AR205402A1 - Procedimiento para la elaboracion de compuestos de 1-(5-sulfamoil - antraniloil) - piperazina - Google Patents
Procedimiento para la elaboracion de compuestos de 1-(5-sulfamoil - antraniloil) - piperazinaInfo
- Publication number
- AR205402A1 AR205402A1 AR260094A AR26009475A AR205402A1 AR 205402 A1 AR205402 A1 AR 205402A1 AR 260094 A AR260094 A AR 260094A AR 26009475 A AR26009475 A AR 26009475A AR 205402 A1 AR205402 A1 AR 205402A1
- Authority
- AR
- Argentina
- Prior art keywords
- antraniloil
- sulfamoil
- elaboration
- piperazine
- compounds
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
- GLUUGHFHXGJENI-UHFFFAOYSA-N diethylenediamine Natural products C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/205—Radicals derived from carbonic acid
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH764373 | 1973-05-28 | ||
| CH450774 | 1974-04-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR205402A1 true AR205402A1 (es) | 1976-04-30 |
Family
ID=25695649
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR260094A AR205402A1 (es) | 1973-05-28 | 1975-01-01 | Procedimiento para la elaboracion de compuestos de 1-(5-sulfamoil - antraniloil) - piperazina |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US3933802A (es) |
| JP (1) | JPS5019760A (es) |
| AR (1) | AR205402A1 (es) |
| AU (1) | AU6939974A (es) |
| DE (1) | DE2423847A1 (es) |
| DK (1) | DK285974A (es) |
| FR (1) | FR2231381A1 (es) |
| IL (1) | IL44864A0 (es) |
| LU (1) | LU70158A1 (es) |
| NL (1) | NL7406684A (es) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2611705A1 (de) * | 1976-03-18 | 1977-09-22 | Josef Dipl Chem Dr Rer N Klosa | N-5-(nitrofurfuryliden-)-1-amino- hydantoin enthaltende kristalloesungsmittel |
| US4268536A (en) * | 1978-12-07 | 1981-05-19 | Western Electric Company, Inc. | Method for depositing a metal on a surface |
| JPS56124740A (en) * | 1980-02-29 | 1981-09-30 | Mitsubishi Electric Corp | Bushing |
| GB8823775D0 (en) * | 1988-10-11 | 1988-11-16 | Scras | New 2-carbonyl substituted n n'-di-(trimethoxybenzoyl)piperazines |
| GB0030710D0 (en) * | 2000-12-15 | 2001-01-31 | Hoffmann La Roche | Piperazine derivatives |
| CA2537292C (en) * | 2003-09-09 | 2013-04-02 | F. Hoffmann-La Roche Ag | 1- (2-amino-benzol) -piperazine derivatives as glycine uptake inhibitors for the treatment of psychoses |
| RU2395502C2 (ru) * | 2004-12-09 | 2010-07-27 | Ф.Хоффманн-Ля Рош Аг | Производные фенил-пиперазин метанона |
| ES2338139T3 (es) * | 2004-12-15 | 2010-05-04 | F. Hoffmann-La Roche Ag | Fenil-metanonas bi- y triciclicas sustituidas como inhibidores del transportador de la glicina i (glyt-1) para el tratamiento de la enfermedad de alzheimer. |
| US7485637B2 (en) * | 2005-01-04 | 2009-02-03 | Hoffmann-La Roche Inc. | Benzoyl-tetrahydropiperidine derivatives |
| CA2593453A1 (en) * | 2005-01-06 | 2006-07-13 | F. Hoffmann-La Roche Ag | Sulfanyl substituted phenyl methanones as glycine transporter 1 (glyt-1) inhibitors for the treatment of neurological and neuropsychiatric disorders |
| ES2346335T3 (es) * | 2005-01-07 | 2010-10-14 | F. Hoffmann-La Roche Ag | Derivados de (4-(heteroaril)piperacin-1-il)-(fenil 2,5-sustituido)metanona como inhibidores del transportador de glicina 1 (glyt-1) para el tratamiento de trastornos neurologicos e neuropsiquiatricos. |
| CN101141959B (zh) * | 2005-01-18 | 2010-12-15 | 弗·哈夫曼-拉罗切有限公司 | 作为甘氨酸转运体1(GlyT-1)抑制剂用于治疗神经学和神经精神病学障碍的2,5-二取代的苯甲酮衍生物 |
| KR100915472B1 (ko) * | 2005-01-26 | 2009-09-03 | 에프. 호프만-라 로슈 아게 | 페닐 메탄온 유도체 및 그의 글라이신 트랜스포터 1억제제로서의 용도 |
| PT1848694E (pt) * | 2005-02-07 | 2010-02-02 | Hoffmann La Roche | Fenil-metanonas heterocíclicas substituídas, como inibidores do transportador de glicina 1 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2598E (fr) * | 1903-05-19 | 1904-05-20 | Joseph Francois Antoine Franci | Renforceur du bois pour cannes à peche, mats, vergues, manches et articles d'utilité et de jeux |
| US2910488A (en) * | 1958-01-22 | 1959-10-27 | Merck & Co Inc | Aniline derivatives |
| CH433378A (de) * | 1962-03-09 | 1967-04-15 | Ciba Geigy | Verfahren zur Herstellung neuer Anthranilsäurederivate |
-
1974
- 1974-05-16 DE DE2423847A patent/DE2423847A1/de active Pending
- 1974-05-17 NL NL7406684A patent/NL7406684A/xx unknown
- 1974-05-20 IL IL44864A patent/IL44864A0/xx unknown
- 1974-05-22 US US05/472,333 patent/US3933802A/en not_active Expired - Lifetime
- 1974-05-27 AU AU69399/74A patent/AU6939974A/en not_active Expired
- 1974-05-27 DK DK285974A patent/DK285974A/da unknown
- 1974-05-27 LU LU70158*A patent/LU70158A1/xx unknown
- 1974-05-27 FR FR7418225A patent/FR2231381A1/fr not_active Withdrawn
- 1974-05-28 JP JP49059409A patent/JPS5019760A/ja active Pending
-
1975
- 1975-01-01 AR AR260094A patent/AR205402A1/es active
Also Published As
| Publication number | Publication date |
|---|---|
| DK285974A (es) | 1975-01-20 |
| JPS5019760A (es) | 1975-03-01 |
| FR2231381A1 (es) | 1974-12-27 |
| DE2423847A1 (de) | 1975-01-02 |
| US3933802A (en) | 1976-01-20 |
| IL44864A0 (en) | 1975-02-10 |
| NL7406684A (es) | 1974-12-02 |
| LU70158A1 (es) | 1976-04-13 |
| AU6939974A (en) | 1975-11-27 |
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