AU2001281989A1 - Novel heteroaryl derivatives and use thereof as anti-tumour agents - Google Patents

Novel heteroaryl derivatives and use thereof as anti-tumour agents

Info

Publication number: AU2001281989A1
Authority: AU; Australia
Prior art keywords: tumour agents; heteroaryl derivatives; novel heteroaryl; novel; tumour
Prior art date: 2000-07-21
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2001281989A

Other versions

AU2001281989B2 (en

Inventor

Peter Emig

Eckhard Gunther

Bernhard Kutscher

Bernd Nickel

Jurgen Schmidt

Anita Storch

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Aeterna Zentaris GmbH

Original Assignee

Zentaris AG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-07-21

Filing date

2001-07-18

Publication date

2002-05-02

2000-07-21 Priority claimed from DE10035908A external-priority patent/DE10035908A1/en

2001-07-18 Application filed by Zentaris AG filed Critical Zentaris AG

2002-05-02 Publication of AU2001281989A1 publication Critical patent/AU2001281989A1/en

2004-09-30 Assigned to ZENTARIS GMBH reassignment ZENTARIS GMBH Request for Assignment Assignors: ZENTARIS AG

2005-05-12 Application granted granted Critical

2005-05-12 Publication of AU2001281989B2 publication Critical patent/AU2001281989B2/en

2021-07-18 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Links

AU2001281989A 2000-07-21 2001-07-18 Novel heteroaryl derivatives and use thereof as anti-tumour agents Ceased AU2001281989B2 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE10035908.6		2000-07-21
DE10035908A DE10035908A1 (en)	2000-07-21	2000-07-21	New heteroaryl derivatives and their use as medicines
PCT/EP2001/008262 WO2002008190A2 (en)	2000-07-21	2001-07-18	Novel heteroaryl derivatives and use thereof as anti-tumour agents

Publications (2)

Publication Number	Publication Date
AU2001281989A1 true AU2001281989A1 (en)	2002-05-02
AU2001281989B2 AU2001281989B2 (en)	2005-05-12

Family

ID=7649970

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU2001281989A Ceased AU2001281989B2 (en)	2000-07-21	2001-07-18	Novel heteroaryl derivatives and use thereof as anti-tumour agents
AU8198901A Pending AU8198901A (en)	2000-07-21	2001-07-18	Novel heteroaryl derivatives and use thereof as medicaments

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
AU8198901A Pending AU8198901A (en)	2000-07-21	2001-07-18	Novel heteroaryl derivatives and use thereof as medicaments

Country Status (21)

Country	Link
US (1)	US6638935B2 (en)
EP (1)	EP1305289A2 (en)
JP (1)	JP2004516243A (en)
KR (1)	KR20030015894A (en)
CN (1)	CN1447796A (en)
AR (1)	AR032467A1 (en)
AU (2)	AU2001281989B2 (en)
BG (1)	BG107506A (en)
BR (1)	BR0112711A (en)
CA (1)	CA2353353A1 (en)
DE (1)	DE10035908A1 (en)
HU (1)	HUP0300743A2 (en)
IL (1)	IL153931A0 (en)
MX (1)	MXPA03000596A (en)
NO (1)	NO20030302L (en)
NZ (1)	NZ524156A (en)
PL (1)	PL361354A1 (en)
RU (1)	RU2003105238A (en)
SK (1)	SK1942003A3 (en)
WO (1)	WO2002008190A2 (en)
ZA (1)	ZA200300545B (en)

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US8592409B2 (en)	2008-01-24	2013-11-26	Vitae Pharmaceuticals, Inc.	Cyclic carbazate and semicarbazide inhibitors of 11β-hydroxysteroid dehydrogenase 1
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CA2715290A1 (en) *	2008-02-15	2009-08-20	Vitae Pharmaceuticals, Inc.	Inhibitors of 11beta-hydroxysteroid dehydrogenase 1
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JP5538365B2 (en)	2008-05-01	2014-07-02	ヴァイティーファーマシューティカルズ，インコーポレイテッド	Cyclic inhibitor of 11β-hydroxysteroid dehydrogenase 1
US8242111B2 (en) *	2008-05-01	2012-08-14	Vitae Pharmaceuticals, Inc.	Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1
EP2291371B1 (en)	2008-05-01	2015-06-10	Vitae Pharmaceuticals, Inc.	Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8569337B2 (en)	2008-07-23	2013-10-29	Vertex Pharmaceuticals Incorporated	Tri-cyclic pyrazolopyridine kinase inhibitors
AU2009274023A1 (en)	2008-07-23	2010-01-28	Vertex Pharmaceuticals Incorporated	Tri-cyclic pyrazolopyridine kinase inhibitors
KR20110039563A (en)	2008-07-23	2011-04-19	버텍스 파마슈티칼스 인코포레이티드	Pyrazolopyridine Kinase Inhibitor
WO2010127237A2 (en) *	2009-04-30	2010-11-04	Boehringer Ingelheim International Gmbh	Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2324017B1 (en)	2008-07-25	2014-12-31	Boehringer Ingelheim International GmbH	INHIBITORS OF 11beta-HYDROXYSTEROID DEHYDROGENASE 1
CN104327062A (en)	2008-07-25	2015-02-04	贝林格尔·英格海姆国际有限公司	Cyclic Inhibitors of 11Beta-Hydroxysteroid Dehydrogenase 1
MX2011001319A (en)	2008-08-06	2011-04-05	Vertex Pharma	Aminopyridine kinase inhibitors.
US8637505B2 (en)	2009-02-04	2014-01-28	Boehringer Ingelheim International Gmbh	Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
TW201039034A (en) *	2009-04-27	2010-11-01	Chunghwa Picture Tubes Ltd	Pixel structure and the method of forming the same
US8680093B2 (en)	2009-04-30	2014-03-25	Vitae Pharmaceuticals, Inc.	Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
AU2010245914A1 (en)	2009-05-06	2011-12-15	Vertex Pharmaceuticals Incorporated	Pyrazolopyridines
US8927539B2 (en)	2009-06-11	2015-01-06	Vitae Pharmaceuticals, Inc.	Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1 based on the 1,3-oxazinan-2-one structure
US8883778B2 (en)	2009-07-01	2014-11-11	Vitae Pharmaceuticals, Inc.	Cyclic inhibitors of 11 beta-hydroxysteroid dehydrogenase 1
US9067932B2 (en)	2010-01-27	2015-06-30	Vertex Pharmaceuticals Incorporated	Pyrazolopyridine kinase inhibitors
AU2011209651A1 (en)	2010-01-27	2012-08-09	Vertex Pharmaceuticals Incorporated	Pyrazolopyrimidine kinase inhibitors
EP2550272A1 (en)	2010-01-27	2013-01-30	Vertex Pharmaceuticals Incorporated	Pyrazolopyrazine kinase inhibitors
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EP2585444B1 (en)	2010-06-25	2014-10-22	Boehringer Ingelheim International GmbH	Azaspirohexanones as inhibitors of 11-beta-hsd1 for the treatment of metabolic disorders
CA2813671A1 (en)	2010-11-02	2012-05-10	Boehringer Ingelheim International Gmbh	Pharmaceutical combinations for the treatment of metabolic disorders

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WO1999043682A1 (en) *	1998-02-26	1999-09-02	Neurogen Corporation	2-(het-)aryl-4-(cyclic amino substituted) heteroaryl fused pyridine derivatives, their preparation and their use as (ant-)agonists for gaba (a) brain receptors
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2000
- 2000-07-21 DE DE10035908A patent/DE10035908A1/en not_active Withdrawn
2001
- 2001-07-18 WO PCT/EP2001/008262 patent/WO2002008190A2/en not_active Ceased
- 2001-07-18 NZ NZ524156A patent/NZ524156A/en unknown
- 2001-07-18 MX MXPA03000596A patent/MXPA03000596A/en unknown
- 2001-07-18 EP EP01960509A patent/EP1305289A2/en not_active Withdrawn
- 2001-07-18 AU AU2001281989A patent/AU2001281989B2/en not_active Ceased
- 2001-07-18 JP JP2002514097A patent/JP2004516243A/en not_active Withdrawn
- 2001-07-18 BR BR0112711-0A patent/BR0112711A/en not_active IP Right Cessation
- 2001-07-18 KR KR10-2003-7000880A patent/KR20030015894A/en not_active Withdrawn
- 2001-07-18 SK SK194-2003A patent/SK1942003A3/en not_active Application Discontinuation
- 2001-07-18 IL IL15393101A patent/IL153931A0/en unknown
- 2001-07-18 PL PL36135401A patent/PL361354A1/en unknown
- 2001-07-18 AU AU8198901A patent/AU8198901A/en active Pending
- 2001-07-18 CN CN01814312A patent/CN1447796A/en active Pending
- 2001-07-18 HU HU0300743A patent/HUP0300743A2/en unknown
- 2001-07-18 RU RU2003105238/04A patent/RU2003105238A/en not_active Application Discontinuation
- 2001-07-20 AR ARP010103479A patent/AR032467A1/en unknown
- 2001-07-20 US US09/910,139 patent/US6638935B2/en not_active Expired - Fee Related
- 2001-07-20 CA CA002353353A patent/CA2353353A1/en not_active Abandoned
2002
- 2002-01-21 ZA ZA200300545A patent/ZA200300545B/en unknown
2003
- 2003-01-20 NO NO20030302A patent/NO20030302L/en unknown
- 2003-01-30 BG BG107506A patent/BG107506A/en unknown

Publication	Publication Date	Title
AU2001281989A1 (en)	2002-05-02	Novel heteroaryl derivatives and use thereof as anti-tumour agents
IL153931A0 (en)	2003-07-31	Novel heteroaryl derivatives and use thereof as anti-tumour agents
AU2002226486A1 (en)	2002-07-08	Novel c-glycoside derivatives and use thereof
AU2001279757A1 (en)	2002-05-02	Novel heteroaryl derivatives and the use thereof as pharmaceuticals
AU2001289675A1 (en)	2002-05-02	Novel Heteroaryl Derivatives and the Use Thereof as Pharmaceuticals
AU2001294814A1 (en)	2002-04-08	Pumpcn compositions and uses thereof
AU2002226487A1 (en)	2002-07-08	Novel c-glycoside derivatives and use thereof
AU2001250875A1 (en)	2001-10-15	Anti-microbial and immunostimulating composition
AU2001277754A1 (en)	2002-05-23	Proline derivatives and use thereof as drugs
IL153476A0 (en)	2003-07-06	Novel heteroaryl derivatives and the use thereof as pharmaceuticals
IL153361A0 (en)	2003-07-06	Novel heteroaryl derivatives and the use thereof as pharmaceuticals
AU2002219135A1 (en)	2002-06-18	Substituted 2-anilino-benzimidazoles and the use thereof as NHE-inhibitors
AU2001234313A1 (en)	2001-09-03	Novel phenylheteroalkylamine derivatives
AU4432001A (en)	2001-10-08	Trityl-type compounds and their use
AU2002338989A1 (en)	2003-05-08	Substituted C-furan-2-yl-methylamine and C-thiophen-2-yl-methylamine derivatives
AUPR099200A0 (en)	2000-11-16	New formulation
AU2001232080A1 (en)	2001-09-17	Compound, compositions and use
AU2001282268A1 (en)	2002-02-18	Phenantridine derivatives and their use as anti-telomerase agent
AU2002219846A1 (en)	2002-05-27	Novel use
AU2001288484A1 (en)	2002-03-13	Novel metallotexaphyrin derivatives
AU2002251543A1 (en)	2003-04-17	Novel atisane compound and use thereof
AU2001284465A1 (en)	2002-03-22	Tetraphenylporphyrin derivatives and compositions comprising the same
AU6042601A (en)	2001-11-20	Compounds and their uses
AU2002307237A1 (en)	2002-10-08	Carboxybenzopyran derivatives and compositions
AU2002306336A1 (en)	2003-01-02	Novel isoxazolopyridone derivatives and use thereof