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BRPI0416909A - método de tratamento de aterosclerose - Google Patents

método de tratamento de aterosclerose

Info

Publication number
BRPI0416909A
BRPI0416909A BRPI0416909-3A BRPI0416909A BRPI0416909A BR PI0416909 A BRPI0416909 A BR PI0416909A BR PI0416909 A BRPI0416909 A BR PI0416909A BR PI0416909 A BRPI0416909 A BR PI0416909A
Authority
BR
Brazil
Prior art keywords
treatment method
atherosclerosis treatment
atherosclerosis
mammal
administering
Prior art date
Application number
BRPI0416909-3A
Other languages
English (en)
Inventor
Paul Steven Changelian
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of BRPI0416909A publication Critical patent/BRPI0416909A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

"MéTODO DE TRATAMENTO DE ATEROSCLEROSE". A presente invenção refere-se a um método de tratamento ou prevenção de aterosclerose compreendendo a administração ao referido mamífero de uma quantidade de um composto da fórmula em que R¬ 1¬, R¬ 2¬ e R¬ 3¬ São conforme acima definidos.
BRPI0416909-3A 2003-11-25 2004-11-15 método de tratamento de aterosclerose BRPI0416909A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US52549603P 2003-11-25 2003-11-25
PCT/IB2004/003788 WO2005051393A1 (en) 2003-11-25 2004-11-15 Method of treatment of atherosclerosis

Publications (1)

Publication Number Publication Date
BRPI0416909A true BRPI0416909A (pt) 2007-01-16

Family

ID=34632985

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0416909-3A BRPI0416909A (pt) 2003-11-25 2004-11-15 método de tratamento de aterosclerose

Country Status (9)

Country Link
US (1) US20050113395A1 (pt)
EP (1) EP1689407A1 (pt)
JP (1) JP2007512316A (pt)
AR (1) AR046660A1 (pt)
BR (1) BRPI0416909A (pt)
CA (1) CA2545192A1 (pt)
MX (1) MXPA06005882A (pt)
TW (1) TW200528109A (pt)
WO (1) WO2005051393A1 (pt)

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US9193733B2 (en) 2012-05-18 2015-11-24 Incyte Holdings Corporation Piperidinylcyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as JAK inhibitors
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Also Published As

Publication number Publication date
JP2007512316A (ja) 2007-05-17
CA2545192A1 (en) 2005-06-09
WO2005051393A1 (en) 2005-06-09
AR046660A1 (es) 2005-12-14
TW200528109A (en) 2005-09-01
MXPA06005882A (es) 2006-06-27
US20050113395A1 (en) 2005-05-26
EP1689407A1 (en) 2006-08-16

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Legal Events

Date Code Title Description
B08F Application fees: application dismissed [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A, 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012.