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AU2001279757A1 - Novel heteroaryl derivatives and the use thereof as pharmaceuticals - Google Patents

Novel heteroaryl derivatives and the use thereof as pharmaceuticals

Info

Publication number
AU2001279757A1
AU2001279757A1 AU2001279757A AU2001279757A AU2001279757A1 AU 2001279757 A1 AU2001279757 A1 AU 2001279757A1 AU 2001279757 A AU2001279757 A AU 2001279757A AU 2001279757 A AU2001279757 A AU 2001279757A AU 2001279757 A1 AU2001279757 A1 AU 2001279757A1
Authority
AU
Australia
Prior art keywords
pharmaceuticals
heteroaryl derivatives
novel heteroaryl
novel
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU2001279757A
Other versions
AU2001279757B2 (en
Inventor
Peter Emig
Eckhard Gunther
Bernhard Kutscher
Bernd Nickel
Jurgen Schmidt
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aeterna Zentaris GmbH
Original Assignee
Zentaris AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10035928A external-priority patent/DE10035928A1/en
Application filed by Zentaris AG filed Critical Zentaris AG
Publication of AU2001279757A1 publication Critical patent/AU2001279757A1/en
Assigned to ZENTARIS GMBH reassignment ZENTARIS GMBH Request for Assignment Assignors: ZENTARIS AG
Application granted granted Critical
Publication of AU2001279757B2 publication Critical patent/AU2001279757B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

AU2001279757A 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals Ceased AU2001279757B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10035928A DE10035928A1 (en) 2000-07-21 2000-07-21 New heteroaryl derivatives and their use as medicines
DE10035928.0 2000-07-21
PCT/EP2001/008261 WO2002008192A1 (en) 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals

Publications (2)

Publication Number Publication Date
AU2001279757A1 true AU2001279757A1 (en) 2002-05-02
AU2001279757B2 AU2001279757B2 (en) 2005-05-26

Family

ID=7649980

Family Applications (2)

Application Number Title Priority Date Filing Date
AU7975701A Pending AU7975701A (en) 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals
AU2001279757A Ceased AU2001279757B2 (en) 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AU7975701A Pending AU7975701A (en) 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals

Country Status (23)

Country Link
US (5) US6890926B2 (en)
EP (1) EP1305290A1 (en)
JP (1) JP2004504381A (en)
KR (1) KR20030022287A (en)
CN (1) CN1443171A (en)
AR (1) AR033678A1 (en)
AU (2) AU7975701A (en)
BG (1) BG107508A (en)
BR (1) BR0112589A (en)
CA (1) CA2353369A1 (en)
CZ (1) CZ2003415A3 (en)
DE (1) DE10035928A1 (en)
HU (1) HUP0300838A2 (en)
IL (1) IL153361A0 (en)
MX (1) MXPA02012565A (en)
NO (1) NO20030298L (en)
NZ (1) NZ524154A (en)
PL (1) PL358788A1 (en)
RU (1) RU2265602C2 (en)
SK (1) SK1842003A3 (en)
TW (1) TWI228505B (en)
WO (1) WO2002008192A1 (en)
ZA (1) ZA200210180B (en)

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JP2005537258A (en) * 2002-07-17 2005-12-08 ツェンタリス ゲゼルシャフト ミット ベシュレンクテル ハフツング Novel anthracene derivatives and their use as pharmaceuticals
AU2004218260A1 (en) * 2003-01-28 2004-09-16 Aventis Pharma S.A. N-aryl heteroaromatic products, compositions containing same and use thereof
FR2855825B1 (en) * 2003-06-04 2008-08-22 Aventis Pharma Sa ARYL-HETEROAROMATIC PRODUCTS, COMPOSITIONS CONTAINING SAME AND USE THEREOF
AR044586A1 (en) * 2003-06-04 2005-09-21 Aventis Pharma Sa ARIL PRODUCTS - HETEROAROMATICOS, COMPOSITIONS THAT CONTAIN THEM AND THEIR USE
US7723362B2 (en) * 2004-01-08 2010-05-25 Syngenta Crop Protection, Inc. Pesticidal heterocyclic dihaloallyl compounds
DE102004003428A1 (en) * 2004-01-23 2005-08-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg New long-acting beta-2 agonists, and their use as pharmaceuticals
FR2871157A1 (en) * 2004-06-04 2005-12-09 Aventis Pharma Sa BIARYL AROMATIC PRODUCTS, COMPOSITIONS CONTAINING SAME AND USE THEREOF
CN1830964B (en) * 2005-03-11 2011-06-15 中国科学院上海药物研究所 4-Substituting anilino-3-nitroquinoline compounds, prepn. method and use thereof
EP2468747B1 (en) * 2006-12-07 2014-09-03 China Medical University 2-Selenophene-4-quinolones as anticancer agents
US8835426B2 (en) * 2007-02-26 2014-09-16 Vitae Pharmaceuticals, Inc. Cyclic urea and carbamate inhibitors of 11β-hydroxysteroid dehydrogenase 1
CL2008002199A1 (en) * 2007-07-26 2009-10-23 Vitae Pharmaceuticals Inc Compounds derived from 1,3-oxazin-2-one; pharmaceutical composition comprising said compounds; and use to treat a disease associated with the activity of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-hsd1) such as dyslipidemia, hyperlipidemia, hypertension, obesity and cardiovascular disease, among others.
AR069207A1 (en) * 2007-11-07 2010-01-06 Vitae Pharmaceuticals Inc CYCLIC UREAS AS INHIBITORS OF THE 11 BETA - HIDROXI-ESTEROIDE DESHIDROGENASA 1
CA2708303A1 (en) 2007-12-11 2009-06-18 Vitae Pharmaceuticals, Inc. Cyclic urea inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1
TW200934490A (en) * 2008-01-07 2009-08-16 Vitae Pharmaceuticals Inc Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
US8592409B2 (en) * 2008-01-24 2013-11-26 Vitae Pharmaceuticals, Inc. Cyclic carbazate and semicarbazide inhibitors of 11β-hydroxysteroid dehydrogenase 1
EP2252598A2 (en) * 2008-02-11 2010-11-24 Vitae Pharmaceuticals, Inc. 1,3-oxazepan-2-one and 1,3-diazepan-2-one inhibitors of 11beta-hydroxysteroid dehydrogenase 1
CA2715290A1 (en) * 2008-02-15 2009-08-20 Vitae Pharmaceuticals, Inc. Inhibitors of 11beta-hydroxysteroid dehydrogenase 1
WO2009117109A1 (en) * 2008-03-18 2009-09-24 Vitae Pharmaceuticals, Inc. Inhibitors of 11beta-hydroxysteroid dehydrogenase type 1
EP2291371B1 (en) 2008-05-01 2015-06-10 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8242111B2 (en) * 2008-05-01 2012-08-14 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1
JP5538365B2 (en) 2008-05-01 2014-07-02 ヴァイティー ファーマシューティカルズ，インコーポレイテッド Cyclic inhibitor of 11β-hydroxysteroid dehydrogenase 1
TW200946520A (en) * 2008-05-01 2009-11-16 Vitae Pharmaceuticals Inc Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
WO2010127237A2 (en) * 2009-04-30 2010-11-04 Boehringer Ingelheim International Gmbh Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2324017B1 (en) 2008-07-25 2014-12-31 Boehringer Ingelheim International GmbH INHIBITORS OF 11beta-HYDROXYSTEROID DEHYDROGENASE 1
CN104327062A (en) 2008-07-25 2015-02-04 贝林格尔·英格海姆国际有限公司 Cyclic Inhibitors of 11Beta-Hydroxysteroid Dehydrogenase 1
US8637505B2 (en) 2009-02-04 2014-01-28 Boehringer Ingelheim International Gmbh Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
TW201039034A (en) * 2009-04-27 2010-11-01 Chunghwa Picture Tubes Ltd Pixel structure and the method of forming the same
US8680093B2 (en) 2009-04-30 2014-03-25 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8927539B2 (en) 2009-06-11 2015-01-06 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1 based on the 1,3-oxazinan-2-one structure
US8883778B2 (en) 2009-07-01 2014-11-11 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11 beta-hydroxysteroid dehydrogenase 1
US8933072B2 (en) 2010-06-16 2015-01-13 Vitae Pharmaceuticals, Inc. Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use
EP2585444B1 (en) 2010-06-25 2014-10-22 Boehringer Ingelheim International GmbH Azaspirohexanones as inhibitors of 11-beta-hsd1 for the treatment of metabolic disorders
CA2813671A1 (en) 2010-11-02 2012-05-10 Boehringer Ingelheim International Gmbh Pharmaceutical combinations for the treatment of metabolic disorders
JP7471818B2 (en) * 2016-08-18 2024-04-22 ヴィダック ファーマ リミテッド Piperazine derivatives, pharmaceutical compositions, and methods of use thereof

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AU646519B2 (en) 1990-10-10 1994-02-24 Schering Corporation Pyridine and pyridine N-oxide derivatives of diaryl methyl piperidines or piperazines, and compositions and methods of use thereof
EP0703905A1 (en) * 1993-06-18 1996-04-03 Merck & Co. Inc. Inhibitors of farnesyl-protein transferase
JP4176148B2 (en) 1996-05-20 2008-11-05 帝人ファーマ株式会社 Diarylalkyl cyclic diamine derivatives and their use as therapeutics
DE69738949D1 (en) * 1996-05-20 2008-10-09 Darwin Discovery Ltd CHINOLINE CARBOXAMIDES AS TNF INHIBITORS AND AS PDE IV INHIBITORS
SK27598A3 (en) * 1996-06-29 1998-11-04 Samjin Pharm Co Ltd Piperazine derivatives and process for the preparation thereof
US5861395A (en) 1996-09-13 1999-01-19 Schering Corporation Compounds useful for inhibition of farnesyl proteins transferase
FR2753706B1 (en) 1996-09-20 1998-10-30 NOVEL N-SUBSTITUTED CYCLIC AMINES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
DK0957100T3 (en) * 1997-07-07 2005-01-31 Kowa Co Diamond derivatives and pharmaceutical preparations containing the same
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US6410540B1 (en) * 1998-08-28 2002-06-25 Scios, Inc. Inhibitors of p38-αkinase
WO2000051614A1 (en) 1999-03-03 2000-09-08 Merck & Co., Inc. Inhibitors of prenyl-protein transferases
DE10035927A1 (en) * 2000-07-21 2002-03-07 Asta Medica Ag New heteroaryl derivatives and their use as medicines
US6610274B1 (en) * 2000-12-22 2003-08-26 Wallace J. Gardner Anti-inflammatory composition comprising tetracycline

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