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AU2001266689A1 - 4-benzyl-2-hydroxy-1,4-oxazin-3-one and polymorphic forms thereof - Google Patents

4-benzyl-2-hydroxy-1,4-oxazin-3-one and polymorphic forms thereof

Info

Publication number
AU2001266689A1
AU2001266689A1 AU2001266689A AU6668901A AU2001266689A1 AU 2001266689 A1 AU2001266689 A1 AU 2001266689A1 AU 2001266689 A AU2001266689 A AU 2001266689A AU 6668901 A AU6668901 A AU 6668901A AU 2001266689 A1 AU2001266689 A1 AU 2001266689A1
Authority
AU
Australia
Prior art keywords
oxazin
benzyl
hydroxy
polymorphic forms
polymorphic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001266689A
Inventor
Karel M. Jos Brands
Louis S. Crocker
Todd D Nelson
Philip J. Pye
Jonathan D. Rosen
Kai Rossen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of AU2001266689A1 publication Critical patent/AU2001266689A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • C07D265/32—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings with oxygen atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2001266689A 2000-06-08 2001-06-04 4-benzyl-2-hydroxy-1,4-oxazin-3-one and polymorphic forms thereof Abandoned AU2001266689A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US21025400P 2000-06-08 2000-06-08
US21020400P 2000-06-08 2000-06-08
US60210204 2000-06-08
US60210254 2000-06-08
PCT/US2001/018038 WO2001094322A1 (en) 2000-06-08 2001-06-04 4-benzyl-2-hydroxy-1,4-oxazin-3-one and polymorphic forms thereof

Publications (1)

Publication Number Publication Date
AU2001266689A1 true AU2001266689A1 (en) 2001-12-17

Family

ID=26904943

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001266689A Abandoned AU2001266689A1 (en) 2000-06-08 2001-06-04 4-benzyl-2-hydroxy-1,4-oxazin-3-one and polymorphic forms thereof

Country Status (4)

Country Link
US (1) US6538134B2 (en)
EP (1) EP1292582A1 (en)
AU (1) AU2001266689A1 (en)
WO (1) WO2001094322A1 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6861426B2 (en) * 2001-02-27 2005-03-01 Teva Pharmaceutical Industries Ltd. Crystal forms of lamotrigine and processes for their preparations
DE60312670T2 (en) * 2002-04-23 2007-12-06 Teva Pharmaceutical Industries Ltd. PHARMACEUTICAL COMPOSITION CONTAINING LAMOTRIGINE PARTICLES WITH DEFINED MORPHOLOGY
FR2953720B1 (en) * 2009-12-11 2012-05-11 Oreal USE OF BENZYLOXY ETHYLAMINE DERIVATIVES AS A CONSERVATIVE,
WO2012146692A1 (en) 2011-04-29 2012-11-01 Sandoz Ag Novel intermediates for the preparation of highly pure aprepitant or fosaprepitant
CN102675240B (en) 2012-04-13 2015-01-14 浙江海正药业股份有限公司 4-substitute-2-hydroxy morpholine-3-ketone and preparation method thereof
WO2019013244A1 (en) * 2017-07-13 2019-01-17 大正製薬株式会社 Method for producing (2s)-2-[(1h-pyrazol-1-yl)methyl]-1,3-oxazinane derivative
CN110483436B (en) * 2019-09-19 2021-07-16 西安凯立新材料股份有限公司 Method for preparing 4-benzyl-2-hydroxy-morpholine-3-one

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9819890D0 (en) * 1998-09-11 1998-11-04 Merck Sharp & Dohme Chemical synthesis

Also Published As

Publication number Publication date
US6538134B2 (en) 2003-03-25
WO2001094322A1 (en) 2001-12-13
US20020042510A1 (en) 2002-04-11
EP1292582A1 (en) 2003-03-19

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