BR9608721A - Composição farmacêutica, e, processo para tratar inflamação - Google Patents
Composição farmacêutica, e, processo para tratar inflamaçãoInfo
- Publication number
- BR9608721A BR9608721A BR9608721-8A BR9608721A BR9608721A BR 9608721 A BR9608721 A BR 9608721A BR 9608721 A BR9608721 A BR 9608721A BR 9608721 A BR9608721 A BR 9608721A
- Authority
- BR
- Brazil
- Prior art keywords
- pharmaceutical composition
- metal
- treating inflammation
- degradation
- conditions
- Prior art date
Links
- 206010061218 Inflammation Diseases 0.000 title abstract 2
- 230000004054 inflammatory process Effects 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- KCXVZYZYPLLWCC-UHFFFAOYSA-N EDTA Chemical compound OC(=O)CN(CC(O)=O)CCN(CC(O)=O)CC(O)=O KCXVZYZYPLLWCC-UHFFFAOYSA-N 0.000 abstract 2
- 229940071106 ethylenediaminetetraacetate Drugs 0.000 abstract 2
- 239000002184 metal Substances 0.000 abstract 2
- 239000007864 aqueous solution Substances 0.000 abstract 1
- 239000003637 basic solution Substances 0.000 abstract 1
- 230000015556 catabolic process Effects 0.000 abstract 1
- 238000006555 catalytic reaction Methods 0.000 abstract 1
- 230000007423 decrease Effects 0.000 abstract 1
- 238000006731 degradation reaction Methods 0.000 abstract 1
- 229910021645 metal ion Inorganic materials 0.000 abstract 1
- 230000007935 neutral effect Effects 0.000 abstract 1
- 238000010525 oxidative degradation reaction Methods 0.000 abstract 1
- 239000003352 sequestering agent Substances 0.000 abstract 1
- 229960002117 triamcinolone acetonide Drugs 0.000 abstract 1
- YNDXUCZADRHECN-JNQJZLCISA-N triamcinolone acetonide Chemical compound C1CC2=CC(=O)C=C[C@]2(C)[C@]2(F)[C@@H]1[C@@H]1C[C@H]3OC(C)(C)O[C@@]3(C(=O)CO)[C@@]1(C)C[C@@H]2O YNDXUCZADRHECN-JNQJZLCISA-N 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
- A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Colloid Chemistry (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
"COMPOSIçãO FARMACêUTICA, E, PROCESSO PARA TRATAR INFLAMAçãO". A degradação de triancinolona acetonida em soluções aquosas é estudada sob condições de armazenagem acelerada de 70‹C sobre a faixa de pH de 1-10. Os íons metálicos a níveis bem baixos podem acelerar fortemente a degradação oxidativa em soluções neutras e básicas, mas as condições de pH e/ou a inclusão de agentes seq³estrantes de metal, tais como acetato de tetra etilenodiamina (EDTA), em uma preparação diminui a catálise de metal.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US48533995A | 1995-06-07 | 1995-06-07 | |
| PCT/US1996/009651 WO1996040042A2 (en) | 1995-06-07 | 1996-06-05 | Stabilized steroid compositions |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9608721A true BR9608721A (pt) | 1999-10-13 |
Family
ID=23927770
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9608721-8A BR9608721A (pt) | 1995-06-07 | 1996-06-05 | Composição farmacêutica, e, processo para tratar inflamação |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP0843548A4 (pt) |
| JP (1) | JPH11507359A (pt) |
| AU (1) | AU6164196A (pt) |
| BR (1) | BR9608721A (pt) |
| CA (1) | CA2223385A1 (pt) |
| WO (1) | WO1996040042A2 (pt) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6315985B1 (en) | 1999-06-18 | 2001-11-13 | 3M Innovative Properties Company | C-17/21 OH 20-ketosteroid solution aerosol products with enhanced chemical stability |
| WO2006089656A2 (en) * | 2005-02-25 | 2006-08-31 | Chiesi Farmaceutici S.P.A. | Pharmaceutical aerosol formulations for pressurized metered dose inhalers comprising a sequestering agent |
| BRPI0720588B8 (pt) | 2006-12-21 | 2021-05-25 | Nerviano Medical Sciences Srl | derivados de pirazol-quinazolina substituídos, processo para sua preparação e seu uso como inibidores da quinase |
| EP3456314A1 (en) | 2017-09-14 | 2019-03-20 | Tiofarma B.V. | Topical formulation comprising 17-ketolic corticosteroid |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4344940A (en) * | 1981-11-30 | 1982-08-17 | E. R. Squibb & Sons, Inc. | Steroid formulation containing dipotassium EDTA |
| US5542935A (en) * | 1989-12-22 | 1996-08-06 | Imarx Pharmaceutical Corp. | Therapeutic delivery systems related applications |
| EP0611301B1 (en) * | 1990-04-26 | 2003-06-11 | The Procter & Gamble Company | Chelator compositions comprising oxime compounds |
| KR950000032A (ko) * | 1993-06-09 | 1995-01-03 | 류경열 | 맛참기름 제조방법 |
-
1996
- 1996-06-05 CA CA002223385A patent/CA2223385A1/en not_active Abandoned
- 1996-06-05 BR BR9608721-8A patent/BR9608721A/pt not_active Application Discontinuation
- 1996-06-05 AU AU61641/96A patent/AU6164196A/en not_active Abandoned
- 1996-06-05 EP EP96919250A patent/EP0843548A4/en not_active Withdrawn
- 1996-06-05 JP JP9501925A patent/JPH11507359A/ja active Pending
- 1996-06-05 WO PCT/US1996/009651 patent/WO1996040042A2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO1996040042A3 (en) | 1997-02-06 |
| EP0843548A4 (en) | 1998-10-28 |
| CA2223385A1 (en) | 1996-12-19 |
| JPH11507359A (ja) | 1999-06-29 |
| MX9709431A (es) | 1998-10-31 |
| EP0843548A2 (en) | 1998-05-27 |
| WO1996040042A2 (en) | 1996-12-19 |
| AU6164196A (en) | 1996-12-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA10 | Dismissal: dismissal - article 33 of industrial property law |