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BRPI0406875A - Derivados de monossacarìdeo de avermectina tendo propriedades pesticidas - Google Patents

Derivados de monossacarìdeo de avermectina tendo propriedades pesticidas

Info

Publication number
BRPI0406875A
BRPI0406875A BR0406875-0A BRPI0406875A BRPI0406875A BR PI0406875 A BRPI0406875 A BR PI0406875A BR PI0406875 A BRPI0406875 A BR PI0406875A BR PI0406875 A BRPI0406875 A BR PI0406875A
Authority
BR
Brazil
Prior art keywords
monosaccharide derivatives
compounds
pesticidal properties
avermectin monosaccharide
formula
Prior art date
Application number
BR0406875-0A
Other languages
English (en)
Inventor
Thomas Pitterna
Peter Maienfisch
Fiona Nurphy Kessabi
Hans Tobler
Jerome Cassayre
Laura Quaranta
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of BRPI0406875A publication Critical patent/BRPI0406875A/pt
Publication of BRPI0406875B1 publication Critical patent/BRPI0406875B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

"DERIVADOS DE MONOSSACARìDEO DE AVERMECTINA TENDO PROPRIEDADES PESTICIDAS". A presente invenção refere-se a um composto da fórmula geral (I), composições pesticidas cujo composto ativo é selecionado destes compostos e seus tautómeros; intermediários para a preparação dos referidos compostos da fórmula (I), métodos para a preparação dos compostos da fórmula (I), e um método para controlar pestes empregando-se estas composições.
BRPI0406875-0A 2003-01-31 2004-01-30 Derivados de monossacarídeo de avermectina tendo propriedades pesticidas BRPI0406875B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0302309.0 2003-01-31
GBGB0302309.0A GB0302309D0 (en) 2003-01-31 2003-01-31 Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
PCT/EP2004/000899 WO2004067534A1 (en) 2003-01-31 2004-01-30 Avermectin monosaccharide derivatives having pesticidal properties

Publications (2)

Publication Number Publication Date
BRPI0406875A true BRPI0406875A (pt) 2006-01-03
BRPI0406875B1 BRPI0406875B1 (pt) 2014-05-27

Family

ID=9952240

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0406875-0A BRPI0406875B1 (pt) 2003-01-31 2004-01-30 Derivados de monossacarídeo de avermectina tendo propriedades pesticidas

Country Status (28)

Country Link
US (1) US20060205595A1 (pt)
EP (1) EP1594878B1 (pt)
JP (1) JP2006518347A (pt)
KR (1) KR20050097524A (pt)
CN (1) CN100410259C (pt)
AR (1) AR042967A1 (pt)
AT (1) ATE397610T1 (pt)
AU (1) AU2004207073B2 (pt)
BR (1) BRPI0406875B1 (pt)
CA (1) CA2513573C (pt)
CL (1) CL2004000147A1 (pt)
CY (1) CY1108295T1 (pt)
DE (1) DE602004014252D1 (pt)
DK (1) DK1594878T3 (pt)
ES (1) ES2308140T3 (pt)
GB (1) GB0302309D0 (pt)
IL (1) IL169598A (pt)
MA (1) MA27587A1 (pt)
MX (1) MXPA05007923A (pt)
NZ (1) NZ541252A (pt)
PL (1) PL218731B1 (pt)
PT (1) PT1594878E (pt)
RU (1) RU2329268C2 (pt)
SI (1) SI1594878T1 (pt)
TW (1) TW200508240A (pt)
UA (1) UA81012C2 (pt)
WO (1) WO2004067534A1 (pt)
ZA (1) ZA200505545B (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
AR040073A1 (es) 2002-05-07 2005-03-16 Syngenta Participations Ag Derivados de 4''-desoxi-4''-(s)-amido avermectina y su uso como plaguicidas
GB0302310D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302547D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
GB0320176D0 (en) 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively
RU2566189C2 (ru) * 2010-08-26 2015-10-20 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Пестицидные композиции
CN103214532B (zh) * 2013-02-28 2018-07-06 河北威远生物化工有限公司 阿维菌素B2a/2b胺基衍生物、衍生物盐和阿维菌素B2a/2b胺基衍生物盐的制备方法及用途
CN103613625B (zh) * 2013-12-02 2016-03-02 兰州大学 一种阿维菌素类化合物及其制备方法和在农药中的用途
CN104402953B (zh) * 2014-11-28 2017-07-28 大庆志飞生物化工有限公司 阿维菌素单糖化合物及其制备方法和用途
CN104402954A (zh) * 2014-11-28 2015-03-11 大庆志飞生物化工有限公司 甲胺基阿维菌素单糖化合物及其制备方法和用途
CN107501368B (zh) * 2017-09-30 2020-02-21 中国科学院成都生物研究所 一种多拉菌素衍生物的合成及其杀虫应用
CN108690108B (zh) * 2018-07-27 2022-03-11 河北威远生物化工有限公司 一种磺酰胺基取代的阿维菌素B2a/B2b衍生物及其制备方法与应用
CN113150053B (zh) * 2020-01-22 2024-10-01 华东理工大学 偶氮苯类阿维菌素衍生物及其制备方法和应用

Family Cites Families (33)

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Publication number Priority date Publication date Assignee Title
US4206205A (en) * 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
US4203976A (en) * 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4427663A (en) * 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4622313A (en) * 1985-08-01 1986-11-11 Merck & Co., Inc. O-sulfate derivatives of avermectins and milbemycins having improved water solubility
US4886828A (en) * 1986-09-12 1989-12-12 American Cyanamid Company Δ22 -derivatives of LL-F28249 compounds
US4831016A (en) * 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives
US4895837A (en) * 1988-01-29 1990-01-23 Merck & Co., Inc. Avermectin derivatives
NZ228866A (en) * 1988-05-02 1991-10-25 Merck & Co Inc Fluoro-substituted milbemycins and avermectins for combatting parasites and insects
US5008250A (en) * 1988-05-25 1991-04-16 Merck & Co., Inc. Avermectins with a cleaved furan ring and an 8a hydroxy group
GB2220856A (en) * 1988-07-18 1990-01-24 Merck & Co Inc Novel synergistic agricultural insecticidal and acaricidal combinations containing avermectin derivatives
NZ231773A (en) * 1988-12-23 1992-09-25 Merck & Co Inc Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof
FR2646237B1 (fr) * 1989-04-21 1994-01-07 Fabrication Instruments Mesure Dispositif de jaugeage de gaz haute pression, en particulier pour la reserve d'oxygene gazeux embarquee a bord d'un avion
US5057499A (en) * 1989-06-02 1991-10-15 Merck & Co. Inc. Avermectin derivatives
US5023241A (en) * 1989-07-31 1991-06-11 Merck & Co., Inc. Avermectin derivatives
US5169839A (en) * 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
US5192546A (en) * 1991-01-15 1993-03-09 Mycogen Corporation Synergistic pesticidal compositions
US5346698A (en) * 1991-01-15 1994-09-13 Mycogen Corporation Synergistic pesticidal compositions
US5208222A (en) * 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
GB9201505D0 (en) * 1992-01-24 1992-03-11 Pfizer Ltd Antiparasitic agents
US5229415A (en) * 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
US5362863A (en) * 1993-09-29 1994-11-08 Merck & Co., Inc. Process for the preparation of 4"-amino avermectin compounds
US5981500A (en) * 1994-01-12 1999-11-09 Pfizer Inc. Antiparasitic agents related to the milbemycins and avermectins
US5436355A (en) * 1994-02-03 1995-07-25 Merck & Co., Inc. Process for making avermectin/zein compositions
TW327125B (en) * 1994-02-07 1998-02-21 Merck & Co Inc Composition and method for protecting against pine exhausted
US6875727B2 (en) * 1997-12-23 2005-04-05 Syngenta Crop Protection, Inc. Use of macrolides in pest control
KR20010101819A (ko) * 1999-02-09 2001-11-14 오무라 사토시 에바멕틴 유도체
JPWO2002012248A1 (ja) * 2000-08-09 2004-01-15 社団法人北里研究所 エバーメクチン誘導体
EG23124A (en) * 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
CR6574A (es) * 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
TW200301079A (en) * 2001-12-21 2003-07-01 Syngenta Participations Ag Avermectin B1 derivatives having an aminosulfonyloxy substituent in the 4"-position
GB0302308D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302548D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins substituted in the 4"- and 4' -positions having pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively

Also Published As

Publication number Publication date
UA81012C2 (en) 2007-11-26
KR20050097524A (ko) 2005-10-07
RU2005127321A (ru) 2006-01-27
WO2004067534A1 (en) 2004-08-12
MA27587A1 (fr) 2005-10-03
AU2004207073A1 (en) 2004-08-12
PL218731B1 (pl) 2015-01-30
MXPA05007923A (es) 2005-09-30
ZA200505545B (en) 2006-04-26
CL2004000147A1 (es) 2005-03-04
EP1594878A1 (en) 2005-11-16
PL378024A1 (pl) 2006-02-20
ATE397610T1 (de) 2008-06-15
DE602004014252D1 (de) 2008-07-17
AR042967A1 (es) 2005-07-13
IL169598A0 (en) 2007-07-04
TW200508240A (en) 2005-03-01
US20060205595A1 (en) 2006-09-14
AU2004207073B2 (en) 2010-09-16
BRPI0406875B1 (pt) 2014-05-27
CN1751049A (zh) 2006-03-22
CA2513573C (en) 2012-03-27
SI1594878T1 (sl) 2008-10-31
GB0302309D0 (en) 2003-03-05
IL169598A (en) 2010-05-17
DK1594878T3 (da) 2008-10-06
JP2006518347A (ja) 2006-08-10
CA2513573A1 (en) 2004-08-12
ES2308140T3 (es) 2008-12-01
CY1108295T1 (el) 2014-02-12
RU2329268C2 (ru) 2008-07-20
PT1594878E (pt) 2008-09-10
NZ541252A (en) 2008-05-30
EP1594878B1 (en) 2008-06-04
CN100410259C (zh) 2008-08-13

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06G Technical and formal requirements: other requirements [chapter 6.7 patent gazette]

Free format text: PARA QUE A SOLICITACAO DE DEVOLUCAO DE PRAZO SEJA ANALISADA, A MESMA DEVERA SER APRESENTADA AO INPI ACOMPANHADA DA COPIA DO PEDIDO DE FOTOCOPIA E DOS DEMAIS DOCUMENTOS LEGALMENTE EXIGIVEIS, DE ACORDO COM O ART. 3O DA RESOLUCAO 116/04.

B15Z Prolongation of time limit refused

Free format text: NEGADA A SOLICITACAO DE DEVOLUCAO DE PRAZO POR MOTIVO DE INSUFICIENCIA DE DOCUMENTOS, UMA VEZ QUE A MESMA NAO FOI APRESENTADA AO INPI ACOMPANHADA DA COPIA DO PEDIDO DE FOTOCOPIA E DOS DEMAIS DOCUMENTOS LEGALMENTE EXIGIVEIS, DE ACORDO COM O ART. 3O DA RESOLUCAO 116/04.

B25C Requirement related to requested transfer of rights

Owner name: SYNGENTA PARTICIPATIONS AG (CH)

Free format text: AFIM DE ATENDER A TRANSFERENCIA REQUERIDA ATRAVES DA PETICAO NO 020100074169/RJ DE 11/08/2010, E NECESSARIO REAPRESENTAR O DOCUMENTO DE CESSAO COM A DEVIDA LEGALIZACAO CONSULAR.

B25A Requested transfer of rights approved

Owner name: MERIAL LIMITED (GB)

Free format text: TRANSFERIDO DE: SYNGENTA PARTICIPATIONS AG

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 27/05/2014, OBSERVADAS AS CONDICOES LEGAIS.

B25A Requested transfer of rights approved
B25A Requested transfer of rights approved
B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 20A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2759 DE 21-11-2023 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.