BR9916774A - Derivados de imidazo[4,5-c]piridina-4-ona - Google Patents

Derivados de imidazo[4,5-c]piridina-4-ona

Info

Publication number: BR9916774A
Authority: BR; Brazil
Prior art keywords: pyridine; derivatives; imidazo; deimidazo; decoagulation
Prior art date: 1999-01-08

Application number

BR9916774-3A

Other languages

English (en)

Portuguese (pt)

Inventor

Werner Mederski

Horst Juraszyk

Hanns Wurziger

Christostsaklakidis

Dieter Dorsch

Sabine Bernotat-Danielowski

Guidomelzer

Soheila Anzali

Original Assignee

Merck Patent Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-01-08

Filing date

1999-12-21

Publication date

2001-10-30

1999-12-21 Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh

2001-10-30 Publication of BR9916774A publication Critical patent/BR9916774A/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Hematology (AREA)
Diabetes (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

BR9916774-3A 1999-01-08 1999-12-21 Derivados de imidazo[4,5-c]piridina-4-ona BR9916774A (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19900471A DE19900471A1 (de)	1999-01-08	1999-01-08	Imidazo[4,5c]-pyridin-4-on-derivate
PCT/EP1999/010236 WO2000040583A2 (de)	1999-01-08	1999-12-21	Imidazo[4,5-c]-pyridin-4-on-derivate

Publications (1)

Publication Number	Publication Date
BR9916774A true BR9916774A (pt)	2001-10-30

Family

ID=7893790

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BR9916774-3A BR9916774A (pt)	1999-01-08	1999-12-21	Derivados de imidazo[4,5-c]piridina-4-ona

Country Status (16)

Country	Link
EP (1)	EP1149099A2 (de)
JP (1)	JP2002534429A (de)
KR (1)	KR20010086085A (de)
CN (1)	CN1333772A (de)
AR (1)	AR022220A1 (de)
AU (1)	AU3041700A (de)
BR (1)	BR9916774A (de)
CA (1)	CA2357771A1 (de)
CZ (1)	CZ20012407A3 (de)
DE (1)	DE19900471A1 (de)
HU (1)	HUP0105054A3 (de)
NO (1)	NO20013384D0 (de)
PL (1)	PL349341A1 (de)
SK (1)	SK9442001A3 (de)
WO (1)	WO2000040583A2 (de)
ZA (1)	ZA200106454B (de)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL142959A0 (en)	1998-12-23	2002-04-21	Du Pont Pharm Co	Nitrogen containing heterobicycles as factor xa inhibitors
US6506771B2 (en)	2000-06-23	2003-01-14	Bristol-Myers Squibb Pharma Company	Heteroaryl-phenyl heterobicyclic factor Xa inhibitors
WO2002094197A2 (en)	2001-05-22	2002-11-28	Bristol-Myers Squibb Company	Bicyclic inhibitors of factor xa
GB0215293D0 (en)	2002-07-03	2002-08-14	Rega Foundation	Viral inhibitors
GB0225399D0 (en) *	2002-10-31	2002-12-11	Merck Sharp & Dohme	Therapeutic agents
AU2003302238A1 (en)	2002-12-03	2004-06-23	Axys Pharmaceuticals, Inc.	2-(2-hydroxybiphenyl-3-yl)-1h-benzoimidazole-5-carboxamidine derivatives as factor viia inhibitors
US7550590B2 (en)	2003-03-25	2009-06-23	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
EP1625122A1 (de)	2003-05-14	2006-02-15	Takeda San Diego, Inc.	Dipeptidylpeptidase-hemmer
US20050070531A1 (en)	2003-08-13	2005-03-31	Syrrx, Inc.	Dipeptidyl peptidase inhibitors
EP1706403B9 (de)	2003-12-22	2012-07-25	K.U.Leuven Research & Development	Imidazo[4,5-c]pyridinverbindungen und verfahren zur antiviralen behandlung
ATE426601T1 (de)	2004-12-21	2009-04-15	Gilead Sciences Inc	Imidazoa4,5-cupyridinverbindung und verfahren zur antiviralen behandlung
KR101083506B1 (ko)	2005-07-15	2011-11-16	에프. 호프만-라 로슈 아게	신규한 헤테로아릴 융합된 환형 아민
US20070060530A1 (en)	2005-09-14	2007-03-15	Christopher Ronald J	Administration of dipeptidyl peptidase inhibitors
EP1924567B1 (de)	2005-09-16	2012-08-22	Takeda Pharmaceutical Company Limited	Verfahren zur herstellung von pyrimidindionderivaten
WO2007112347A1 (en)	2006-03-28	2007-10-04	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
ATE454384T1 (de)	2006-07-07	2010-01-15	Gilead Sciences Inc	Neue pyridazinverbindung und ihre verwendung
TW200838536A (en)	2006-11-29	2008-10-01	Takeda Pharmaceutical	Polymorphs of succinate salt of 2-[6-(3-amino-piperidin-1-yl)-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethy]-4-fluor-benzonitrile and methods of use therefor
UA99466C2 (en)	2007-07-06	2012-08-27	Гилиад Сайенсиз, Инк.	Crystalline pyridazine compound
CN107074846B (zh) *	2014-08-12	2020-05-19	先正达参股股份有限公司	具有含硫取代基的杀有害生物活性杂环衍生物

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW219935B (de) *	1991-12-25	1994-02-01	Mitsubishi Chemicals Co Ltd
CA2309347A1 (en) *	1997-12-01	1999-06-10	Merck & Co., Inc.	Thrombin inhibitors

1999
- 1999-01-08 DE DE19900471A patent/DE19900471A1/de not_active Withdrawn
- 1999-12-21 CZ CZ20012407A patent/CZ20012407A3/cs unknown
- 1999-12-21 KR KR1020017007074A patent/KR20010086085A/ko not_active Withdrawn
- 1999-12-21 CA CA002357771A patent/CA2357771A1/en not_active Abandoned
- 1999-12-21 HU HU0105054A patent/HUP0105054A3/hu unknown
- 1999-12-21 CN CN99815465A patent/CN1333772A/zh active Pending
- 1999-12-21 PL PL99349341A patent/PL349341A1/xx unknown
- 1999-12-21 JP JP2000592291A patent/JP2002534429A/ja active Pending
- 1999-12-21 BR BR9916774-3A patent/BR9916774A/pt not_active Application Discontinuation
- 1999-12-21 EP EP99964639A patent/EP1149099A2/de not_active Withdrawn
- 1999-12-21 SK SK944-2001A patent/SK9442001A3/sk unknown
- 1999-12-21 AU AU30417/00A patent/AU3041700A/en not_active Abandoned
- 1999-12-21 WO PCT/EP1999/010236 patent/WO2000040583A2/de not_active Ceased
2000
- 2000-01-07 AR ARP000100062A patent/AR022220A1/es unknown
2001
- 2001-07-06 NO NO20013384A patent/NO20013384D0/no not_active Application Discontinuation
- 2001-08-06 ZA ZA200106454A patent/ZA200106454B/en unknown

Also Published As

Publication number	Publication date
NO20013384L (no)	2001-07-06
WO2000040583A3 (de)	2000-09-21
ZA200106454B (en)	2002-11-06
CA2357771A1 (en)	2000-07-13
PL349341A1 (en)	2002-07-15
AR022220A1 (es)	2002-09-04
DE19900471A1 (de)	2000-07-13
CZ20012407A3 (cs)	2001-12-12
JP2002534429A (ja)	2002-10-15
SK9442001A3 (en)	2002-05-09
HUP0105054A2 (hu)	2002-05-29
EP1149099A2 (de)	2001-10-31
HUP0105054A3 (en)	2002-12-28
AU3041700A (en)	2000-07-24
KR20010086085A (ko)	2001-09-07
WO2000040583A2 (de)	2000-07-13
NO20013384D0 (no)	2001-07-06
CN1333772A (zh)	2002-01-30

Publication	Publication Date	Title
BR9916774A (pt)	2001-10-30	Derivados de imidazo[4,5-c]piridina-4-ona
BR9813477A (pt)	2000-10-24	Derivados de benzamidina
BR9812699A (pt)	2000-08-22	Derivados de benzamidina
BR9917080A (pt)	2002-03-12	Composto, composição farmacêutica, uso do composto e método de tratamento ou prevenção de uma disfunção tromboembólica
BRPI0307057B8 (pt)	2021-05-25	compostos 2-(piridin-2-ilamino)-pirido[2,3-d]pirimidin-7-onas
BR0208891A (pt)	2004-04-20	Derivados de dihidro-benzo[b]-[1,4]diazepin-2-ona como antagonistas de mglur2 ii
MY130736A (en)	2007-07-31	Imidazo(4,5-c) pyridin-4-one derivatives
BRPI0409366A (pt)	2006-04-25	compostos de pirimido
BR0116034A (pt)	2004-08-03	Imidazopiridinas substituìdas
CO4910133A1 (es)	2000-04-24	Antagonistas de 5-h[1f]
NZ517758A (en)	2004-06-25	Pyrazolopyrimidines useful as therapeutic agents
BRPI0412291A (pt)	2006-09-19	antagonistas duplos de nka/nk3 para o tratamento de esquizofrenia
AU2002246728A1 (en)	2002-08-28	Carboline derivatives
MXPA03006483A (es)	2003-09-22	Derivados de fenilo.
DK1222195T3 (da)	2004-04-19	Hidtil ukendte thiazolo[4,5-d]pyrimidinforbindelser
BR0309342A (pt)	2005-02-15	Composto, composição farmacêutica, uso de um composto, e, método de tratamento ou profilaxia de doenças ou condições humanas
BR0309463A (pt)	2005-02-09	Derivados de 1,2,3,4,7,8-hexaidro-6h-[1,4]diazepino[6,7,1-ij]quinolina como agentes antipsicóticos e antiobesidade
AU2002213421A1 (en)	2002-04-15	Condensed pyridoindole derivatives
AU2002249890A1 (en)	2002-08-28	Carboline derivatives
BR0210531A (pt)	2004-06-22	Derivados de ácido sulfÈnico
BR0207166A (pt)	2004-02-10	Composto, e, composição farmacêutica
AU2002213419A1 (en)	2002-04-15	Condensed pyridoindole derivatives
BR0008608A (pt)	2002-01-02	Derivados de pirazol-3-ona
NO975028L (no)	1997-12-30	Piperazinoderivater som neurokininantagonister
PT916670E (pt)	2003-09-30	Pirrolo-(3,2-b) piridinas e o seu uso como agonistas do 5-ht1f

Legal Events

Date	Code	Title	Description
2003-12-09	FA10	Dismissal: dismissal - article 33 of industrial property law
2004-07-27	B11Y	Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]