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BR9611628A - Derivados de pirido [2,3-d] pirimidina e composições medicinais dos mesmos - Google Patents

Derivados de pirido [2,3-d] pirimidina e composições medicinais dos mesmos

Info

Publication number
BR9611628A
BR9611628A BR9611628A BR9611628A BR9611628A BR 9611628 A BR9611628 A BR 9611628A BR 9611628 A BR9611628 A BR 9611628A BR 9611628 A BR9611628 A BR 9611628A BR 9611628 A BR9611628 A BR 9611628A
Authority
BR
Brazil
Prior art keywords
pyrido
pyrimidine derivatives
medicinal compositions
medicinal
compositions
Prior art date
Application number
BR9611628A
Other languages
English (en)
Inventor
Kazuhisa Takayama
Hiroyuki Hisamichi
Masahiro Iwata
Hideki Kubota
Motonori Aoki
Original Assignee
Yamanouchi Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd
Publication of BR9611628A publication Critical patent/BR9611628A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BR9611628A 1995-11-21 1996-11-20 Derivados de pirido [2,3-d] pirimidina e composições medicinais dos mesmos BR9611628A (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP30306595 1995-11-21
JP772596 1996-01-19
JP4385396 1996-02-29
JP14186896 1996-06-04
PCT/JP1996/003389 WO1997019078A1 (fr) 1995-11-21 1996-11-20 DERIVES DE PYRIDO[2,3-d] PYRIMIDINE ET LEURS COMPOSES A USAGE MEDICAL

Publications (1)

Publication Number Publication Date
BR9611628A true BR9611628A (pt) 1999-06-01

Family

ID=27454776

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9611628A BR9611628A (pt) 1995-11-21 1996-11-20 Derivados de pirido [2,3-d] pirimidina e composições medicinais dos mesmos

Country Status (12)

Country Link
US (1) US6136810A (pt)
EP (1) EP0885894A4 (pt)
JP (1) JP3110765B2 (pt)
KR (1) KR19990071520A (pt)
CN (1) CN1202171A (pt)
AU (1) AU705039B2 (pt)
BR (1) BR9611628A (pt)
CA (1) CA2236683A1 (pt)
HU (1) HUP9900607A3 (pt)
NZ (1) NZ322197A (pt)
TW (1) TW377352B (pt)
WO (1) WO1997019078A1 (pt)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6417190B1 (en) * 1998-12-17 2002-07-09 Boehringer Ingelheim Pharma Kg Tricyclic nitrogen heterocycles as PDE IV inhibitors
EP1671651B1 (en) 1999-08-21 2009-11-11 Nycomed GmbH Synergistic combination of pumafentrine and salmeterol
EP1267903A4 (en) * 2000-02-08 2003-08-06 Pharmacia Corp METHOD FOR TREATING GLAUCOMA
US6413968B1 (en) * 2000-06-30 2002-07-02 O'donnell, Jr. Francis E. Treatment of myasthenia gravis by cyclic nucleotide phosphodiesterase inhibition
AU2002224417A1 (en) * 2000-10-18 2002-04-29 Immunex Corporation Methods for treating il-18 mediated disorders
WO2002060479A1 (en) * 2001-01-29 2002-08-08 Applied Research Systems Ars Holding N.V. Use of il-18 inhibitors for the treatment and/or prevention of heart disease
EP1364950A4 (en) * 2001-02-26 2005-03-09 Tanabe Seiyaku Co Pyridopyrimidine and naphthyridine derivatives
AU2002324625B2 (en) * 2001-08-07 2008-05-08 Immunex Corporation Interleukin-1 receptors in the treatment of diseases
KR100490970B1 (ko) * 2002-03-22 2005-05-24 씨제이 주식회사 신규 피리도[2,3-ｄ]피리미딘 카르보알데히드 옥심계ＰＤＥ Ⅳ 효소 저해 화합물 및 이의 제조방법
WO2004087211A2 (en) 2003-04-01 2004-10-14 Applied Research Systems Ars Holding N.V. Inhibitors of phosphodiesterases in infertility
ES2378374T3 (es) * 2003-11-20 2012-04-11 Astellas Pharma Inc. Inhibidores de la PDE 4 para el tratamiento de la cistitis intersticial
TW200738243A (en) * 2005-11-15 2007-10-16 Glaxo Group Ltd Novel process and formulations
US7750019B2 (en) * 2006-08-11 2010-07-06 Kowa Company, Ltd. Pyrimidine compound having benzyl(pyridylmethyl)amine structure and medicament comprising the same
MX2009008253A (es) 2007-01-31 2009-10-12 Vertex Pharma Derivados de 2-aminopiridina utiles como inhibidores de cinasa.
US7790737B2 (en) 2007-03-13 2010-09-07 Kowa Company, Ltd. Substituted pyrimidine compounds and their utility as CETP inhibitors
JP5240205B2 (ja) 2008-01-11 2013-07-17 アステラス製薬株式会社 精巣の疼痛又は不快感行動及び頻尿併発モデル動物
KR20110039563A (ko) 2008-07-23 2011-04-19 버텍스 파마슈티칼스 인코포레이티드 피라졸로피리딘 키나제 억제제
US8569337B2 (en) 2008-07-23 2013-10-29 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
AU2009274023A1 (en) 2008-07-23 2010-01-28 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
MX2011001319A (es) 2008-08-06 2011-04-05 Vertex Pharma Inhibidores de aminopiridina cinasa.
AU2010245914A1 (en) 2009-05-06 2011-12-15 Vertex Pharmaceuticals Incorporated Pyrazolopyridines
AU2011209651A1 (en) 2010-01-27 2012-08-09 Vertex Pharmaceuticals Incorporated Pyrazolopyrimidine kinase inhibitors
US9067932B2 (en) 2010-01-27 2015-06-30 Vertex Pharmaceuticals Incorporated Pyrazolopyridine kinase inhibitors
EP2550272A1 (en) 2010-01-27 2013-01-30 Vertex Pharmaceuticals Incorporated Pyrazolopyrazine kinase inhibitors
BR112021010842A2 (pt) * 2018-12-10 2021-08-24 Ideaya Biosciences, Inc. Derivados de 2-oxoquinazolina como inibidores de metionina adenosiltransferase 2a

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA932731A (en) * 1968-12-10 1973-08-28 E. Hardtmann Goetz 1,2-dihydro-pyrido(2,3-d)pyrimidin-2-ones
BE757702A (fr) * 1969-10-20 1971-04-19 Sandoz Sa Derives de la pyrido (2,3-d) pyrimidine, leur preparation et medicaments les contenant.
US3709888A (en) * 1970-06-01 1973-01-09 Sandoz Ag Aryl-substituted-pyrido(2,3-d)pyrimidin-2-ones
US3853898A (en) * 1971-07-20 1974-12-10 Sandoz Ag 3-(2-substituted amino) pyridyl-phenyl ketone imines
US3758475A (en) * 1971-07-20 1973-09-11 Sandoz Ag Pyrido(2,3-d)pyrimidin 2 ones
JPS5394040A (en) * 1976-12-06 1978-08-17 Sandoz Ag Coagolation controlling agent for blood platelet
US4224328A (en) * 1979-04-11 1980-09-23 Sandoz, Inc. Methods with 1-substituted-4-aryl-quinazolin-2(1H)-ones and thiones and pyrido[2,3-d]pyrimidin-2-ones as platelet aggregation inhibitors
PH23853A (en) * 1986-08-21 1989-11-23 Pfizer Pyridopyrimidinediones
US5264437A (en) * 1992-03-20 1993-11-23 Syntex (U.S.A.) Inc. Optionally substituted pyrido[2,3-d]pyridine-2,4(1H,3H)-diones and pyrido[2,]pyrimidine-2(1H,3H)-ones
TW299333B (pt) * 1992-12-29 1997-03-01 Takeda Pharm Industry Co Ltd

Also Published As

Publication number Publication date
JP3110765B2 (ja) 2000-11-20
AU705039B2 (en) 1999-05-13
EP0885894A1 (en) 1998-12-23
US6136810A (en) 2000-10-24
WO1997019078A1 (fr) 1997-05-29
EP0885894A4 (en) 2000-01-19
TW377352B (en) 1999-12-21
NZ322197A (en) 1999-02-25
HUP9900607A2 (hu) 1999-06-28
CN1202171A (zh) 1998-12-16
AU7588696A (en) 1997-06-11
KR19990071520A (ko) 1999-09-27
CA2236683A1 (en) 1997-05-29
HUP9900607A3 (en) 1999-11-29

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law