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BR9914521A - Glycuronides of pregnane - Google Patents

Glycuronides of pregnane

Info

Publication number
BR9914521A
BR9914521A BR9914521-9A BR9914521A BR9914521A BR 9914521 A BR9914521 A BR 9914521A BR 9914521 A BR9914521 A BR 9914521A BR 9914521 A BR9914521 A BR 9914521A
Authority
BR
Brazil
Prior art keywords
beta
pregnane
glycuronides
pregnan
alpha
Prior art date
Application number
BR9914521-9A
Other languages
Portuguese (pt)
Inventor
Christopher Paul Miller
Bach Dinh Tran
Michael David Collini
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Publication of BR9914521A publication Critical patent/BR9914521A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J17/005—Glycosides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C07J5/0007—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa
    • C07J5/0015—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa not substituted in position 16

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Patente de Invenção: <B>GLICURONìDEOS DE PREGNANO"<D>. Esta invenção provê 5-alfa-pregnano-3-beta, (20S), 21-triol, 20-O-beta-glicuronídeo e 5-alfa-pregnano-3-beta,20R-diol, 20-O-beta glicuronídeo e seus sais farmaceuticamente aceitáveis que são úteis como agentes progestacionais.Invention Patent: <B> PREGNANE GLYCURONIDS "<D>. This invention provides 5-alpha-pregnan-3-beta, (20S), 21-triol, 20-O-beta-glucuronide and 5-alpha-pregnan- 3-beta, 20R-diol, 20-O-beta glucuronide and their pharmaceutically acceptable salts which are useful as progestational agents.

BR9914521-9A 1998-10-13 1999-10-07 Glycuronides of pregnane BR9914521A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17034298A 1998-10-13 1998-10-13
PCT/US1999/023467 WO2000021977A1 (en) 1998-10-13 1999-10-07 Pregnane glucuronides

Publications (1)

Publication Number Publication Date
BR9914521A true BR9914521A (en) 2001-06-26

Family

ID=22619512

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9914521-9A BR9914521A (en) 1998-10-13 1999-10-07 Glycuronides of pregnane

Country Status (17)

Country Link
EP (1) EP1121376A1 (en)
JP (1) JP2002527448A (en)
KR (1) KR20010080102A (en)
CN (1) CN1330659A (en)
AR (1) AR020778A1 (en)
AU (1) AU751708B2 (en)
BR (1) BR9914521A (en)
CA (1) CA2346693A1 (en)
CZ (1) CZ20011343A3 (en)
EA (1) EA200100437A1 (en)
HU (1) HUP0103992A3 (en)
IL (1) IL142441A0 (en)
NO (1) NO20011825L (en)
PL (1) PL347270A1 (en)
TW (1) TW499435B (en)
WO (1) WO2000021977A1 (en)
ZA (1) ZA200103012B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0104423D0 (en) * 2001-12-27 2001-12-27 Umecrine Ab Pregnane steroids and their use in the treatment of CNS disorders
KR100440607B1 (en) * 2001-12-28 2004-07-15 주식회사 엘컴사이언스 Pregnan glycoside compounds and preventives and remedies of neurodegenerative disease containing them as active ingredients

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2029011B (en) * 1978-09-01 1983-02-02 Coulson W Use of a synthetic bifunctional ligand for the immunimetric determination of the concentration ratio of two solutes

Also Published As

Publication number Publication date
CA2346693A1 (en) 2000-04-20
EP1121376A1 (en) 2001-08-08
HUP0103992A3 (en) 2002-12-28
PL347270A1 (en) 2002-03-25
AR020778A1 (en) 2002-05-29
NO20011825D0 (en) 2001-04-10
TW499435B (en) 2002-08-21
JP2002527448A (en) 2002-08-27
KR20010080102A (en) 2001-08-22
ZA200103012B (en) 2002-07-11
CZ20011343A3 (en) 2002-04-17
EA200100437A1 (en) 2001-10-22
CN1330659A (en) 2002-01-09
WO2000021977A1 (en) 2000-04-20
AU6511599A (en) 2000-05-01
AU751708B2 (en) 2002-08-22
NO20011825L (en) 2001-06-05
HUP0103992A2 (en) 2002-04-29
IL142441A0 (en) 2002-03-10

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 5A, 6A, 7A E 8A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1913 DE 04/09/2007.