AR224997A1 - METHOD FOR PREPARING 5-BENZOIL OR SUBSTITUTED 5-BENZOIL 1,2-DIHYDRO-3H-PIRROLO (1,2-A) PIRROL-1-CARBOXILICOS - Google Patents

METHOD FOR PREPARING 5-BENZOIL OR SUBSTITUTED 5-BENZOIL 1,2-DIHYDRO-3H-PIRROLO (1,2-A) PIRROL-1-CARBOXILICOS

Info

Publication number: AR224997A1
Authority: AR; Argentina
Prior art keywords: benzoil; carboxilicos; pirrol; pirrolo; dihydro
Prior art date: 1976-07-14

Application number

AR268356A

Other languages

Spanish (es)

Original Assignee

Syntex Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-07-14

Filing date

1977-07-07

Publication date

1982-02-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR224997(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1977-02-23 Priority claimed from US05/771,286 external-priority patent/US4089969A/en

1977-07-07 Application filed by Syntex Inc filed Critical Syntex Inc

1982-02-15 Application granted granted Critical

1982-02-15 Publication of AR224997A1 publication Critical patent/AR224997A1/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pain & Pain Management (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Rheumatology (AREA)
Urology & Nephrology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)

AR268356A 1976-07-14 1977-07-07 METHOD FOR PREPARING 5-BENZOIL OR SUBSTITUTED 5-BENZOIL 1,2-DIHYDRO-3H-PIRROLO (1,2-A) PIRROL-1-CARBOXILICOS AR224997A1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US70490976A	1976-07-14	1976-07-14
US05/771,286 US4089969A (en)	1976-07-14	1977-02-23	5-Aroyl-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof

Publications (1)

Publication Number	Publication Date
AR224997A1 true AR224997A1 (en)	1982-02-15

Family

ID=27107410

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AR268356A AR224997A1 (en)	1976-07-14	1977-07-07	METHOD FOR PREPARING 5-BENZOIL OR SUBSTITUTED 5-BENZOIL 1,2-DIHYDRO-3H-PIRROLO (1,2-A) PIRROL-1-CARBOXILICOS

Country Status (27)

Country	Link
JP (1)	JPS539788A (en)
AR (1)	AR224997A1 (en)
CA (1)	CA1102809A (en)
CH (3)	CH641458A5 (en)
CS (1)	CS204954B2 (en)
DE (2)	DE2731678A1 (en)
DK (1)	DK151886C (en)
ES (2)	ES460706A1 (en)
FI (1)	FI63406C (en)
FR (2)	FR2358406A1 (en)
GB (1)	GB1554075A (en)
GR (1)	GR61111B (en)
HK (1)	HK15981A (en)
HU (1)	HU174224B (en)
IE (1)	IE45253B1 (en)
IL (2)	IL52493A (en)
IT (1)	IT1117313B (en)
MX (1)	MX163202B (en)
MY (1)	MY8100357A (en)
NL (2)	NL186318C (en)
NO (1)	NO147564C (en)
NZ (1)	NZ184610A (en)
PL (4)	PL109390B1 (en)
PT (1)	PT66780B (en)
SE (1)	SE434643B (en)
SU (1)	SU695558A3 (en)
YU (1)	YU40816B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4140698A (en) *	1977-07-25	1979-02-20	Syntex (Usa) Inc.	1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
JPS55124633A (en) *	1979-03-19	1980-09-25	Sohachi Takeuchi	Manufacturing method of tubular vessel
US4344943A (en) *	1980-06-09	1982-08-17	Syntex (U.S.A.) Inc.	6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof
US4353829A (en) *	1980-11-21	1982-10-12	Syntex (U.S.A.) Inc.	Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
US4511724A (en) *	1982-06-10	1985-04-16	Merck & Co., Inc.	5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents
JPS5910589A (en) *	1982-06-10	1984-01-20	メルク　エンド　カムパニー　インコーポレーテツド	Antiinflammatory and analgesic novel 5-(pyrrol-2-oyl)-1,2-dihydro-3h-pyrrolo(1,2-a) pyrrole derivative
US4874871A (en) *	1987-03-25	1989-10-17	Syntex (U.S.A.) Inc.	Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds
JPH0739418B2 (en) *	1987-09-10	1995-05-01	久光製薬株式会社	Novel 3-aroyl-6,7-dihydro-5H-pyrrolo [1,2-c] imidazole-7-carboxylic acid derivative
JP2649168B2 (en) *	1988-02-25	1997-09-03	久光製薬株式会社	Novel 5,6-diphenyl-1,2-dihydro-3H-pyrrolo [1,2-a] pyrrole-1-carboxylic acid derivatives
IT1250691B (en) *	1991-07-22	1995-04-21	Giancarlo Santus	THERAPEUTIC COMPOSITIONS FOR INTRANASAL ADMINISTRATION INCLUDING KETOROLAC.
ES2136093T3 (en) *	1991-11-11	1999-11-16	Hisamitsu Pharmaceutical Co	PROMOTION CONTAINING CETOROLAC.
DE4300697C1 (en) *	1993-01-13	1994-05-19	Roemmers Sa	New 2-pyrrolidino-ethyl ester of ketorolac - useful as analgesic, antiinflammatory and antipyretic agent with low ulcerogenicity
US5622948A (en) *	1994-12-01	1997-04-22	Syntex (U.S.A.) Inc.	Pyrrole pyridazine and pyridazinone anti-inflammatory agents
JP2008210666A (en) *	2007-02-27	2008-09-11	Okamura Corp	Lighting system in merchandise display shelf
KR20230131182A (en) *	2020-12-16	2023-09-12	뉴 프런티어 랩스 엘엘씨	Dicarboxylic acid esters to induce analgesic effects

1977
- 1977-05-17 JP JP5697777A patent/JPS539788A/en active Granted
- 1977-07-07 GR GR53907A patent/GR61111B/en unknown
- 1977-07-07 DK DK307577A patent/DK151886C/en active
- 1977-07-07 AR AR268356A patent/AR224997A1/en active
- 1977-07-08 NL NLAANVRAGE7707651,A patent/NL186318C/en not_active IP Right Cessation
- 1977-07-08 IE IE1423/77A patent/IE45253B1/en not_active IP Right Cessation
- 1977-07-08 IL IL52493A patent/IL52493A/en unknown
- 1977-07-08 PT PT66780A patent/PT66780B/en unknown
- 1977-07-08 CH CH850077A patent/CH641458A5/en not_active IP Right Cessation
- 1977-07-11 GB GB28919/77A patent/GB1554075A/en not_active Expired
- 1977-07-11 NZ NZ184610A patent/NZ184610A/en unknown
- 1977-07-11 FI FI772153A patent/FI63406C/en not_active IP Right Cessation
- 1977-07-11 FR FR7721356A patent/FR2358406A1/en active Granted
- 1977-07-11 YU YU1721/77A patent/YU40816B/en unknown
- 1977-07-12 CS CS774646A patent/CS204954B2/en unknown
- 1977-07-12 CA CA282,599A patent/CA1102809A/en not_active Expired
- 1977-07-13 DE DE19772731678 patent/DE2731678A1/en active Granted
- 1977-07-13 IT IT68630/77A patent/IT1117313B/en active Protection Beyond IP Right Term
- 1977-07-13 PL PL1977199603A patent/PL109390B1/en unknown
- 1977-07-13 PL PL1977227290A patent/PL124444B1/en unknown
- 1977-07-13 PL PL1977227291A patent/PL124445B1/en unknown
- 1977-07-13 SE SE7708141A patent/SE434643B/en not_active IP Right Cessation
- 1977-07-13 NO NO772494A patent/NO147564C/en unknown
- 1977-07-13 DE DE2760330A patent/DE2760330C2/de not_active Expired
- 1977-07-13 ES ES460706A patent/ES460706A1/en not_active Expired
- 1977-07-13 PL PL1977227289A patent/PL124711B1/en unknown
- 1977-07-13 SU SU772501050A patent/SU695558A3/en active
- 1977-07-14 HU HU77SI1582A patent/HU174224B/en unknown
- 1977-12-20 FR FR7738508A patent/FR2375234A1/en active Granted
1978
- 1978-05-24 ES ES470214A patent/ES470214A1/en not_active Expired
1979
- 1979-11-22 IL IL58779A patent/IL58779A0/en unknown
1981
- 1981-04-23 HK HK159/81A patent/HK15981A/en unknown
- 1981-12-30 MY MY357/81A patent/MY8100357A/en unknown
1984
- 1984-02-22 CH CH86584A patent/CH646972A5/en not_active IP Right Cessation
- 1984-02-22 CH CH86684A patent/CH646973A5/en not_active IP Right Cessation
1991
- 1991-07-05 MX MX9100104A patent/MX163202B/en unknown
1993
- 1993-03-23 NL NL930021C patent/NL930021I2/en unknown

Also Published As

Publication number	Publication date
PL124711B1 (en)	1983-02-28
CA1102809A (en)	1981-06-09
PL109390B1 (en)	1980-05-31
IL52493A0 (en)	1977-10-31
AU2697577A (en)	1979-01-18
CH646972A5 (en)	1984-12-28
ES460706A1 (en)	1978-12-01
IT1117313B (en)	1986-02-17
PL124444B1 (en)	1983-01-31
FI63406C (en)	1983-06-10
DE2731678C2 (en)	1989-06-08
GB1554075A (en)	1979-10-17
FR2358406A1 (en)	1978-02-10
NZ184610A (en)	1979-03-28
PL124445B1 (en)	1983-01-31
MX163202B (en)	1992-02-20
DK307577A (en)	1978-01-15
NO147564C (en)	1983-05-18
YU40816B (en)	1986-06-30
NL930021I1 (en)	1993-05-03
FR2358406B1 (en)	1981-04-17
NL930021I2 (en)	1997-03-03
DK151886C (en)	1988-06-06
JPS539788A (en)	1978-01-28
JPS6254109B2 (en)	1987-11-13
AU513384B2 (en)	1980-11-27
PT66780A (en)	1977-08-01
IE45253B1 (en)	1982-07-14
SU695558A3 (en)	1979-10-30
MY8100357A (en)	1981-12-31
IL58779A0 (en)	1980-02-29
HU174224B (en)	1979-11-28
CS204954B2 (en)	1981-04-30
NL186318C (en)	1990-11-01
FI772153A7 (en)	1978-01-15
YU172177A (en)	1983-09-30
FR2375234B1 (en)	1980-11-07
IL52493A (en)	1982-02-28
DE2760330C2 (en)	1989-06-15
PT66780B (en)	1978-12-18
CH641458A5 (en)	1984-02-29
NL186318B (en)	1990-06-01
DK151886B (en)	1988-01-11
ES470214A1 (en)	1979-09-16
GR61111B (en)	1978-09-12
SE7708141L (en)	1978-01-15
NO147564B (en)	1983-01-24
FR2375234A1 (en)	1978-07-21
PL199603A1 (en)	1978-04-24
FI63406B (en)	1983-02-28
DE2731678A1 (en)	1978-03-16
SE434643B (en)	1984-08-06
IE45253L (en)	1978-01-14
HK15981A (en)	1981-05-01
NO772494L (en)	1978-01-17
CH646973A5 (en)	1984-12-28
NL7707651A (en)	1978-01-17

Publication	Publication Date	Title
ES507715A0 (en)	1983-02-01	PROCEDURE FOR PREPARING 1-SULFO-2-OXOAZETIDINE DERIVATIVES.
ES508454A0 (en)	1983-08-01	PROCEDURE FOR PREPARING 2-AMINO-4-HYDROXY-QUINAZOLINE DERIVATIVES.
ES507126A0 (en)	1983-07-01	PROCEDURE FOR PREPARING PIRIDONA DERIVATIVES.
AR221887A1 (en)	1981-03-31	PROCEDURE FOR PREPARING 6-CYAN-4-4-PHENYL-2-ALKYL (C1-C4) 1,4-DIHYDROPYRIDINE COMPOUNDS
AR220684A1 (en)	1980-11-28	METHOD FOR THE PREPARATION OF 1-PHENYL-3-AZABICICLO (3.1.0) HEXANS
AR224997A1 (en)	1982-02-15	METHOD FOR PREPARING 5-BENZOIL OR SUBSTITUTED 5-BENZOIL 1,2-DIHYDRO-3H-PIRROLO (1,2-A) PIRROL-1-CARBOXILICOS
AR220892A1 (en)	1980-12-15	PROCEDURE FOR PREPARING (PIRIDAZINIL-3) -5-DITIOL-1,2 TIONA-3
AR220675A1 (en)	1980-11-28	PROCEDURE FOR THE PREPARATION OF SUBSTITUTED DERIVATIVES OF PIRIDO (1,2-A) PIRIMIDINAS
BG26949A4 (en)	1979-07-12	METHOD FOR OBTAINING 5,11-DIHYDRO-6H- PYRIDO(2,3-B)(1,4)BENZODIAZEPIN-6-ONES SUBSTITUTED IN THE 11TH POSITION
FI801033A7 (en)	1981-01-01	Method for the preparation of 2,6-diaminonebularins.
FI800314A7 (en)	1981-01-01	Method for the selective preparation of isosorbide-5-nitrate.
AR221732A1 (en)	1981-03-13	PROCEDURE FOR OBTAINING 2,6-DIALKYL-N- (PYRAZOLE OR 4,5-DIHALOIMIDAZOLMETIL) -2-HALO ACETANILIDAS
ES479189A0 (en)	1981-09-01	PROCEDURE FOR OBTAINING BENZ-ACILOBEN-ZIMIDAZOLE-2-CARBOXYLIC DERIVATIVES.
MX4499E (en)	1982-05-21	PROCEDURE FOR PREPARING 2-OXI-5-ISOPROPILIDEN-7-HYDROXI-9-SUBSTITUTED-2,6-METHANE-3,4,5,6-TETRAHYDRO-2H-1-BENZOXOCINES
MX5340E (en)	1983-06-27	PROCEDURE FOR PREPARING HEXAHYDRO DERIVATIVES 1,2,3,3A.4,5-OXO-6-6H-INDOLO (3,2,1-DE) NAFTIRIDINE
MX5194E (en)	1983-04-22	PROCEDURE FOR PREPARING 3-AMINOMETI-4-BETA-HIDROXI-8-BETA-ALCOXI-2,9-DIOXATRICICLO (4,3,1,03,7) DEAN
MX4697E (en)	1982-08-04	PROCEDURE FOR PREPARING 1,2,3-TIADIAZOLE-5-IL-UREAS
AR226853A1 (en)	1982-08-31	METHOD FOR PREPARING 1,2-DIHYDRO-2-OXO-5- (PIRIDINIL) -NICOTINONITRILS
AR228244A1 (en)	1983-02-15	PROCEDURE FOR PREPARING OCTAHIDRO-1H-PIRROLO- (2,3-G) ISOQUINOLIN-4-ONAS
MX5916E (en)	1984-08-24	IMPROVED PROCEDURE FOR PREPARING 7-CHLORINE-2-METHYL-3-3A-DIHYDRO-2H, 9H-ISOXAZOL (3,2-B) (1,3) BENZOXAZIN-9-ONA
MX4851E (en)	1982-11-01	PROCEDURE FOR OBTAINING 2,9-DIOXATRICICLO (4,3,1,03,7) DEAN
ES513070A0 (en)	1983-02-16	PROCEDURE FOR PREPARING BUTIROTIOLACTONES.
AR214527A1 (en)	1979-06-29	PROCEDURE FOR THE PREPARATION OF-N-6-CLORONICOTIONOIL-D, 1 HOMOCISTEIN THIOLACTONE
AR231640A1 (en)	1985-01-31	PROCEDURE FOR PREPARING CYCLOALCA 4,5 PYRROLLO 2,3-G-ISOQUINOLINAS
MX4815E (en)	1982-10-19	PROCEDURE FOR PREPARING 1,2 ', 6'-TRI-T-BUTOXICARBONIL-FORTIMICINA B