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BRPI1009860A2 - composto, uso do mesmo, composição farmacêutica e método para tratamento terapêutico ou prevenção de doenças em humanos ou animais - Google Patents

composto, uso do mesmo, composição farmacêutica e método para tratamento terapêutico ou prevenção de doenças em humanos ou animais

Info

Publication number
BRPI1009860A2
BRPI1009860A2 BRPI1009860A BRPI1009860A BRPI1009860A2 BR PI1009860 A2 BRPI1009860 A2 BR PI1009860A2 BR PI1009860 A BRPI1009860 A BR PI1009860A BR PI1009860 A BRPI1009860 A BR PI1009860A BR PI1009860 A2 BRPI1009860 A2 BR PI1009860A2
Authority
BR
Brazil
Prior art keywords
humans
animals
disease
prevention
compound
Prior art date
Application number
BRPI1009860A
Other languages
English (en)
Inventor
Amaia Marcilla Etxnike
Daniel Horacio López
Gwendolyn Barceló Coblijn
María Laura Martín
Mónica Higuera Urbano
Pablo Vicente Escribá Ruiz
Rafael Álvarez Martínez
Silvia Terés Jiménez
Victoria Lladó Cañellas
Xavier Busquets Xaubet
Original Assignee
Lipopharma Therapeutics S L
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lipopharma Therapeutics S L filed Critical Lipopharma Therapeutics S L
Publication of BRPI1009860A2 publication Critical patent/BRPI1009860A2/pt
Publication of BRPI1009860A8 publication Critical patent/BRPI1009860A8/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • A61K31/202Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids having three or more double bonds, e.g. linolenic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40Unsaturated compounds
    • C07C59/42Unsaturated compounds containing hydroxy or O-metal groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • A61K31/201Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids having one or two double bonds, e.g. oleic, linoleic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/23Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/661Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BRPI1009860A 2009-03-16 2010-03-15 composto, uso do mesmo, composição farmacêutica e método para tratamento terapêutico ou prevenção de doenças em humanos ou animais BRPI1009860A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES200900725A ES2345241B1 (es) 2009-03-16 2009-03-16 Uso de 2-hidroxiderivados de acidos grasos poliinsaturados como medicamentos.
PCT/ES2010/070153 WO2010106211A1 (es) 2009-03-16 2010-03-15 Uso de derivados de ácidos grasos poliinsaturados como medicamentos

Publications (2)

Publication Number Publication Date
BRPI1009860A2 true BRPI1009860A2 (pt) 2016-03-08
BRPI1009860A8 BRPI1009860A8 (pt) 2019-12-17

Family

ID=42673244

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1009860A BRPI1009860A8 (pt) 2009-03-16 2010-03-15 composto, uso do mesmo, composição farmacêutica e método para tratamento terapêutico ou prevenção de doenças em humanos ou animais

Country Status (18)

Country Link
US (7) US9161928B2 (pt)
EP (2) EP3159329B1 (pt)
JP (1) JP5904592B2 (pt)
KR (4) KR102233102B1 (pt)
CN (4) CN102356057A (pt)
AU (6) AU2010224749B2 (pt)
BR (1) BRPI1009860A8 (pt)
CA (1) CA2754963C (pt)
CL (1) CL2011002268A1 (pt)
DK (2) DK2409963T3 (pt)
ES (3) ES2345241B1 (pt)
HU (2) HUE051850T2 (pt)
MX (1) MX2011009614A (pt)
PL (1) PL2409963T3 (pt)
PT (2) PT3159329T (pt)
RU (1) RU2513995C2 (pt)
SI (1) SI3159329T1 (pt)
WO (1) WO2010106211A1 (pt)

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Publication number Priority date Publication date Assignee Title
ES2345241B1 (es) * 2009-03-16 2011-09-08 Lipopharma Therapeutics Uso de 2-hidroxiderivados de acidos grasos poliinsaturados como medicamentos.
WO2011053870A1 (en) 2009-10-30 2011-05-05 Retrotope, Inc. Alleviating oxidative stress disorders with pufa derivatives
KR102014526B1 (ko) 2011-04-26 2019-08-26 레트로토프 인코포레이티드 Pufa 산화와 관련된 장애
CA2834342C (en) 2011-04-26 2021-08-31 Retrotope, Inc. Impaired energy processing disorders and mitochondrial deficiency
KR102110200B1 (ko) 2011-04-26 2020-05-13 레트로토프 인코포레이티드 산화성 망막 질환
AU2012249917B2 (en) * 2011-04-26 2017-06-15 Biojiva Llc Neurodegenerative disorders and muscle diseases implicating PUFAs
ES2401629B1 (es) * 2011-10-07 2014-03-04 Universitat De Les Illes Balears Enantiómeros de 2-hidroxiderivados de ácidos grasos y su uso como medicamentos.
EP3209637B1 (en) 2014-10-21 2019-05-08 Universitat de les Illes Balears 2-hydroxy-triacylglycerol compounds for use in treating disease
US20180024150A1 (en) * 2015-03-06 2018-01-25 Niigata University Biomarker of dementia with lewy bodies
JP7048976B2 (ja) 2015-11-23 2022-04-06 レトロトップ、 インコーポレイテッド 1,4-ジエン系の部位特異的同位体標識
GB201521085D0 (en) * 2015-11-30 2016-01-13 Biozep As Use
KR102569052B1 (ko) 2017-05-16 2023-08-22 어빌리티 파마슈티컬스 에스.엘. 암의 치료를 위한 약제학적 조합물
WO2019157516A1 (en) 2018-02-12 2019-08-15 resTORbio, Inc. Combination therapies
LT3813946T (lt) 2018-06-15 2024-07-10 Janssen Pharmaceutica Nv Rapamicino analogai ir jų panaudojimas
CN115209897A (zh) 2019-12-05 2022-10-18 安纳库利亚治疗公司 雷帕霉素类似物及其用途
ES2846824B2 (es) * 2020-01-29 2022-01-19 Univ Illes Balears Profarmacos de acidos grasos poliinsaturados y usos medicos de los mismos
US20230097753A1 (en) * 2020-01-29 2023-03-30 Universitat De Les Illes Balears Alpha-hydroxylated fatty-acid metabolites, medical uses and use as biomarkers
CA3163864A1 (en) 2020-02-10 2021-08-19 Ability Pharmaceuticals S.L. A pharmaceutical combination for the treatment of a cancer
IL295783B1 (en) 2020-02-21 2025-11-01 Retrotope Inc Processes for isotopic modification of polyunsaturated fatty acids and derivatives thereof
US12109194B2 (en) 2021-02-05 2024-10-08 Biojiva Llc Synergistic combination therapy for treating ALS

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GB2218984B (en) * 1988-05-27 1992-09-23 Renafield Limited Process for preparing high-concentration mixtures of polyunsaturated fatty acids & their esters and their prophylactic or therapeutic uses
JPH05974A (ja) * 1991-06-21 1993-01-08 Sagami Chem Res Center ハロゲン化不飽和アルキル化合物及びその前駆体
ES2161146B1 (es) * 1999-06-29 2002-07-01 Consejo Superior Investigacion Compuestos antimicrobianos, uso y metodo para inducir resistencia a infecciones de bacterias en plantas.
US6344574B1 (en) * 2000-07-20 2002-02-05 The United States Of America As Represented By The Secretary Of Agriculture Solvent fractionation of chicken fat for making lipid compositions enriched in unsaturated fatty acid-containing triacylglycerols
DE10106660A1 (de) * 2001-02-12 2002-08-29 Celanese Ventures Gmbh Verfahren zur Herstellung von gamma-Linolensäure aus einer Ciliaten-Kultur durch Zusatz geeigneter Vorläufermoleküle zu dem Kulturmedium
ES2186576B1 (es) * 2001-10-11 2004-09-16 Universitat De Les Illes Balears Acido 2-hidroxioleico para utilizar como medicamento.
DK2022775T3 (en) * 2002-04-01 2015-01-19 Univ Southern California polyunsaturated TRIHYDROXYEICOSANOIDER
US7135575B2 (en) * 2003-03-03 2006-11-14 Array Biopharma, Inc. P38 inhibitors and methods of use thereof
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CN101213281B (zh) * 2005-05-04 2013-03-13 普罗诺瓦生物医药挪威公司 新的dha衍生物及其作为药物的用途
JP2008540394A (ja) * 2005-05-04 2008-11-20 プロノヴァ バイオファーマ ノルゲ アクティーゼルスカブ 脂肪酸組成物、即ち、dha誘導体の医薬としての使用
US8059805B2 (en) * 2005-06-30 2011-11-15 Emc Corporation Enhanced services provided using communication redirection and processing
MX336435B (es) 2005-07-08 2016-01-19 Dsm Ip Assets Bv Acidos grasos poliinsaturados para el tratamiento de demencia y condiciones relacionadas con pre-demencia.
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PL1800675T4 (pl) * 2005-12-23 2012-02-29 Nutricia Nv Kompozycja zawierająca wielonienasycone kwasy tłuszczowe, białka, mangan, i/lub molibden oraz nukleozydy/nukleotydy do leczenia otępienia
BRPI0717883A2 (pt) 2006-11-01 2013-10-29 Pronova Biopharma Norge As Compostos lipídicos, composição contendo os mesmos e uso dos referidos compostos
WO2008053331A1 (en) 2006-11-01 2008-05-08 Pronova Biopharma Norge A/S Alpha-substituted omega-3 lipids that are activators or modulators of the peroxisome proliferators-activated receptor (ppar).
WO2008053340A1 (en) * 2006-11-03 2008-05-08 Pronova Biopharma Norge As A combination product comprising at least one lipid substituted in the alpha position and at least one hypoglycemic agent
US20080234377A1 (en) * 2007-03-23 2008-09-25 Martek Biosciences Corporation Polyunsaturated fatty acids for treatment of dementia and pre-dementia-related conditions
ES2345241B1 (es) 2009-03-16 2011-09-08 Lipopharma Therapeutics Uso de 2-hidroxiderivados de acidos grasos poliinsaturados como medicamentos.
ES2401629B1 (es) * 2011-10-07 2014-03-04 Universitat De Les Illes Balears Enantiómeros de 2-hidroxiderivados de ácidos grasos y su uso como medicamentos.

Also Published As

Publication number Publication date
AU2010224749A1 (en) 2011-10-13
AU2020205213A1 (en) 2020-07-30
AU2018203976A1 (en) 2018-06-21
AU2020205214A1 (en) 2020-07-30
US11253497B2 (en) 2022-02-22
RU2513995C2 (ru) 2014-04-27
ES2345241B1 (es) 2011-09-08
AU2010224749B2 (en) 2016-07-07
PT2409963T (pt) 2017-02-15
KR101833772B1 (ko) 2018-03-02
US20120108550A1 (en) 2012-05-03
US10201515B2 (en) 2019-02-12
KR102233102B1 (ko) 2021-03-26
RU2011141850A (ru) 2013-04-27
US20200352891A1 (en) 2020-11-12
AU2019226257A1 (en) 2019-09-26
PL2409963T3 (pl) 2017-05-31
US20190365690A1 (en) 2019-12-05
AU2019226257B2 (en) 2020-05-07
CN106420686B (zh) 2020-05-22
KR20110137365A (ko) 2011-12-22
US9907772B2 (en) 2018-03-06
US20180085332A1 (en) 2018-03-29
KR20180021931A (ko) 2018-03-05
US20160158181A1 (en) 2016-06-09
HUE051850T2 (hu) 2021-03-29
MX2011009614A (es) 2012-01-20
HUE032027T2 (en) 2017-08-28
AU2016238970B2 (en) 2018-03-08
EP2409963B1 (en) 2017-01-04
HK1232207A1 (zh) 2018-01-05
ES2820025T3 (es) 2021-04-19
JP2012520344A (ja) 2012-09-06
CN106349058B (zh) 2020-01-14
CA2754963A1 (en) 2010-09-23
DK2409963T3 (en) 2017-02-27
ES2613606T3 (es) 2017-05-24
AU2016238970A1 (en) 2016-11-03
EP2409963A4 (en) 2013-10-02
JP5904592B2 (ja) 2016-04-13
CN109999018A (zh) 2019-07-12
US20170035720A1 (en) 2017-02-09
AU2020205214B2 (en) 2021-02-18
KR20200024953A (ko) 2020-03-09
CA2754963C (en) 2022-02-08
CL2011002268A1 (es) 2012-01-27
EP3159329B1 (en) 2020-08-12
US20160158180A1 (en) 2016-06-09
CN106420686A (zh) 2017-02-22
EP3159329A1 (en) 2017-04-26
WO2010106211A1 (es) 2010-09-23
CN106349058A (zh) 2017-01-25
EP2409963A1 (en) 2012-01-25
US9763907B2 (en) 2017-09-19
PT3159329T (pt) 2020-11-13
AU2020205213B2 (en) 2021-02-25
US9763906B2 (en) 2017-09-19
KR20190018754A (ko) 2019-02-25
CN102356057A (zh) 2012-02-15
US9161928B2 (en) 2015-10-20
BRPI1009860A8 (pt) 2019-12-17
AU2018203976B2 (en) 2019-06-06
SI3159329T1 (sl) 2021-01-29
ES2345241A1 (es) 2010-09-17
DK3159329T3 (da) 2020-11-09

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06T Formal requirements before examination [chapter 6.20 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B12B Appeal against refusal [chapter 12.2 patent gazette]