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BRPI0512108A - antibióticos contendo complexos de ácido borìnico e métodos de uso - Google Patents

antibióticos contendo complexos de ácido borìnico e métodos de uso

Info

Publication number
BRPI0512108A
BRPI0512108A BRPI0512108-6A BRPI0512108A BRPI0512108A BR PI0512108 A BRPI0512108 A BR PI0512108A BR PI0512108 A BRPI0512108 A BR PI0512108A BR PI0512108 A BRPI0512108 A BR PI0512108A
Authority
BR
Brazil
Prior art keywords
methods
antibiotics
acid complexes
boronic acid
containing boronic
Prior art date
Application number
BRPI0512108-6A
Other languages
English (en)
Inventor
Ving Lee
Stephen J Benkovic
Stephen J Baker
Kirk R Maples
Tsutomu Akama
Rajeshwar Singh
Vittorio Sauro
Chetan Pandit
Zhuoyi Su
Zhixiang Yang
Yong-Kang Zhang
Original Assignee
Anacor Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anacor Pharmaceuticals Inc filed Critical Anacor Pharmaceuticals Inc
Publication of BRPI0512108A publication Critical patent/BRPI0512108A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/69—Boron compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/04—Esters of boric acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

ANTIBIóTICOS CONTENDO COMPLEXOS DE áCIDO BORìNICO E MéTODOS E USO A estrutura e preparação de antibióticos que incorporam complexos de ácido borínico são reveladas, especialmente derivados de hidroxiquinolina, imidazol e ácido picolínico, juntamente com composições desses antibióticos e métodos de utilização dos antibióticos e composições como agentes bactericidas e fungicidas, bem como agentes terapêuticos para o tratamento de doenças causadas por bactérias e fungos.
BRPI0512108-6A 2004-06-14 2005-06-14 antibióticos contendo complexos de ácido borìnico e métodos de uso BRPI0512108A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/867,465 US7390806B2 (en) 2002-12-18 2004-06-14 Antibiotics containing borinic acid complexes and methods of use
PCT/US2005/021214 WO2006007384A2 (en) 2004-06-14 2005-06-14 Antibiotics containing borinic acid complexes and methods of use

Publications (1)

Publication Number Publication Date
BRPI0512108A true BRPI0512108A (pt) 2008-02-06

Family

ID=35415124

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0512108-6A BRPI0512108A (pt) 2004-06-14 2005-06-14 antibióticos contendo complexos de ácido borìnico e métodos de uso

Country Status (13)

Country Link
US (2) US7390806B2 (pt)
EP (1) EP1765359A2 (pt)
JP (1) JP2008502701A (pt)
KR (1) KR20070026783A (pt)
CN (1) CN1972694A (pt)
AU (1) AU2005262536A1 (pt)
BR (1) BRPI0512108A (pt)
CA (1) CA2570591A1 (pt)
IL (1) IL179748A0 (pt)
MX (1) MXPA06014418A (pt)
RU (1) RU2007101284A (pt)
TW (2) TW200938195A (pt)
WO (1) WO2006007384A2 (pt)

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US7390806B2 (en) * 2002-12-18 2008-06-24 Anacor Pharmaceuticals, Inc. Antibiotics containing borinic acid complexes and methods of use
FR2864083B1 (fr) * 2003-12-18 2007-04-13 Galderma Res & Dev Nouveaux derives d'acides phenyl-boroniques et leurs procedes de preparation.
AR049916A1 (es) * 2004-06-14 2006-09-13 Anacor Pharmaceuticals Inc Usos anti-parasitarios de complejos de acido borinico
ZA200707408B (en) 2005-02-16 2009-11-25 Anacor Pharmaceuticals Inc Boron-containing small molecules
EP1965647A2 (en) * 2005-12-28 2008-09-10 Anacor Pharmaceuticals, Inc. Process for manufacturing picolinate borinic esters
JP2009526751A (ja) 2005-12-30 2009-07-23 アナコール ファーマシューティカルズ，インコーポレイテッド ホウ素含有小分子
CA2642583C (en) 2006-02-16 2016-08-23 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-inflammatory agents
US20070286822A1 (en) * 2006-06-12 2007-12-13 Anacor Pharmaceuticals Inc. Compounds for the Treatment of Periodontal Disease
MX2008015918A (es) * 2006-06-12 2009-01-14 Anacor Pharmaceuticals Inc Compuestos para el tratamiento de enfermedad periodontal.
JO3598B1 (ar) 2006-10-10 2020-07-05 Infinity Discovery Inc الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني
EP2564857B1 (en) 2008-03-06 2017-05-03 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-inflammatory agents
JP5637982B2 (ja) 2008-04-09 2014-12-10 インフィニティー ファーマシューティカルズ， インコーポレイテッド 脂肪酸アミド加水分解酵素の阻害剤
WO2009140309A2 (en) * 2008-05-12 2009-11-19 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2010027975A1 (en) * 2008-09-04 2010-03-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US8461336B2 (en) 2008-09-04 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2010045503A1 (en) * 2008-10-15 2010-04-22 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agents
MX2011006334A (es) * 2008-12-17 2011-09-22 Anacor Pharmaceuticals Inc Polimorfos de (s)-3-amino-metil-7-(3-hidroxi-propoxi)-3h-benzo-[c] [1,2]-oxaborol-1-ol.
AU2010234445A1 (en) 2009-04-07 2011-11-03 Infinity Pharmaceuticals, Inc. Inhibitors of fatty acid amide hydrolase
US8541581B2 (en) 2009-04-07 2013-09-24 Infinity Pharmaceuticals, Inc. Inhibitors of fatty acid amide hydrolase
TW201110996A (en) 2009-06-03 2011-04-01 Colgate Palmolive Co Borinic compositions
AU2010281439A1 (en) * 2009-07-28 2012-03-15 Anacor Pharmaceuticals, Inc. Trisubstituted boron-containing molecules
AP4039A (en) 2009-08-14 2017-02-28 Daitao Chen Boron-containing small molecules as antiprotozoal agents
US20110207701A1 (en) * 2009-08-19 2011-08-25 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US20110124597A1 (en) * 2009-09-25 2011-05-26 Anacor Pharmaceuticals, Inc. Boron containing small molecules
WO2011049971A1 (en) 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
WO2011060199A1 (en) * 2009-11-11 2011-05-19 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US8716478B2 (en) 2010-01-27 2014-05-06 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011097233A1 (en) 2010-02-03 2011-08-11 Infinity Pharmaceuticals, Inc. Fatty acid amide hydrolase inhibitors
US8623911B2 (en) 2010-03-19 2014-01-07 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agent
EP2613788B1 (en) 2010-09-07 2017-06-21 Anacor Pharmaceuticals, Inc. Benzoxaborole derivatives for treating bacterial infections
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
US9585396B2 (en) 2013-01-30 2017-03-07 Agrofresh Inc. Volatile applications against pathogens
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
US8669207B1 (en) 2013-01-30 2014-03-11 Dow Agrosciences, Llc. Compounds and compositions
UA116557C2 (uk) 2013-01-30 2018-04-10 Доу Агросайенсіс Ллс Спосіб застосування бензоксаборолів як летких антимікробних сполук проти патогенів, що уражають м'якоть плодів, рослини або частини рослин
KR101636431B1 (ko) 2013-07-30 2016-07-05 동아에스티 주식회사 트리사이클릭 벤즈옥사보롤 화합물, 이의 제조방법 및 용도
KR101756785B1 (ko) * 2015-03-10 2017-07-12 한국화학연구원 4배위 유기 붕소 화합물의 제조방법
WO2017155879A1 (en) 2016-03-07 2017-09-14 Agrofresh Inc. Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops
CA3054138A1 (en) * 2017-03-09 2018-09-13 The Penn State Research Foundation Boron-containing small molecules for inhibiting activity of a receptor-like protein tyrosine phosphatase
US10526343B2 (en) 2018-03-26 2020-01-07 University Of Sharjah Heterocyclic systems and pharmaceutical applications thereof
CN111995634B (zh) * 2020-08-28 2022-08-05 深圳大学 一种四配位有机硼化合物、荧光探针及其制备方法与应用
US20230340530A1 (en) 2020-08-31 2023-10-26 Pfizer Inc. Methods of Protecting RNA

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US5348948A (en) * 1993-05-07 1994-09-20 American Cyanamid Company 2,2-diaryl-1-(oxa and thia)-2a-azonia-2-borataacenaphthene fungicidal
US5348947A (en) * 1993-05-07 1994-09-20 American Cyanamid Company Diarylboron ester and thioester fungicidal agents
WO2000044387A1 (fr) * 1999-01-29 2000-08-03 Nitto Kasei Co., Ltd. Composes organobores presentant une activite de coccidiostats
AU774404C (en) 1999-05-25 2005-06-30 Board Of Trustees Of The Leland Stanford Junior University DNA methyltransferase inhibitors
CN1325504C (zh) 2002-01-10 2007-07-11 宾夕法尼亚州研究基金会 制备二芳基硼酸烷基酯和络合的二芳基硼酸的方法
US20040007657A1 (en) 2002-07-08 2004-01-15 Mcenroe John D. Casting form for a cast-in-place structural element and fencing system including cast-in-place structural elements
US7390806B2 (en) 2002-12-18 2008-06-24 Anacor Pharmaceuticals, Inc. Antibiotics containing borinic acid complexes and methods of use
MXPA05006685A (es) 2002-12-18 2005-12-14 Anacor Pharmaceuticals Inc Antibioticos que contienen complejos de acido borinico y metodos de uso.

Also Published As

Publication number Publication date
US20050070503A1 (en) 2005-03-31
WO2006007384A3 (en) 2006-04-06
RU2007101284A (ru) 2008-07-20
WO2006007384B1 (en) 2006-08-17
MXPA06014418A (es) 2007-03-08
US7888356B2 (en) 2011-02-15
CN1972694A (zh) 2007-05-30
CA2570591A1 (en) 2006-01-19
TW200938195A (en) 2009-09-16
JP2008502701A (ja) 2008-01-31
TW200612939A (en) 2006-05-01
US7390806B2 (en) 2008-06-24
US20080293675A1 (en) 2008-11-27
EP1765359A2 (en) 2007-03-28
IL179748A0 (en) 2007-05-15
KR20070026783A (ko) 2007-03-08
AU2005262536A1 (en) 2006-01-19
WO2006007384A2 (en) 2006-01-19

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012.