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AU1606197A - Novel piperidine derivatives 4-substituted by an imidazolidin-2-on-1-yl-ethyl, tetrahydropyrimidin-2-on-1-yl-ethyl and 1,3-diazepin-2-on-1-yl-ethyl group, and use thereof as alpha2-adrenergic receptor antagonists - Google Patents

Novel piperidine derivatives 4-substituted by an imidazolidin-2-on-1-yl-ethyl, tetrahydropyrimidin-2-on-1-yl-ethyl and 1,3-diazepin-2-on-1-yl-ethyl group, and use thereof as alpha2-adrenergic receptor antagonists

Info

Publication number
AU1606197A
AU1606197A AU16061/97A AU1606197A AU1606197A AU 1606197 A AU1606197 A AU 1606197A AU 16061/97 A AU16061/97 A AU 16061/97A AU 1606197 A AU1606197 A AU 1606197A AU 1606197 A AU1606197 A AU 1606197A
Authority
AU
Australia
Prior art keywords
ethyl
tetrahydropyrimidin
diazepin
alpha2
imidazolidin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU16061/97A
Inventor
Michael Briley
Thierry Imbert
Marc Marien
Jean-Louis Vidaluc
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pierre Fabre Medicament SA
Original Assignee
Pierre Fabre Medicament SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pierre Fabre Medicament SA filed Critical Pierre Fabre Medicament SA
Publication of AU1606197A publication Critical patent/AU1606197A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU16061/97A 1996-02-01 1997-01-30 Novel piperidine derivatives 4-substituted by an imidazolidin-2-on-1-yl-ethyl, tetrahydropyrimidin-2-on-1-yl-ethyl and 1,3-diazepin-2-on-1-yl-ethyl group, and use thereof as alpha2-adrenergic receptor antagonists Abandoned AU1606197A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9601220A FR2744451B1 (en) 1996-02-01 1996-02-01 NOVEL IMIDAZOLIDINONES, PYRIMIDINONES, AND 1,3-DIAZEPIN-2 -ONES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATIONS
FR9601220 1996-02-01
PCT/FR1997/000179 WO1997028157A1 (en) 1996-02-01 1997-01-30 NOVEL PIPERIDINE DERIVATIVES 4-SUBSTITUTED BY AN IMIDAZOLIDIN-2-ON-1-YL-ETHYL, TETRAHYDROPYRIMIDIN-2-ON-1-YL-ETHYL AND 1,3-DIAZEPIN-2-ON-1-YL-ETHYL GROUP, AND USE THEREOF AS α2-ADRENERGIC RECEPTOR ANTAGONISTS

Publications (1)

Publication Number Publication Date
AU1606197A true AU1606197A (en) 1997-08-22

Family

ID=9488732

Family Applications (1)

Application Number Title Priority Date Filing Date
AU16061/97A Abandoned AU1606197A (en) 1996-02-01 1997-01-30 Novel piperidine derivatives 4-substituted by an imidazolidin-2-on-1-yl-ethyl, tetrahydropyrimidin-2-on-1-yl-ethyl and 1,3-diazepin-2-on-1-yl-ethyl group, and use thereof as alpha2-adrenergic receptor antagonists

Country Status (3)

Country Link
AU (1) AU1606197A (en)
FR (1) FR2744451B1 (en)
WO (1) WO1997028157A1 (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6133277A (en) * 1997-12-05 2000-10-17 Janssen Pharmaceutica N.V. (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
FR2789681A1 (en) * 1999-02-12 2000-08-18 Pf Medicament Benzodioxanyl azabicyclo-octane alkyl ureas and imidazolidones having alpha 2 adrenergic receptor antagonist activity
HRP20010868A2 (en) 1999-06-02 2003-04-30 Janssen Pharmaceutica Nv Aminoalkyl substituted (benzodioxan, benzofuran or benzopyran) derivatives
EA004648B1 (en) 1999-06-02 2004-06-24 Янссен Фармацевтика Н.В. Pyrrolidinyl, piperidinyl or homopiperidinyl substituted derivatives, process for preparing thereof, use thereof in medicine, pharmaceutical composition containing them and method for its preparation
FR2803298A1 (en) * 1999-12-30 2001-07-06 Adir NOVEL LINEAR OR CYCLIC UREAS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
AU2004202768B2 (en) * 1999-12-30 2007-04-05 Les Laboratoires Servier New linear or cyclic ureas, a process for their preparation and pharmaceutical compositions containing them
JO2352B1 (en) * 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for treating fundic disaccomodation
US20060052362A1 (en) * 2003-01-17 2006-03-09 Ryuichi Tozawa Skeletal muscle protecting agent
TWI457122B (en) * 2007-07-20 2014-10-21 Orion Corp 2,3-dihydrobenzo[1,4]dioxin-2-ylmethyl derivatives as alpha2c antagonists for use in the treatment of peripheric and central nervous system diseases

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2852945A1 (en) * 1978-12-07 1980-06-26 Boehringer Sohn Ingelheim Benzo:dioxanyl-hydroxyethyl-piperidyl-imidazolidone derivs. - having hypotensive activity, and prepd. by reacting a piperidin-4-yl-imidazolidinone with a halo-hydroxyethyl-benzodioxan
IL59619A0 (en) * 1979-03-28 1980-06-30 Pfizer Phthalazine derivatives,their preparation and pharmaceutical compositions containing them
JPS61215389A (en) * 1985-03-20 1986-09-25 Kyowa Hakko Kogyo Co Ltd Quinazoline derivative and cardiac containing same
NZ221485A (en) * 1986-08-28 1991-04-26 Merck & Co Inc Hexahydroarylquinolizine derivatives and pharmaceutical compositions
WO1992015301A1 (en) * 1991-03-01 1992-09-17 H. Lundbeck A/S Treatment of hypertension and peripheral vascular diseases
JPH09165385A (en) * 1994-08-26 1997-06-24 Kyowa Hakko Kogyo Co Ltd Quinazoline derivatives

Also Published As

Publication number Publication date
FR2744451B1 (en) 1998-04-24
WO1997028157A1 (en) 1997-08-07
FR2744451A1 (en) 1997-08-08

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