BE801079A - 2-(heteroaryl-methyl)-5,9 beta-dialcoyl-6,7-benzomorphanes et leurs sels d'addition avec des acides - Google Patents

2-(heteroaryl-methyl)-5,9 beta-dialcoyl-6,7-benzomorphanes et leurs sels d'addition avec des acides

Info

Publication number: BE801079A
Authority: BE; Belgium
Prior art keywords: dialcoyl; benzomorphanes; heteroaryl; beta; acids
Prior art date: 1972-06-19

Application number

BE132406A

Other languages

English (en)

Original Assignee

Boehringer Sohn Ingelheim

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1972-06-19

Filing date

1973-06-18

Publication date

1973-12-18

1973-06-18 Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim

1973-12-18 Publication of BE801079A publication Critical patent/BE801079A/fr

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/14—Antitussive agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurosurgery (AREA)
Epidemiology (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Psychiatry (AREA)
Addiction (AREA)
Pulmonology (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Other In-Based Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Steroid Compounds (AREA)

BE132406A 1972-06-19 1973-06-18 2-(heteroaryl-methyl)-5,9 beta-dialcoyl-6,7-benzomorphanes et leurs sels d'addition avec des acides BE801079A (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE2229695A DE2229695A1 (de)	1972-06-19	1972-06-19	2-(heteroaryl-methyl)-5,9 beta-dialkyl6,7-benzomorphane, deren saeureadditionssalze sowie verfahren zu deren herstellung

Publications (1)

Publication Number	Publication Date
BE801079A true BE801079A (fr)	1973-12-18

Family

ID=5848060

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BE132406A BE801079A (fr)	1972-06-19	1973-06-18	2-(heteroaryl-methyl)-5,9 beta-dialcoyl-6,7-benzomorphanes et leurs sels d'addition avec des acides

Country Status (13)

Country	Link
US (1)	US3931194A (fr)
JP (1)	JPS5711908B2 (fr)
AT (6)	AT328627B (fr)
BE (1)	BE801079A (fr)
CH (9)	CH582698A5 (fr)
DE (1)	DE2229695A1 (fr)
DK (1)	DK136904C (fr)
ES (8)	ES416037A1 (fr)
FR (1)	FR2189056B1 (fr)
GB (1)	GB1433817A (fr)
NL (1)	NL7308483A (fr)
NO (1)	NO137694C (fr)
SE (1)	SE405121B (fr)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2437610A1 (de) *	1974-08-05	1976-02-26	Boehringer Sohn Ingelheim	Neue 5,9-beta-disubstituierte 2-tetrahydrofurfuryl-6,7-benzomorphane, deren saeureadditionssalze, ihre verwendung als arzneimittel und verfahren zu deren herstellung
GB1575009A (en) *	1976-06-21	1980-09-17	Acf Chemiefarma Nv	6,7-benzomorphan derivatives
JPS63177704A (ja) *	1987-01-16	1988-07-21	松山株式会社	農作業機連結装置
AR067673A1 (es)	2007-07-26	2009-10-21	Vitae Pharmaceuticals Inc	Derivados de 1,3 oxazinan - 2 - ona como inhibidores ciclicos de la 11 beta -hidroxiesteroide deshidrogenasa 1. composiciones farmaceuticas.
AR069545A1 (es) *	2007-11-16	2010-02-03	Boehringer Ingelheim Pharma	Derivados de aril y heteroarilcarbonilo de benzomorfanos y estructuras relacionadas, composiciones farmaceuticas que contienen dichos compuestos, obtencion de las mismas, su uso en el tratamiento de enfermedades mediadas por la inhibicion de la enzima 11beta-hidroxiesteroide deshidrogenasa (hsd) 1 y
US8440658B2 (en)	2007-12-11	2013-05-14	Vitae Pharmaceuticals, Inc.	Cyclic urea inhibitors of 11β-hydroxysteroid dehydrogenase 1
TW200934490A (en)	2008-01-07	2009-08-16	Vitae Pharmaceuticals Inc	Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
JP5490020B2 (ja)	2008-01-24	2014-05-14	ヴァイティーファーマシューティカルズ，インコーポレイテッド	１１β−ヒドロキシステロイドデヒドロゲナーゼ１の環状カルバゼート及びセミカルバジドインヒビター
EP2245014B1 (fr) *	2008-02-12	2011-11-02	Boehringer Ingelheim International GmbH	Derives d'uree de benzomorphanes et structures associees, medicaments contenant de tels composes et leur utilisation
WO2009102460A2 (fr)	2008-02-15	2009-08-20	Vitae Pharmaceuticals, Inc.	Inhibiteurs de 11beta-hydroxystéroïde deshydrogénase 1
WO2009134392A1 (fr)	2008-05-01	2009-11-05	Vitae Pharmaceuticals, Inc.	Inhibiteurs cycliques de la 11-bêta-hydroxystéroïde déhydrogénase 1
WO2009134387A1 (fr)	2008-05-01	2009-11-05	Vitae Pharmaceuticals, Inc.	Inhibiteurs cycliques de la 11-bêta-hydroxystéroïde déhydrogénase 1
MX2010011935A (es)	2008-05-01	2011-05-19	Vitae Pharmaceuticals Inc	Inhibidores ciclicos de 11 beta-hidroxiesteroide deshidrogenasa 1.
JP5711115B2 (ja)	2008-05-13	2015-04-30	ベーリンガーインゲルハイムインターナショナルゲゼルシャフトミットベシュレンクテルハフツング	ベンゾモルファン及び関連骨格のアリサイクリックカルボン酸誘導体、そのような化合物を含有する医薬及びその使用
NZ590495A (en)	2008-07-25	2012-10-26	Vitae Pharmaceuticals Inc	Dihydropyridin-phenyl-3-oxazinan-2-ones as inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2324017B1 (fr)	2008-07-25	2014-12-31	Boehringer Ingelheim International GmbH	INHIBITEURS DE LA 11 bêta-HYDROXYSTÉROÏDE DÉSHYDROGÉNASE 1
UA109255C2 (ru)	2009-04-30	2015-08-10	Берінгер Інгельхайм Інтернешнл Гмбх	Циклические ингибиторы 11бета-гидроксистероиддегидрогеназы 1
EP2440537A1 (fr)	2009-06-11	2012-04-18	Vitae Pharmaceuticals, Inc.	Inhibiteurs cycliques de la 11-bêta-hydroxystéroïde déshydrogénase 1 basée sur la structure 1,3-oxazinan-2-one
TWI531571B (zh) *	2009-11-06	2016-05-01	維它藥物公司	六氫茚并吡啶及八氫苯并喹啉之芳基－及雜芳基羰基衍生物
WO2011159760A1 (fr)	2010-06-16	2011-12-22	Vitae Pharmaceuticals, Inc.	Hétérocycles à 5, 6 et 7 chaînons substitués, médicaments contenant ces composés et leur utilisation
TWI537258B (zh)	2010-11-05	2016-06-11	百靈佳殷格翰國際股份有限公司	六氫茚并吡啶及八氫苯并喹啉之芳基－及雜環芳基羰基衍生物
EP2744783A1 (fr)	2011-08-17	2014-06-25	Boehringer Ingelheim International GmbH	Dérivés d'indénopyridine

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE582575A (fr) *	1958-09-22
FR1281227A (fr) *	1958-09-22	1962-01-12	Smith Kline French Lab	Perfectionnements apportés aux procédés pour la préparation de dérivés d'aralcoylbenzomorphane
CS166803B2 (fr) *	1971-02-08	1976-03-29	Boehringer Sohn Ingelheim
SE392895B (sv) *	1971-08-24	1977-04-25	Sumitomo Chemical Co	Forfarande for framstellning av bensomorfanderivat och deras salter

1972
- 1972-06-19 DE DE2229695A patent/DE2229695A1/de not_active Withdrawn
1973
- 1973-06-05 US US05/367,114 patent/US3931194A/en not_active Expired - Lifetime
- 1973-06-06 AT AT489474*7A patent/AT328627B/de not_active IP Right Cessation
- 1973-06-06 AT AT490074*7A patent/AT328629B/de not_active IP Right Cessation
- 1973-06-06 AT AT494373A patent/AT325218B/de not_active IP Right Cessation
- 1973-06-06 AT AT489874*7A patent/AT329199B/de not_active IP Right Cessation
- 1973-06-06 AT AT489774*7A patent/AT328628B/de not_active IP Right Cessation
- 1973-06-06 AT AT489974*7A patent/AT329200B/de not_active IP Right Cessation
- 1973-06-14 CH CH1041376A patent/CH582698A5/xx not_active IP Right Cessation
- 1973-06-14 CH CH1041476A patent/CH589649A5/xx not_active IP Right Cessation
- 1973-06-14 CH CH1041076A patent/CH583230A5/xx not_active IP Right Cessation
- 1973-06-14 CH CH1041276A patent/CH589648A5/xx not_active IP Right Cessation
- 1973-06-14 CH CH864373A patent/CH583227A5/xx not_active IP Right Cessation
- 1973-06-14 CH CH1040876A patent/CH583228A5/xx not_active IP Right Cessation
- 1973-06-14 CH CH1041576A patent/CH583231A5/xx not_active IP Right Cessation
- 1973-06-14 CH CH1040976A patent/CH583229A5/xx not_active IP Right Cessation
- 1973-06-14 CH CH1041176A patent/CH582697A5/xx not_active IP Right Cessation
- 1973-06-18 JP JP6863473A patent/JPS5711908B2/ja not_active Expired
- 1973-06-18 SE SE7308564A patent/SE405121B/xx unknown
- 1973-06-18 DK DK336173A patent/DK136904C/da active
- 1973-06-18 NO NO2518/73A patent/NO137694C/no unknown
- 1973-06-18 ES ES416037A patent/ES416037A1/es not_active Expired
- 1973-06-18 GB GB2886973A patent/GB1433817A/en not_active Expired
- 1973-06-18 BE BE132406A patent/BE801079A/fr unknown
- 1973-06-19 NL NL7308483A patent/NL7308483A/xx not_active Application Discontinuation
- 1973-06-19 FR FR7322249A patent/FR2189056B1/fr not_active Expired
1974
- 1974-10-30 ES ES431512A patent/ES431512A1/es not_active Expired
- 1974-10-30 ES ES431511A patent/ES431511A1/es not_active Expired
- 1974-10-30 ES ES0431516A patent/ES431516A1/es not_active Expired
- 1974-10-30 ES ES431514A patent/ES431514A1/es not_active Expired
- 1974-10-30 ES ES431510A patent/ES431510A1/es not_active Expired
- 1974-10-30 ES ES431513A patent/ES431513A1/es not_active Expired
- 1974-10-30 ES ES431515A patent/ES431515A1/es not_active Expired

Also Published As

Publication number	Publication date
AT325218B (de)	1975-10-10
US3931194A (en)	1976-01-06
FR2189056A1 (fr)	1974-01-25
NL7308483A (fr)	1973-12-21
CH583229A5 (fr)	1976-12-31
ATA489874A (de)	1975-07-15
AT329200B (de)	1976-04-26
ES416037A1 (es)	1976-02-16
CH583227A5 (fr)	1976-12-31
CH589649A5 (fr)	1977-07-15
AU5704673A (en)	1974-12-19
AT328629B (de)	1976-03-25
CH583230A5 (fr)	1976-12-31
JPS5711908B2 (fr)	1982-03-08
ES431513A1 (es)	1976-11-01
ES431510A1 (es)	1976-11-01
ES431516A1 (es)	1976-11-16
AT328628B (de)	1976-03-25
CH589648A5 (fr)	1977-07-15
ES431514A1 (es)	1976-11-01
SE405121B (sv)	1978-11-20
ES431515A1 (es)	1976-11-01
ATA489474A (de)	1975-06-15
JPS4961170A (fr)	1974-06-13
ES431511A1 (es)	1976-11-01
ES431512A1 (es)	1976-11-01
CH583228A5 (fr)	1976-12-31
DE2229695A1 (de)	1974-01-31
AT328627B (de)	1976-03-25
CH583231A5 (fr)	1976-12-31
GB1433817A (en)	1976-04-28
NO137694C (no)	1978-04-05
FR2189056B1 (fr)	1976-10-22
AT329199B (de)	1976-04-26
CH582698A5 (fr)	1976-12-15
ATA489974A (de)	1975-07-15
CH582697A5 (fr)	1976-12-15
NO137694B (no)	1977-12-27
ATA490074A (de)	1975-06-15
DK136904C (da)	1978-06-26
DK136904B (da)	1977-12-12
ATA489774A (de)	1975-06-15

Publication	Publication Date	Title
BE801079A (fr)	1973-12-18	2-(heteroaryl-methyl)-5,9 beta-dialcoyl-6,7-benzomorphanes et leurs sels d'addition avec des acides
FR3548M (fr)	1965-09-20	Thioxanthenesulfamides substitués, et leurs sels d'addition avec des acides.
NL167295C (nl)	1981-12-16	Grondbewerkingsmachine.
CH549931A (de)	1974-06-14	Bodenbearbeitungsmaschine.
CH555315A (fr)	1974-10-31	Procede de preparation d'alkyl- et cycloalkylthiophenylalkylaminoalkanols et leurs sels.
BE787683A (fr)	1973-02-19	2-phenylimino-imidazolidines, leurs sels d'addition avec des acides et procedes pour les fabriquer
NL178644B (nl)	1985-12-02	Grondbewerkingsmachine.
DK136067C (da)	1978-01-09	Herbicidt virksomme tetrahydro-1,3,5-triazin-2,6-dioner
NL167573B (nl)	1981-08-17	Grondbewerkingsmachine.
BE779582A (fr)	1972-08-18	N-(furylmethyl)-morphinanes, leurs sels d'addition avec des acides et procedes pour les fabriquer
BE786028A (fr)	1973-01-08	2,3-dihydro-oxo-imidazo(1,2-a)-pyrimidines, leurs sels d'addition avec des acides et procedes pour les fabriquer
DK130969B (da)	1975-05-12	1-Aminosulfonyl-2-aminobenzimidazoler med fungicid virkning.
DK130970B (da)	1975-05-12	1-Acyl-3-aminosulfonyl-2-imino-benzimidazoliner med fungicid virkning.
BE796086A (fr)	1973-08-28	Tube d'injection de vapeur.
DK139911B (da)	1979-05-14	6-Amino-s-triazindioner med herbicid virkning.
NL168680B (nl)	1981-12-16	Grondbewerkingsmachine.
DK133776C (da)	1976-12-06	Herbicidt aktive n,n'-tetrasubstituerede urinstoffer
NL169541C (nl)	1982-08-02	Landbouwwerktuig.
BE806392A (fr)	1974-02-15	Coprecipites d'aspirine/the
CH546330A (de)	1974-02-28	Viehstallung.
CH548733A (de)	1974-05-15	Viehselbsttraenkebecken.
BE804928A (fr)	1974-01-16	Terpolymeres de styrene, d'un nitrile et d'un acide
DK138640B (da)	1978-10-09	Cyclopropancarboxylsyrederivater med insekticid virkning.
NO136210C (no)	1977-08-03	Cellulosesubstrat med forbedret v}tstyrke.
CH556661A (fr)	1974-12-13	Distributeur d'essuie-mains.