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BR9914306A - Derivados do 1h-imidazopiridina - Google Patents

Derivados do 1h-imidazopiridina

Info

Publication number
BR9914306A
BR9914306A BR9914306-2A BR9914306A BR9914306A BR 9914306 A BR9914306 A BR 9914306A BR 9914306 A BR9914306 A BR 9914306A BR 9914306 A BR9914306 A BR 9914306A
Authority
BR
Brazil
Prior art keywords
group
derivatives
hydrogen atom
chain
imidazopyridine derivatives
Prior art date
Application number
BR9914306-2A
Other languages
English (en)
Inventor
Hideo Kato
Jun Sakaguchi
Makoto Aoyama
Tomoyuki Izumi
Ken-Ichi Kato
Original Assignee
Hokuriku Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hokuriku Pharmaceutical filed Critical Hokuriku Pharmaceutical
Publication of BR9914306A publication Critical patent/BR9914306A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

"DERIVADOS DO 1H-IMIDAZOPIRIDINA". "representado pela fórmula geral seguinte ou sais do mesmo. na qual R1 representa átomo de hidrogênio, grupo hidroxil, um grupo alquila, um grupo cicloalquila, grupo estiril, ou um grupo aril; R2 representa átomo de hidrogênio, um grupo alquila, um átomo de halogênio, grupo hidroxil, grupo amino, um grupo amino ciclico, ou grupo fenoxi; a ligação ou cadeia A representa uma cadeia homocíclica ou heterocíclica a qual pode ser substituída; R3 representa um grupo heterocíclico saturado contendo nitrogênio; e m representa um número inteiro de 0 a 3. Os derivados possuem excelentes ações inibidoras contra a produção de TNF ou IL-1 e são extremamente úteis como agentes preventivos ou terapêuticos para enfermidades nas quais uma citoquina é mediada.
BR9914306-2A 1998-08-12 1999-08-12 Derivados do 1h-imidazopiridina BR9914306A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP24106298 1998-08-12
JP11216125A JP2000119271A (ja) 1998-08-12 1999-07-30 １ｈ―イミダゾピリジン誘導体
PCT/JP1999/004381 WO2000009506A1 (en) 1998-08-12 1999-08-12 1h-imidazopyridine derivatives

Publications (1)

Publication Number Publication Date
BR9914306A true BR9914306A (pt) 2002-05-21

Family

ID=26521247

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9914306-2A BR9914306A (pt) 1998-08-12 1999-08-12 Derivados do 1h-imidazopiridina

Country Status (21)

Country Link
US (1) US6518265B1 (pt)
EP (1) EP1104764A4 (pt)
JP (1) JP2000119271A (pt)
CN (1) CN1323307A (pt)
AU (1) AU744388B2 (pt)
BG (1) BG105271A (pt)
BR (1) BR9914306A (pt)
CA (1) CA2339562A1 (pt)
CZ (1) CZ292544B6 (pt)
EA (1) EA200100230A1 (pt)
HK (1) HK1042295A1 (pt)
HR (1) HRP20010144A2 (pt)
HU (1) HUP0103406A3 (pt)
IL (1) IL141226A0 (pt)
NO (1) NO20010676L (pt)
NZ (1) NZ509939A (pt)
PL (1) PL346155A1 (pt)
SK (1) SK1942001A3 (pt)
TR (1) TR200100439T2 (pt)
TW (1) TW533209B (pt)
WO (1) WO2000009506A1 (pt)

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* Cited by examiner, † Cited by third party
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