BRPI0819914A2 - método para tratar uma doença, uso de um composto e seus sais farmaceuticamente aceitáveis, e, composto. - Google Patents
método para tratar uma doença, uso de um composto e seus sais farmaceuticamente aceitáveis, e, composto.Info
- Publication number
- BRPI0819914A2 BRPI0819914A2 BRPI0819914A BRPI0819914A BRPI0819914A2 BR PI0819914 A2 BRPI0819914 A2 BR PI0819914A2 BR PI0819914 A BRPI0819914 A BR PI0819914A BR PI0819914 A BRPI0819914 A BR PI0819914A BR PI0819914 A2 BRPI0819914 A2 BR PI0819914A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- disease
- treating
- pharmaceutically acceptable
- acceptable salts
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 2
- 201000010099 disease Diseases 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/451—Non condensed piperidines, e.g. piperocaine having a carbocyclic group directly attached to the heterocyclic ring, e.g. glutethimide, meperidine, loperamide, phencyclidine, piminodine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Psychology (AREA)
- Addiction (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Pulmonology (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200701791 | 2007-12-14 | ||
| DKPA200701798 | 2007-12-17 | ||
| PCT/DK2008/050302 WO2009076962A1 (en) | 2007-12-14 | 2008-12-11 | Therapeutic uses of compounds having affinity to the serotonin transporter, serotonin receptors and noradrenalin transporter |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0819914A2 true BRPI0819914A2 (pt) | 2016-05-17 |
Family
ID=40285887
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0819914A BRPI0819914A2 (pt) | 2007-12-14 | 2008-12-11 | método para tratar uma doença, uso de um composto e seus sais farmaceuticamente aceitáveis, e, composto. |
Country Status (18)
| Country | Link |
|---|---|
| US (3) | US20110053978A1 (pt) |
| EP (1) | EP2231154A1 (pt) |
| JP (1) | JP2011506353A (pt) |
| KR (1) | KR20100092956A (pt) |
| CN (1) | CN102202666A (pt) |
| AR (1) | AR069904A1 (pt) |
| AU (1) | AU2008338059A1 (pt) |
| BR (1) | BRPI0819914A2 (pt) |
| CA (1) | CA2708786A1 (pt) |
| CL (1) | CL2008003709A1 (pt) |
| CO (1) | CO6290669A2 (pt) |
| EA (1) | EA201070737A1 (pt) |
| IL (1) | IL205965A0 (pt) |
| MX (1) | MX2010005795A (pt) |
| NZ (1) | NZ586010A (pt) |
| SG (1) | SG185984A1 (pt) |
| TW (1) | TW200938194A (pt) |
| WO (1) | WO2009076962A1 (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE540941T1 (de) | 2006-06-16 | 2012-01-15 | Lundbeck & Co As H | 1-ä2-(2,4-dimethylphenylsulfanyl)phenylüpiperaz n als verbindung mit kombinierter serotoninwiederaufnahme-, 5-ht3- und 5-ht1a- aktivität zur behandlung kognitiver störungen |
| TWI432194B (zh) * | 2007-03-20 | 2014-04-01 | Lundbeck & Co As H | 4-〔2-(4-甲基苯硫基)苯基〕哌啶之新穎治療用途 |
| GEP20166487B (en) * | 2010-04-30 | 2016-06-10 | Takeda Pharmaceutical | Enteric tablet |
| CN104710345B (zh) * | 2013-12-17 | 2017-09-05 | 江苏恩华药业股份有限公司 | 用于制备4‑(2‑(4‑甲基苯基硫基))苯基哌啶的化合物、其制备方法及应用 |
| CN104120177A (zh) * | 2014-06-11 | 2014-10-29 | 杭州艾迪康医学检验中心有限公司 | 检测5-httlpr片段多态性的方法和引物 |
| WO2019008484A1 (en) * | 2017-07-03 | 2019-01-10 | Suven Life Sciences Limited | NEW USES OF A PURE 5-HT6 RECEPTOR ANTAGONIST |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA81749C2 (uk) * | 2001-10-04 | 2008-02-11 | Х. Луннбек А/С | Фенілпіперазинові похідні як інгібітори зворотного захоплення серотоніну |
| DK1626720T3 (da) * | 2003-04-04 | 2008-12-01 | Lundbeck & Co As H | 4-(2-Phenylsulfanyl-phenyl)-piperidinderivater som serotonin-genoptagelseshæmmer |
| CA2656057C (en) * | 2006-06-16 | 2012-10-02 | H. Lundbeck A/S | Crystalline forms of 4-[2-(4-methylphenylsulfanyl)-phenyl]piperidine with combined serotonin and norepinephrine reuptake inhibition for the treatment of neuropathic pain |
| TWI432194B (zh) * | 2007-03-20 | 2014-04-01 | Lundbeck & Co As H | 4-〔2-(4-甲基苯硫基)苯基〕哌啶之新穎治療用途 |
| HRP20140044T1 (hr) * | 2007-06-15 | 2014-02-14 | H. Lundbeck A/S | 4-[2-(4-metilfenilsulfanil)fenil]piperidin za lijeäśenje iritabilnog sindroma crijeva (ibs) |
-
2008
- 2008-12-02 TW TW097146699A patent/TW200938194A/zh unknown
- 2008-12-11 CA CA2708786A patent/CA2708786A1/en not_active Abandoned
- 2008-12-11 CN CN2008801203913A patent/CN102202666A/zh active Pending
- 2008-12-11 MX MX2010005795A patent/MX2010005795A/es not_active Application Discontinuation
- 2008-12-11 BR BRPI0819914A patent/BRPI0819914A2/pt not_active IP Right Cessation
- 2008-12-11 US US12/747,403 patent/US20110053978A1/en not_active Abandoned
- 2008-12-11 AU AU2008338059A patent/AU2008338059A1/en not_active Abandoned
- 2008-12-11 KR KR1020107013095A patent/KR20100092956A/ko not_active Withdrawn
- 2008-12-11 WO PCT/DK2008/050302 patent/WO2009076962A1/en not_active Ceased
- 2008-12-11 EP EP08862439A patent/EP2231154A1/en not_active Withdrawn
- 2008-12-11 EA EA201070737A patent/EA201070737A1/ru unknown
- 2008-12-11 JP JP2010537257A patent/JP2011506353A/ja active Pending
- 2008-12-11 SG SG2012083010A patent/SG185984A1/en unknown
- 2008-12-11 NZ NZ586010A patent/NZ586010A/xx not_active IP Right Cessation
- 2008-12-12 CL CL2008003709A patent/CL2008003709A1/es unknown
- 2008-12-12 AR ARP080105414A patent/AR069904A1/es not_active Application Discontinuation
-
2010
- 2010-05-25 IL IL205965A patent/IL205965A0/en unknown
- 2010-06-11 CO CO10070917A patent/CO6290669A2/es not_active Application Discontinuation
-
2014
- 2014-05-16 US US14/279,504 patent/US20140296290A1/en not_active Abandoned
-
2016
- 2016-05-03 US US15/145,102 patent/US20170087138A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009076962A1 (en) | 2009-06-25 |
| NZ586010A (en) | 2012-08-31 |
| US20110053978A1 (en) | 2011-03-03 |
| JP2011506353A (ja) | 2011-03-03 |
| US20140296290A1 (en) | 2014-10-02 |
| CO6290669A2 (es) | 2011-06-20 |
| TW200938194A (en) | 2009-09-16 |
| CA2708786A1 (en) | 2009-06-25 |
| CL2008003709A1 (es) | 2010-01-15 |
| EP2231154A1 (en) | 2010-09-29 |
| AU2008338059A1 (en) | 2009-06-25 |
| US20170087138A1 (en) | 2017-03-30 |
| SG185984A1 (en) | 2012-12-28 |
| IL205965A0 (en) | 2010-11-30 |
| AR069904A1 (es) | 2010-03-03 |
| MX2010005795A (es) | 2010-08-31 |
| EA201070737A1 (ru) | 2010-12-30 |
| KR20100092956A (ko) | 2010-08-23 |
| CN102202666A (zh) | 2011-09-28 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO2025029I1 (no) | Entrectinib or isomers, tautomers, or pharmaceutically acceptable salts therof - forlenget | |
| BRPI0814688A2 (pt) | composto, uso de um composto, métodos para produzir um efeito antiproliferativo em um animal de sangue quente, e para tratar doenças, e, composição farmacêutica | |
| BR112012003578A2 (pt) | composto, sal farmaceuticamente aceitável, sal de sulfato, composição farmacêutica, método para tratar uma infecção viral, e, uso de um composto ou sal. | |
| BRPI0821274A2 (pt) | composto ou um sal, ou pró-droga farmaceuticamente aceitável do mesmo, uso do mesmo, método para tratar uma doença em um animal de sangue quente, e, composição farmacêutica | |
| BRPI0912539A2 (pt) | composto, composição farmacêutica , método para tratar uma doença, e, uso do composto. | |
| BRPI0910734A2 (pt) | composto, composição farmacêutica, e, processo para preparar um composto ou um sal farmaceuticamente aceitável do mesmo. | |
| BRPI0917705A2 (pt) | composto, pró-droga, composição farmacêutica, método para tratar ou prevenir uma doença ou condição, e, uso do composto | |
| BRPI0815057A2 (pt) | Composto, composição farmacêutica, e, método para tratar infecção. | |
| BRPI0819799A2 (pt) | Composto, intermediário, uso de um composto, composição farmacêutica, e, método para prevenir, tratar ou melhorar uma doença | |
| BRPI0917458A2 (pt) | composto, método de tratamento de doenças e condições, composição farmacêutica, método para tratar ou prevenir doença, e, uso de um composto | |
| BRPI0907976A2 (pt) | Composto, composição farmacêutica, uso de um composto, e, método para tratar ou prevenir doenças | |
| BRPI0818244A2 (pt) | Composto, composição farmacêutica, uso de um composto, e, método para tratamento de um distúrbio ou doença | |
| BRPI0814503A2 (pt) | composto, uso de um composto, métodos para produzir um efeito anti-proliferativo em um animal de sangue quente, e para tratar uma doença, e, composição farmacêutica | |
| BRPI0922475A2 (pt) | composto, composição farmacêutica , método para tratar câncer, e, uso de um composto. | |
| BRPI0819218A2 (pt) | Métodos, estojos e composições para administração de compostos farmacêuticos | |
| BRPI0815894A2 (pt) | Composição farmacêutica, uso da mesma, e, sais farmaceuticamente aceitáveis de um composto. | |
| BR122020011920A2 (pt) | composto, composição farmacêutica, método para tratar uma doença, uso de um composto, e processos para a preparação de um composto, e para a fabricação de um composto | |
| BRPI0922566A2 (pt) | polimorfo cristalino, composição farmacêutica, composto, e, métodos para preparar um composto, e para tratar uma doença. | |
| BRPI0911685A2 (pt) | composto, método para o tratamento de uma doença, uso de um composto, composição farmacêutica, e, kit | |
| BRPI0818193A2 (pt) | composto, sal farmacêuticamente aceitável de um composto, composição farmacêutica, e, uso de um composto | |
| BRPI0912348A2 (pt) | composto de 3-aminocarbazol, composição farmacêutica, método para preparar um composto de 3-aminocarbazol, uso de um composto de 3-aminocarbazol, e, método para tratar ou prevenir doenças | |
| BR112012003280A2 (pt) | composição farmacêutica para administração oral, método para tratar uma doença, uso do composto, e, composto. | |
| BRPI1013984A2 (pt) | composto , composição farmacêutica, método para tratamento ou profilaxia de uma doença ou condição, e, uso de um composto. | |
| BRPI0820474A2 (pt) | método de tratamento de uma doença, uso de composto, e, composto | |
| BRPI0816881A2 (pt) | Composto, composição farmacêutica, uso de um composto, e, métodos para tratar doenças ou distúrbios e para preparar um composto. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 6A E 7A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2372 DE 21-06-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |