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BR9911770A - Processo para a preparação estereoquimicamente controlada de compostos azacìclicos com elevado grau de substituição, isomericamente puros - Google Patents

Processo para a preparação estereoquimicamente controlada de compostos azacìclicos com elevado grau de substituição, isomericamente puros

Info

Publication number
BR9911770A
BR9911770A BR9911770-3A BR9911770A BR9911770A BR 9911770 A BR9911770 A BR 9911770A BR 9911770 A BR9911770 A BR 9911770A BR 9911770 A BR9911770 A BR 9911770A
Authority
BR
Brazil
Prior art keywords
compounds
azomeric
controlled preparation
stereochemically controlled
isomerically pure
Prior art date
Application number
BR9911770-3A
Other languages
English (en)
Inventor
Michael Reggelin
Timo Heinrich
Bernd Junker
Jochen Antel
Ulf Preuschoff
Original Assignee
Solvay Pharm Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Gmbh filed Critical Solvay Pharm Gmbh
Publication of BR9911770A publication Critical patent/BR9911770A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D291/00—Heterocyclic compounds containing rings having nitrogen, oxygen and sulfur atoms as the only ring hetero atoms
    • C07D291/02—Heterocyclic compounds containing rings having nitrogen, oxygen and sulfur atoms as the only ring hetero atoms not condensed with other rings
    • C07D291/04—Five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C381/00—Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/00 - C07C337/00
    • C07C381/10—Compounds containing sulfur atoms doubly-bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/12—Oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Indole Compounds (AREA)

Abstract

Patente de Invenção: <B>"PROCESSO PARA A PREPARAçãO ESTEREOQUIMICAMENTE CONTROLADA DE COMPOSTOS AZACìCLI-COS COM ELEVADO GRAU DE SUBSTITUIçãO, ISOMERICAMENTE PUROS"<D>. Descreve-se um processo para a preparação estereoquimicamente controlada de compostos azacíclicos da fórmula geral (I), em que os substituintes possuem as significações mencionadas na descrição, assim como produtos intermediários deste processo e novos compostos azacíclicos.
BR9911770-3A 1998-05-13 1999-05-10 Processo para a preparação estereoquimicamente controlada de compostos azacìclicos com elevado grau de substituição, isomericamente puros BR9911770A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19821418 1998-05-13
PCT/DE1999/001417 WO1999058500A1 (de) 1998-05-13 1999-05-10 Verfahren zur stereochemisch kontrollierten herstellung isomerenreiner hochsubstituierter azacyclischer verbindungen

Publications (1)

Publication Number Publication Date
BR9911770A true BR9911770A (pt) 2001-02-06

Family

ID=7867628

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9911770-3A BR9911770A (pt) 1998-05-13 1999-05-10 Processo para a preparação estereoquimicamente controlada de compostos azacìclicos com elevado grau de substituição, isomericamente puros

Country Status (28)

Country Link
US (1) US6900322B1 (pt)
EP (1) EP1076646B1 (pt)
JP (1) JP4503833B2 (pt)
KR (1) KR20010043475A (pt)
CN (1) CN1252052C (pt)
AR (1) AR016247A1 (pt)
AT (1) ATE272621T1 (pt)
AU (1) AU758192B2 (pt)
BR (1) BR9911770A (pt)
CA (1) CA2331758C (pt)
DE (2) DE59910141D1 (pt)
DK (1) DK1076646T3 (pt)
DZ (1) DZ2787A1 (pt)
ES (1) ES2228074T3 (pt)
HU (1) HUP0101808A3 (pt)
ID (1) ID26787A (pt)
IL (1) IL139519A0 (pt)
NO (1) NO317986B1 (pt)
NZ (1) NZ508043A (pt)
PL (1) PL197406B1 (pt)
PT (1) PT1076646E (pt)
RU (1) RU2225395C2 (pt)
SK (1) SK17122000A3 (pt)
TR (1) TR200003291T2 (pt)
TW (1) TWI220143B (pt)
UA (1) UA66859C2 (pt)
WO (1) WO1999058500A1 (pt)
ZA (1) ZA200006337B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7119207B2 (en) 2000-04-10 2006-10-10 Pfizer Inc Benzoamide piperidine containing compounds and related compounds
JP4001486B2 (ja) * 2000-04-10 2007-10-31 ファイザー・プロダクツ・インク ベンゾアミドピペリジン含有化合物及び関連化合物
US7968734B2 (en) * 2004-07-01 2011-06-28 Stc.Unm Organocatalysts and methods of use in chemical synthesis
NZ604035A (en) 2010-06-04 2015-02-27 Albany Molecular Res Inc Glycine transporter-1 inhibitors, methods of making them, and uses thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5102877A (en) * 1989-04-28 1992-04-07 Fujisawa Pharmaceutical Co., Ltd. 1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid compounds
US5100891A (en) * 1991-01-18 1992-03-31 Hoechst-Roussel Pharmaceuticals Inc. Substituted 1,2,3,4-tetrahydrocyclopent[b]indoles, 1,2,3,3a,4,8a-hexahydrocyclopent[B]indoles and related compounds
TW214545B (pt) * 1992-02-17 1993-10-11 Ciba Geigy Ag
US5252747A (en) * 1992-09-11 1993-10-12 Abbott Laboratories Chiral quinolone intermediates

Also Published As

Publication number Publication date
DE59910141D1 (de) 2004-09-09
SK17122000A3 (sk) 2001-04-09
WO1999058500B1 (de) 1999-12-29
ZA200006337B (en) 2001-05-16
AU758192B2 (en) 2003-03-20
NZ508043A (en) 2003-05-30
EP1076646B1 (de) 2004-08-04
EP1076646A1 (de) 2001-02-21
US6900322B1 (en) 2005-05-31
UA66859C2 (uk) 2004-06-15
AU5025099A (en) 1999-11-29
NO20005666D0 (no) 2000-11-10
CN1252052C (zh) 2006-04-19
DZ2787A1 (fr) 2003-12-01
HUP0101808A3 (en) 2002-05-28
ID26787A (id) 2001-02-08
ES2228074T3 (es) 2005-04-01
WO1999058500A1 (de) 1999-11-18
DE19921580A1 (de) 1999-11-25
CA2331758A1 (en) 1999-11-18
CA2331758C (en) 2009-01-20
JP2002514624A (ja) 2002-05-21
TWI220143B (en) 2004-08-11
CN1299345A (zh) 2001-06-13
TR200003291T2 (tr) 2001-03-21
AR016247A1 (es) 2001-06-20
NO20005666L (no) 2000-11-10
PL344043A1 (en) 2001-09-24
KR20010043475A (ko) 2001-05-25
PT1076646E (pt) 2004-10-29
HUP0101808A2 (hu) 2001-09-28
IL139519A0 (en) 2001-11-25
PL197406B1 (pl) 2008-03-31
RU2225395C2 (ru) 2004-03-10
NO317986B1 (no) 2005-01-17
ATE272621T1 (de) 2004-08-15
HK1036624A1 (en) 2002-01-11
DK1076646T3 (da) 2004-09-06
JP4503833B2 (ja) 2010-07-14

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Legal Events

Date Code Title Description
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07G Grant request does not fulfill article 229-c lpi (prior consent of anvisa) [chapter 7.7 patent gazette]

Free format text: NOTIFICACAO DE DEVOLUCAO DO PEDIDO POR NAO SE ENQUADRAR NO ART. 229-C DA LPI.

B08L Patent application lapsed because of non payment of annual fee [chapter 8.12 patent gazette]

Free format text: ARQUIVAMENTO DEFINITIVO

B08I Publication cancelled [chapter 8.9 patent gazette]

Free format text: ANULADA A PUBLICACAO CODIGO 8.12 NA RPI NO 2253 DE 11/03/2014 POR TER SIDO INDEVIDA.

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

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B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2602 DE 17-11-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.