CA1336905C - Pyrido [3,2,1,ij]-1,3,4-benzoxadiazine derivatives - Google Patents
Pyrido [3,2,1,ij]-1,3,4-benzoxadiazine derivativesInfo
- Publication number
- CA1336905C CA1336905C CA000546674A CA546674A CA1336905C CA 1336905 C CA1336905 C CA 1336905C CA 000546674 A CA000546674 A CA 000546674A CA 546674 A CA546674 A CA 546674A CA 1336905 C CA1336905 C CA 1336905C
- Authority
- CA
- Canada
- Prior art keywords
- methyl
- oxo
- fluoro
- dihydro
- pyrido
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/58—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems with hetero atoms directly attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Quinoline Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP86112619.1 | 1986-09-12 | ||
| EP86112619 | 1986-09-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA1336905C true CA1336905C (en) | 1995-09-05 |
Family
ID=8195410
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA000546674A Expired - Lifetime CA1336905C (en) | 1986-09-12 | 1987-09-11 | Pyrido [3,2,1,ij]-1,3,4-benzoxadiazine derivatives |
Country Status (22)
| Country | Link |
|---|---|
| JP (3) | JPH0696578B2 (es) |
| KR (1) | KR960002857B1 (es) |
| CN (1) | CN1017800B (es) |
| AT (1) | AT389119B (es) |
| AU (1) | AU602534B2 (es) |
| CA (1) | CA1336905C (es) |
| CZ (1) | CZ281195B6 (es) |
| DK (1) | DK173330B1 (es) |
| DZ (1) | DZ1124A1 (es) |
| FI (1) | FI86428C (es) |
| HU (1) | HU199481B (es) |
| IE (1) | IE61624B1 (es) |
| IL (1) | IL83814A (es) |
| MC (1) | MC1850A1 (es) |
| MX (1) | MX8302A (es) |
| NO (1) | NO169125C (es) |
| NZ (1) | NZ221681A (es) |
| PH (1) | PH23930A (es) |
| PT (1) | PT85686B (es) |
| SK (1) | SK278990B6 (es) |
| ZA (1) | ZA876636B (es) |
| ZW (1) | ZW16387A1 (es) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2006248354B2 (en) * | 2005-05-19 | 2011-11-03 | Daiichi Sankyo Company, Limited | Tri- or tetra-substituted-3-aminopyrrolidine derivatives |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZW16387A1 (en) * | 1986-09-12 | 1988-05-25 | Hoffmann La Roche | Tricyclic compounds |
| US7977327B2 (en) | 2004-05-13 | 2011-07-12 | Daiichi Sankyo Company, Limited | Substituted pyrrolidine derivative |
| SI2383271T1 (sl) | 2006-03-13 | 2013-10-30 | Kyorin Pharmaceutical Co., Ltd. | Aminokinoloni kot inhibitorji gsk-3 |
| EP2203458B1 (en) | 2007-09-11 | 2011-11-02 | Kyorin Pharmaceutical Co., Ltd. | Cyanoaminoquinolones as gsk-3 inhibitors |
| KR101597841B1 (ko) | 2007-09-12 | 2016-02-26 | 교린 세이야꾸 가부시키 가이샤 | Gsk-3 억제제로서의 스피로시클릭 아미노퀴놀론 |
| FR2928150A1 (fr) * | 2008-02-29 | 2009-09-04 | Vetoquinol Sa Sa | Nouveaux derives 7-substitues de 3-carboxy-oxadiazino-quinolones, leur preparation et leur application comme anti-bacteriens |
| EP2145891A1 (en) * | 2008-07-09 | 2010-01-20 | Vetoquinol S.A. | 9-substituted-5-carboxy-oxadiazino-quinolone derivatives, their preparation and their application as anti-bacterials |
| US8071591B2 (en) | 2009-03-11 | 2011-12-06 | Kyorin Pharmaceutical Co., Ltd. | 7-cycloalkylaminoquinolones as GSK-3 inhibitors |
| CN107522718B (zh) * | 2017-09-14 | 2019-11-08 | 浙江国邦药业有限公司 | 一种马波沙星的合成方法 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZW16387A1 (en) * | 1986-09-12 | 1988-05-25 | Hoffmann La Roche | Tricyclic compounds |
-
1987
- 1987-08-28 ZW ZW163/87A patent/ZW16387A1/xx unknown
- 1987-09-04 ZA ZA876636A patent/ZA876636B/xx unknown
- 1987-09-04 NZ NZ221681A patent/NZ221681A/en unknown
- 1987-09-07 IL IL83814A patent/IL83814A/xx not_active IP Right Cessation
- 1987-09-07 AU AU78114/87A patent/AU602534B2/en not_active Expired
- 1987-09-09 HU HU874007A patent/HU199481B/hu unknown
- 1987-09-09 DZ DZ870149A patent/DZ1124A1/fr active
- 1987-09-10 MC MC871911A patent/MC1850A1/fr unknown
- 1987-09-11 PH PH35800A patent/PH23930A/en unknown
- 1987-09-11 SK SK6604-87A patent/SK278990B6/sk unknown
- 1987-09-11 FI FI873940A patent/FI86428C/fi not_active IP Right Cessation
- 1987-09-11 KR KR1019870010082A patent/KR960002857B1/ko not_active Expired - Lifetime
- 1987-09-11 NO NO873816A patent/NO169125C/no unknown
- 1987-09-11 PT PT85686A patent/PT85686B/pt unknown
- 1987-09-11 DK DK198704772A patent/DK173330B1/da not_active IP Right Cessation
- 1987-09-11 CZ CS876604A patent/CZ281195B6/cs not_active IP Right Cessation
- 1987-09-11 CA CA000546674A patent/CA1336905C/en not_active Expired - Lifetime
- 1987-09-11 IE IE244487A patent/IE61624B1/en not_active IP Right Cessation
- 1987-09-12 JP JP62227579A patent/JPH0696578B2/ja not_active Expired - Fee Related
- 1987-09-12 CN CN87106838A patent/CN1017800B/zh not_active Expired
- 1987-09-14 MX MX830287A patent/MX8302A/es unknown
- 1987-10-08 AT AT0263887A patent/AT389119B/de not_active IP Right Cessation
-
1994
- 1994-05-25 JP JP6133894A patent/JPH0826030B2/ja not_active Expired - Lifetime
- 1994-05-25 JP JP6133905A patent/JPH0819120B2/ja not_active Expired - Lifetime
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2006248354B2 (en) * | 2005-05-19 | 2011-11-03 | Daiichi Sankyo Company, Limited | Tri- or tetra-substituted-3-aminopyrrolidine derivatives |
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MKEX | Expiry |