BR0208861A - Processo para a preparação de um composto, e, composto - Google Patents
Processo para a preparação de um composto, e, compostoInfo
- Publication number
- BR0208861A BR0208861A BR0208861-4A BR0208861A BR0208861A BR 0208861 A BR0208861 A BR 0208861A BR 0208861 A BR0208861 A BR 0208861A BR 0208861 A BR0208861 A BR 0208861A
- Authority
- BR
- Brazil
- Prior art keywords
- sup
- compound
- formula
- preparation
- alcohol
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Heart & Thoracic Surgery (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Steroid Compounds (AREA)
Abstract
"PROCESSO PARA A PREPARAçãO DE UM COMPOSTO, E, COMPOSTO". é fornecido um processo para a preparação de um composto da fórmula (I): processo este que compreende a reação de um composto da fórmula (II): com um composto da fórmula (III): ou acrilamida, seguido, no último caso, pela reação do intermediário resultante da fórmula (IV): com um álcool da fórmula R^ 2^-OH e um agente que promova ou agentes que em combinação promovam, o rearranjo e oxidação do composto da fórmula IV para um isocianato intermediário, que pode depois reagir com o álcool da fórmula R^ 2^-OH e em que R^ 1^, R^ 2^e R^ 16^ têm os significados dados na descrição.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0101324A SE0101324D0 (sv) | 2001-04-12 | 2001-04-12 | New process |
| PCT/SE2002/000727 WO2002083690A1 (en) | 2001-04-12 | 2002-04-12 | New process for the preparation of oxabispidines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0208861A true BR0208861A (pt) | 2004-10-19 |
Family
ID=20283781
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0208861-4A BR0208861A (pt) | 2001-04-12 | 2002-04-12 | Processo para a preparação de um composto, e, composto |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US7169921B2 (pt) |
| EP (1) | EP1385850B1 (pt) |
| JP (1) | JP4248880B2 (pt) |
| KR (1) | KR100848613B1 (pt) |
| CN (1) | CN1267435C (pt) |
| AT (1) | ATE284405T1 (pt) |
| AU (1) | AU2002249748B2 (pt) |
| BR (1) | BR0208861A (pt) |
| CA (1) | CA2443475A1 (pt) |
| DE (1) | DE60202203T2 (pt) |
| ES (1) | ES2233809T3 (pt) |
| IL (2) | IL158249A0 (pt) |
| MX (1) | MXPA03009211A (pt) |
| NO (1) | NO20034526L (pt) |
| NZ (1) | NZ528515A (pt) |
| PT (1) | PT1385850E (pt) |
| SE (1) | SE0101324D0 (pt) |
| WO (1) | WO2002083690A1 (pt) |
| ZA (1) | ZA200307676B (pt) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0101324D0 (sv) * | 2001-04-12 | 2001-04-12 | Astrazeneca Ab | New process |
| GB0223712D0 (en) | 2002-10-14 | 2002-11-20 | Astrazeneca Ab | Chemical intermediate |
| US20040192738A1 (en) * | 2003-03-18 | 2004-09-30 | Aventis Pharma Deutschland Gmbh | 2-(Butyl-1-sulfonylamino)-N-[1(R)-(6-methoxypyridin-3-yl)propyl] benzamide, its use as a medicament, and pharmaceutical preparations comprising it |
| SE0401539D0 (sv) * | 2004-06-15 | 2004-06-15 | Astrazeneca Ab | New compounds |
| SE0401540D0 (sv) * | 2004-06-15 | 2004-06-15 | Astrazeneca Ab | New compounds |
| AR057064A1 (es) * | 2005-06-13 | 2007-11-14 | Astrazeneca Ab | Compuestos para el tratamiento de arritmias cardiacas, formulacion farmaceutica y preparacion del compuesto |
| AU2006259056A1 (en) * | 2005-06-16 | 2006-12-21 | Girindus Ag | Synthesis of hydroquinone derivatives |
| US20100160626A1 (en) * | 2005-06-20 | 2010-06-24 | Astrazeneca Ab | Process For The Preparation Of 3,7-Dihydroxy-1,5-Diazacyclooctanes |
| AU2006259938B2 (en) * | 2005-06-20 | 2010-07-01 | Astrazeneca Ab | Process for the preparation of sulfonic acid salts of oxabispidines |
| WO2006137774A1 (en) * | 2005-06-20 | 2006-12-28 | Astrazeneca Ab | Process for the production of (alkoxycarbonylamino)alkyl sulfonates |
| AR053901A1 (es) * | 2005-06-20 | 2007-05-23 | Astrazeneca Ab | Formas fisicas de oxabispidinas n,n'- disustituidas |
| AR057364A1 (es) * | 2005-06-20 | 2007-11-28 | Astrazeneca Ab | Proceso para el aislamiento de 4-(oxiranilmetoxi) -benzonitrilos |
| BRPI0611839A2 (pt) * | 2005-06-20 | 2016-08-30 | Astrazeneca Ab | processos para a preparação de um sal de ácido sulfônico e para a preparação de um composto, e, mistura |
| AU2014237340C1 (en) | 2013-03-15 | 2018-11-08 | Global Blood Therapeutics, Inc. | Compounds and uses thereof for the modulation of hemoglobin |
| EA202092627A1 (ru) | 2013-11-18 | 2021-09-30 | Глобал Блад Терапьютикс, Инк. | Соединения и их применения для модуляции гемоглобина |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3196154A (en) | 1962-05-17 | 1965-07-20 | Sterling Drug Inc | 3-substituted-9-methyl-3, 9-diazabicyclo [3.3.1] nonanes |
| US5110933A (en) * | 1989-11-13 | 1992-05-05 | Board Of Regents Of Oklahoma State University | Salts of 3-azabicyclo[3.3.1]nonanes as antiarrhythmic agents, and precursors thereof |
| SE9704709D0 (sv) * | 1997-12-17 | 1997-12-17 | Astra Ab | Pharmaceutically active compounds |
| SE9903759D0 (sv) * | 1999-10-18 | 1999-10-18 | Astra Ab | Pharmaceutically active compounds |
| SE0101324D0 (sv) * | 2001-04-12 | 2001-04-12 | Astrazeneca Ab | New process |
-
2001
- 2001-04-12 SE SE0101324A patent/SE0101324D0/xx unknown
-
2002
- 2002-04-12 CA CA002443475A patent/CA2443475A1/en not_active Abandoned
- 2002-04-12 CN CNB028115759A patent/CN1267435C/zh not_active Expired - Fee Related
- 2002-04-12 JP JP2002581445A patent/JP4248880B2/ja not_active Expired - Fee Related
- 2002-04-12 IL IL15824902A patent/IL158249A0/xx unknown
- 2002-04-12 AU AU2002249748A patent/AU2002249748B2/en not_active Ceased
- 2002-04-12 ES ES02718766T patent/ES2233809T3/es not_active Expired - Lifetime
- 2002-04-12 EP EP02718766A patent/EP1385850B1/en not_active Expired - Lifetime
- 2002-04-12 US US10/474,593 patent/US7169921B2/en not_active Expired - Fee Related
- 2002-04-12 NZ NZ528515A patent/NZ528515A/en unknown
- 2002-04-12 PT PT02718766T patent/PT1385850E/pt unknown
- 2002-04-12 MX MXPA03009211A patent/MXPA03009211A/es active IP Right Grant
- 2002-04-12 WO PCT/SE2002/000727 patent/WO2002083690A1/en not_active Ceased
- 2002-04-12 BR BR0208861-4A patent/BR0208861A/pt not_active IP Right Cessation
- 2002-04-12 DE DE60202203T patent/DE60202203T2/de not_active Expired - Lifetime
- 2002-04-12 KR KR1020037013158A patent/KR100848613B1/ko not_active Expired - Fee Related
- 2002-04-12 AT AT02718766T patent/ATE284405T1/de not_active IP Right Cessation
-
2003
- 2003-10-01 ZA ZA200307676A patent/ZA200307676B/en unknown
- 2003-10-02 IL IL158249A patent/IL158249A/en not_active IP Right Cessation
- 2003-10-09 NO NO20034526A patent/NO20034526L/no not_active Application Discontinuation
-
2006
- 2006-12-19 US US11/612,826 patent/US20070197519A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US7169921B2 (en) | 2007-01-30 |
| ATE284405T1 (de) | 2004-12-15 |
| HK1060886A1 (en) | 2004-08-27 |
| IL158249A0 (en) | 2004-05-12 |
| EP1385850A1 (en) | 2004-02-04 |
| EP1385850B1 (en) | 2004-12-08 |
| SE0101324D0 (sv) | 2001-04-12 |
| AU2002249748B2 (en) | 2008-02-28 |
| CN1267435C (zh) | 2006-08-02 |
| ES2233809T3 (es) | 2005-06-16 |
| MXPA03009211A (es) | 2004-01-29 |
| KR100848613B1 (ko) | 2008-07-28 |
| IL158249A (en) | 2009-09-01 |
| PT1385850E (pt) | 2005-03-31 |
| NZ528515A (en) | 2005-06-24 |
| KR20030087065A (ko) | 2003-11-12 |
| NO20034526D0 (no) | 2003-10-09 |
| NO20034526L (no) | 2003-10-31 |
| JP2004533432A (ja) | 2004-11-04 |
| WO2002083690A1 (en) | 2002-10-24 |
| CA2443475A1 (en) | 2002-10-24 |
| CN1520417A (zh) | 2004-08-11 |
| DE60202203T2 (de) | 2005-12-15 |
| JP4248880B2 (ja) | 2009-04-02 |
| US20070197519A1 (en) | 2007-08-23 |
| ZA200307676B (en) | 2004-07-13 |
| US20040181060A1 (en) | 2004-09-16 |
| DE60202203D1 (de) | 2005-01-13 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE 10A. ANUIDADE(S). |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2144 DE 07/02/2012. |