAT HEPATITIS C.
COMPOUNDS DERIVED FROM SUBSTITUTED PYRIMIDINS; PROCEDURE FOR THE PREPARATION OF SUCH COMPOUNDS; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE TO TREAT HEMATOLOGICAL DISORDERS.
COMPOUNDS DERIVED FROM PYRIDOPIRIMIDINONES; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE TO TREAT PAIN, DEPRESSION, CARDIOVASCULAR DISEASES, RESPIRATORY DISEASES AND PSYCHIATRIC DISEASES.
COMPOUNDS DERIVED FROM MACROCICLES, INHIBITORS OF THE HEPATITIS C VIRUS; PREPARATION PROCEDURE; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUND; AND USE OF THE COMPOUND FOR THE TREATMENT OF HEPATITIS C.
COMPOUNDS DERIVED FROM 2,4-DIAMINO PIRIMIDINA, ANTRANILAMIDE INHIBITORS OF CINASA AURORA; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE TO TREAT CANCER.
COMPOUNDS DERIVED FROM SUBSTITUTED PYRIMIDINS; PROCESS FOR THE PREPARATION OF SUCH COMPOUNDS; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE FOR THE TREATMENT OF Rheumatoid ARTHRITIS, ATEROSCLEROSIS, AMONG OTHER DISEASES
COMPOUNDS DERIVED FROM PIRIMIDO [5,4-D] [2] BENZAZEPINA; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUND; AND USE OF THE COMPOUND FOR THE TREATMENT OF CANCER.
COMPOUNDS DERIVED FROM PIRAZOLILTIENOPIRIDINAS; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUND; AND USE OF THE COMPOUND IN THE INHIBITION OF ESCARAS.
Compounds derived from 4,5-dihydro-oxazol-2-ylamine; preparation procedure; pharmaceutical composition; and its use for the treatment of Alzheimer's disease.
COMPOUNDS DERIVED FROM IMIDAZOPIRIMIDINE; PROCESS TO PREPARE THE COMPOUNDS; PHARMACEUTICAL COMPOSITION; AND USE FOR THE PREVENTION AND / OR TREATMENT OF COGNITIVE DISORDERS.
COMPOUNDS DERIVED FROM SULFUR, INHIBITORS OF THE SERINA PROTEASA NS3 OF THE VIRUS OF HEPATITIS C; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUND; AND USE OF THE COMPOUND FOR THE TREATMENT OF ASSOCIATED DISORDERS TO HCV PROTEASE.
COMPOUNDS DERIVED FROM 3,5-DIOXI-BENZAMIDA; PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE TO TREAT A MEDIUM DISEASE THROUGH GLK, SUCH AS TYPE 2 DIABETES.
COMPOUNDS DERIVED FROM DIOXOALCANS AND DIOXOALKENS; PREPARATION PROCEDURE; PHARMACEUTICAL COMPOSITION; AND ITS USE TO TREAT ASTHMA, TOS, PURITO, HYPERSENSITIVITY.
COMPOUNDS DERIVED FROM IMIDAZOPIRIMIDINE; PROCESS TO PREPARE THE COMPOUNDS; PHARMACEUTICAL COMPOSITION; AND USE FOR THE PREVENTION AND / OR TREATMENT OF COGNITIVE DISORDERS.
COMPOUNDS DERIVED FROM 3-HIDROXI-1H-PIRIMIDIN-4-ONA OR 3-HIDROXI-PIRAN-4-ONA; PREPARATION PROCEDURE; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE TO TREAT A NEURODEGENERATIVE DISEASE CAUSED BY THE PRESENCE OF
COMPOUNDS DERIVED FROM AMINOMETIL-4-IMIDAZOL; PREPARATION PROCEDURE; PHARMACEUTICAL COMPOSITION THAT CONTAINS THEM; AND ITS USE TO TREAT DEPRESSION, ANXIETY, BIPOLAR DISORDER, AMONG OTHERS.
COMPOUNDS DERIVED FROM ISOQUINOLINILO AND ISOINDOLINILO, ANTAGONISTAS DE HISTAMINA-3; PROCEDURE FOR PREPARATION OF SUCH COMPOUNDS; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE TO TREAT NERVOUS SYSTEMS C
COMPOUNDS DERIVED FROM MACROCICLES, INHIBITORS OF THE SERINE PROTEASE OF HEPATITIS C; PREPARATION PROCEDURE; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUND; AND USE OF THE COMPOUND FOR THE TREATMENT OF HEPATITIS C.
COMPOUNDS DERIVED FROM NICOTINAMIDE; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE TO TREAT A DISEASE MEDIATED BY PROSTAGLANDIN D2 PRODUCED BY H-PGDS.