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BR0208628A - Processo para produzir compostos de truncamida a - Google Patents

Processo para produzir compostos de truncamida a

Info

Publication number
BR0208628A
BR0208628A BR0208628-0A BR0208628A BR0208628A BR 0208628 A BR0208628 A BR 0208628A BR 0208628 A BR0208628 A BR 0208628A BR 0208628 A BR0208628 A BR 0208628A
Authority
BR
Brazil
Prior art keywords
truncamide
compounds
producing
cycloheptapeptides
trunkamide
Prior art date
Application number
BR0208628-0A
Other languages
English (en)
Inventor
Fernando Albericio Palomera
Josep Maria Caba Naudi
Ernest Giralt Lledo
Ignacio Manzanares
Ignacio Rodrigues
Original Assignee
Pharma Mar Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharma Mar Sa filed Critical Pharma Mar Sa
Publication of BR0208628A publication Critical patent/BR0208628A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"PROCESSO PARA PRODUZIR COMPOSTOS DE TRUNCAMIDA A". Truncamida A e outros cicloheptapeptídeos podem ser fabricados por síntese em fase sólida de um precursor linear.
BR0208628-0A 2001-04-02 2002-04-02 Processo para produzir compostos de truncamida a BR0208628A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0108234.6A GB0108234D0 (en) 2001-04-02 2001-04-02 Process for producing trunkamide A compounds
PCT/GB2002/001527 WO2002081506A1 (en) 2001-04-02 2002-04-02 Process for producing trunkamide a compounds

Publications (1)

Publication Number Publication Date
BR0208628A true BR0208628A (pt) 2004-08-10

Family

ID=9912086

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0208628-0A BR0208628A (pt) 2001-04-02 2002-04-02 Processo para produzir compostos de truncamida a

Country Status (14)

Country Link
US (1) US7531506B2 (pt)
EP (1) EP1373305B1 (pt)
JP (1) JP4249488B2 (pt)
AT (1) ATE327248T1 (pt)
AU (1) AU2002251221B8 (pt)
BR (1) BR0208628A (pt)
CA (1) CA2443207A1 (pt)
DE (1) DE60211671T2 (pt)
ES (1) ES2265494T3 (pt)
GB (1) GB0108234D0 (pt)
IL (1) IL158145A0 (pt)
MX (1) MXPA03009008A (pt)
NZ (1) NZ528532A (pt)
WO (1) WO2002081506A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070264023A1 (en) * 2006-04-26 2007-11-15 Virgin Islands Microsystems, Inc. Free space interchip communications
NZ583284A (en) 2007-08-17 2012-04-27 Novartis Ag Cyclic depsipeptides from isolated chondromyces crocatus useful as inhibitors of kallikrein 7 and human neutrophil elastase
US8680054B2 (en) 2011-04-20 2014-03-25 Novartis Ag Suspension type topical formulations comprising cyclic depsipeptide
US8614289B2 (en) 2011-04-20 2013-12-24 Novartis Ag Processes for the manufacture of macrocyclic depsipeptides and new intermediates
US8987413B2 (en) 2012-10-09 2015-03-24 Novartis Ag Aldehyde acetal based processes for the manufacture of macrocyclic depsipeptides and new intermediates
US9067978B2 (en) 2012-10-09 2015-06-30 Novartis Ag Solution phase processes for the manufacture of macrocyclic depsipeptides and new intermediates
JOP20190254A1 (ar) 2017-04-27 2019-10-27 Pharma Mar Sa مركبات مضادة للأورام

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9608010D0 (en) * 1996-04-18 1996-06-19 Pharma Mar Sa Trunkamide A
AU3301997A (en) 1996-06-10 1998-01-07 Board Of Trustees Of The Leland Stanford Junior University Total synthesis of bacitracin polypetides

Also Published As

Publication number Publication date
JP4249488B2 (ja) 2009-04-02
CA2443207A1 (en) 2002-10-17
DE60211671D1 (de) 2006-06-29
US20050014684A1 (en) 2005-01-20
JP2004534746A (ja) 2004-11-18
AU2002251221B8 (en) 2008-05-15
MXPA03009008A (es) 2004-02-17
ES2265494T3 (es) 2007-02-16
IL158145A0 (en) 2004-03-28
DE60211671T2 (de) 2007-05-10
EP1373305B1 (en) 2006-05-24
EP1373305A1 (en) 2004-01-02
US7531506B2 (en) 2009-05-12
WO2002081506A8 (en) 2003-12-11
AU2002251221B2 (en) 2007-11-08
GB0108234D0 (en) 2001-05-23
NZ528532A (en) 2005-03-24
ATE327248T1 (de) 2006-06-15
WO2002081506A1 (en) 2002-10-17

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]