BG107865A - Substituted pyridoindoles as serotonin agonists and antagonists - Google Patents
Substituted pyridoindoles as serotonin agonists and antagonistsInfo
- Publication number
- BG107865A BG107865A BG107865A BG10786503A BG107865A BG 107865 A BG107865 A BG 107865A BG 107865 A BG107865 A BG 107865A BG 10786503 A BG10786503 A BG 10786503A BG 107865 A BG107865 A BG 107865A
- Authority
- BG
- Bulgaria
- Prior art keywords
- disorders
- compounds
- antagonists
- serotonin agonists
- certain
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/16—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/16—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/16—Peri-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Child & Adolescent Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25674000P | 2000-12-20 | 2000-12-20 | |
| PCT/US2001/049371 WO2002059129A2 (en) | 2000-12-20 | 2001-12-19 | Substituted tetracyclic pyridoindoles as serotonin agonists and antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG107865A true BG107865A (en) | 2004-07-30 |
Family
ID=22973405
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG107865A BG107865A (en) | 2000-12-20 | 2003-05-30 | Substituted pyridoindoles as serotonin agonists and antagonists |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US6699852B2 (no) |
| EP (1) | EP1343791A2 (no) |
| JP (1) | JP4231290B2 (no) |
| KR (1) | KR20030070073A (no) |
| BG (1) | BG107865A (no) |
| BR (1) | BR0116429A (no) |
| CA (1) | CA2432185C (no) |
| EE (1) | EE200300296A (no) |
| HU (1) | HUP0303432A3 (no) |
| IL (1) | IL156354A0 (no) |
| IS (1) | IS6849A (no) |
| MX (1) | MXPA03005438A (no) |
| NO (1) | NO20032797L (no) |
| PL (1) | PL366233A1 (no) |
| RU (1) | RU2003121304A (no) |
| SK (1) | SK7042003A3 (no) |
| WO (1) | WO2002059129A2 (no) |
| ZA (1) | ZA200304305B (no) |
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| US5328905A (en) | 1987-07-20 | 1994-07-12 | Duphar International Research B.V. | 8,9-anellated-1,2,3,4-tetrahydro-β-carboline derivatives |
| EP0300541B1 (en) | 1987-07-20 | 1996-03-27 | Duphar International Research B.V | 8,9-anellated-1,2,3,4-tetrahydro-beta-carboline derivatives |
| JPH02180885A (ja) | 1988-09-01 | 1990-07-13 | Glaxo Group Ltd | ラクタム誘導体 |
| US5223625A (en) | 1988-12-22 | 1993-06-29 | Duphar International Research B.V. | Annelated indolo [3,2,-C]lactams |
| CA2011107A1 (en) | 1990-02-28 | 1991-08-31 | David E. Bays | Lactam derivatives |
| CA2174543A1 (en) | 1993-10-20 | 1995-04-27 | Nobuyuki Yasuda | Indole derivative |
| AR023574A1 (es) | 1999-04-23 | 2002-09-04 | Pharmacia & Upjohn Co Llc | Compuestos de azepinindol tetraciclico,composiciones farmaceuticas y el uso de dichos compuestos para preparar un medicamento, e intermediarios |
| US6407092B1 (en) * | 1999-04-23 | 2002-06-18 | Pharmacia & Upjohn Company | Tetracyclic azepinoindole compounds |
| IL147108A0 (en) * | 1999-06-15 | 2002-08-14 | Du Pont Pharm Co | Substituted heterocycle fused gamma-carbolines |
-
2001
- 2001-12-19 IL IL15635401A patent/IL156354A0/xx unknown
- 2001-12-19 US US10/026,611 patent/US6699852B2/en not_active Expired - Lifetime
- 2001-12-19 PL PL01366233A patent/PL366233A1/xx unknown
- 2001-12-19 EE EEP200300296A patent/EE200300296A/xx unknown
- 2001-12-19 MX MXPA03005438A patent/MXPA03005438A/es unknown
- 2001-12-19 WO PCT/US2001/049371 patent/WO2002059129A2/en not_active Ceased
- 2001-12-19 BR BRPI0116429-5A patent/BR0116429A/pt unknown
- 2001-12-19 EP EP01994316A patent/EP1343791A2/en not_active Withdrawn
- 2001-12-19 SK SK704-2003A patent/SK7042003A3/sk unknown
- 2001-12-19 HU HU0303432A patent/HUP0303432A3/hu not_active Application Discontinuation
- 2001-12-19 KR KR10-2003-7008272A patent/KR20030070073A/ko not_active Withdrawn
- 2001-12-19 JP JP2002559431A patent/JP4231290B2/ja not_active Expired - Lifetime
- 2001-12-19 RU RU2003121304/04A patent/RU2003121304A/ru not_active Application Discontinuation
- 2001-12-19 CA CA2432185A patent/CA2432185C/en not_active Expired - Lifetime
-
2003
- 2003-05-30 BG BG107865A patent/BG107865A/xx unknown
- 2003-06-02 ZA ZA200304305A patent/ZA200304305B/en unknown
- 2003-06-18 IS IS6849A patent/IS6849A/is unknown
- 2003-06-19 NO NO20032797A patent/NO20032797L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CA2432185A1 (en) | 2002-08-01 |
| CA2432185C (en) | 2011-11-08 |
| PL366233A1 (en) | 2005-01-24 |
| HUP0303432A3 (en) | 2012-09-28 |
| US20020173503A1 (en) | 2002-11-21 |
| BR0116429A (pt) | 2006-05-09 |
| IS6849A (is) | 2003-06-18 |
| WO2002059129A2 (en) | 2002-08-01 |
| KR20030070073A (ko) | 2003-08-27 |
| WO2002059129A3 (en) | 2003-01-30 |
| EE200300296A (et) | 2003-12-15 |
| NO20032797L (no) | 2003-08-19 |
| ZA200304305B (en) | 2004-09-02 |
| SK7042003A3 (en) | 2004-07-07 |
| JP2005506281A (ja) | 2005-03-03 |
| HUP0303432A2 (hu) | 2004-01-28 |
| US6699852B2 (en) | 2004-03-02 |
| NO20032797D0 (no) | 2003-06-19 |
| EP1343791A2 (en) | 2003-09-17 |
| RU2003121304A (ru) | 2005-01-27 |
| MXPA03005438A (es) | 2004-05-05 |
| JP4231290B2 (ja) | 2009-02-25 |
| IL156354A0 (en) | 2004-01-04 |
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