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AR132159A1 - Anticuerpos anti-b7h3 y métodos de uso - Google Patents

Anticuerpos anti-b7h3 y métodos de uso

Info

Publication number
AR132159A1
AR132159A1 ARP240100660A ARP240100660A AR132159A1 AR 132159 A1 AR132159 A1 AR 132159A1 AR P240100660 A ARP240100660 A AR P240100660A AR P240100660 A ARP240100660 A AR P240100660A AR 132159 A1 AR132159 A1 AR 132159A1
Authority
AR
Argentina
Prior art keywords
antigen
antibody
seq
binding fragment
human
Prior art date
Application number
ARP240100660A
Other languages
English (en)
Inventor
Liang Qu
Yao Ding
Ya Zhang
Original Assignee
Beigene Switzerland Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beigene Switzerland Gmbh filed Critical Beigene Switzerland Gmbh
Publication of AR132159A1 publication Critical patent/AR132159A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/705Receptors; Cell surface antigens; Cell surface determinants
    • C07K14/70503Immunoglobulin superfamily
    • C07K14/70532B7 molecules, e.g. CD80, CD86
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2803Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against the immunoglobulin superfamily
    • C07K16/2827Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against the immunoglobulin superfamily against B7 molecules, e.g. CD80, CD86
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/22Immunoglobulins specific features characterized by taxonomic origin from camelids, e.g. camel, llama or dromedary
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/24Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/30Immunoglobulins specific features characterized by aspects of specificity or valency
    • C07K2317/31Immunoglobulins specific features characterized by aspects of specificity or valency multispecific
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/40Immunoglobulins specific features characterized by post-translational modification
    • C07K2317/41Glycosylation, sialylation, or fucosylation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/50Immunoglobulins specific features characterized by immunoglobulin fragments
    • C07K2317/56Immunoglobulins specific features characterized by immunoglobulin fragments variable (Fv) region, i.e. VH and/or VL
    • C07K2317/569Single domain, e.g. dAb, sdAb, VHH, VNAR or nanobody®
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/60Immunoglobulins specific features characterized by non-natural combinations of immunoglobulin fragments
    • C07K2317/64Immunoglobulins specific features characterized by non-natural combinations of immunoglobulin fragments comprising a combination of variable region and constant region components
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/73Inducing cell death, e.g. apoptosis, necrosis or inhibition of cell proliferation
    • C07K2317/732Antibody-dependent cellular cytotoxicity [ADCC]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/73Inducing cell death, e.g. apoptosis, necrosis or inhibition of cell proliferation
    • C07K2317/734Complement-dependent cytotoxicity [CDC]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/90Immunoglobulins specific features characterized by (pharmaco)kinetic aspects or by stability of the immunoglobulin
    • C07K2317/92Affinity (KD), association rate (Ka), dissociation rate (Kd) or EC50 value

Landscapes

  • Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Cell Biology (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

La presente divulgación proporciona anticuerpos o fragmentos de unión a antígeno de los mismos que se unen a 4Ig-B7H3 humana. Reivindicación 1: Un anticuerpo o fragmento de unión a antígeno del mismo que se une específicamente a 4Ig-B7H3 humana, comprendiendo el anticuerpo o fragmento de unión a antígeno del mismo: (1) una región variable de la cadena pesada (VH) que comprende (a) una HCDR1 (Región Determinante de la Complementariedad de la Cadena Pesada 1) de SEQ ID Nº 7, (b) una HCDR2 de SEQ ID Nº 8, y (c) una HCDR3 de SEQ ID Nº 9; o (2) una región variable de la cadena pesada que comprende (a) una HCDR1 de SEQ ID Nº 12, (b) una HCDR2 de SEQ ID Nº 13, y (c) una HCDR3 de SEQ ID Nº 14. Reivindicación 7: Un anticuerpo multiespecífico o fragmento de unión a antígeno del mismo que comprende al menos un primer dominio de unión a antígeno que se une específicamente a un primer antígeno tumoral humano (TAA), en donde el primer TAA es 4Ig-B7H3 humana y el primer dominio de unión a antígeno comprende el anticuerpo o fragmento de unión a antígeno del mismo de una cualquiera de las reivindicaciones anteriores; y al menos un segundo dominio de unión a antígeno que se une específicamente a un segundo TAA humano. Reivindicación 15: Una composición farmacéutica que comprende el anticuerpo o fragmento de unión a antígeno del mismo de una cualquiera de las reivindicaciones anteriores y un portador farmacéuticamente aceptable. Reivindicación 16: Un ácido nucleico aislado que codifica el anticuerpo o fragmento de unión a antígeno del mismo de una cualquiera de las reivindicaciones 1 a 14. Reivindicación 17: Un vector que comprende el ácido nucleico de la reivindicación 16. Reivindicación 18: Una célula huésped que comprende el ácido nucleico de la reivindicación 16 o el vector de la reivindicación 17. Reivindicación 19: Un proceso para producir un anticuerpo o fragmento de unión a antígeno del mismo que comprende cultivar la célula huésped de la reivindicación 18 y recuperar el anticuerpo o fragmento de anticuerpo del cultivo.
ARP240100660A 2023-03-17 2024-03-18 Anticuerpos anti-b7h3 y métodos de uso AR132159A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN2023082099 2023-03-17

Publications (1)

Publication Number Publication Date
AR132159A1 true AR132159A1 (es) 2025-05-28

Family

ID=92840909

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP240100660A AR132159A1 (es) 2023-03-17 2024-03-18 Anticuerpos anti-b7h3 y métodos de uso

Country Status (10)

Country Link
EP (1) EP4680643A1 (es)
KR (1) KR20250160360A (es)
CN (1) CN120958028A (es)
AR (1) AR132159A1 (es)
AU (1) AU2024237990A1 (es)
CO (1) CO2025013921A2 (es)
IL (1) IL323120A (es)
MX (1) MX2025010929A (es)
TW (1) TW202438527A (es)
WO (1) WO2024193450A1 (es)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110642948B (zh) * 2019-10-09 2021-06-29 达石药业(广东)有限公司 B7-h3纳米抗体、其制备方法及用途
AU2020370125A1 (en) * 2019-10-22 2022-05-19 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services High affinity nanobodies targeting B7H3 (CD276) for treating multiple solid tumors
WO2021097800A1 (en) * 2019-11-22 2021-05-27 Abl Bio Inc. Anti-pd-l1/anti-b7-h3 multispecific antibodies and uses thereof
CA3182602A1 (en) * 2020-06-26 2021-12-30 Taekyo PARK Antibody-drug conjugates comprising anti-b7-h3 antibodies
US12133890B2 (en) * 2021-07-01 2024-11-05 Ningbo T-Maximum Biopharmaceuticals Co., Ltd. Antigen-binding polypeptide targeting B7H3 and application thereof

Also Published As

Publication number Publication date
IL323120A (en) 2025-11-01
MX2025010929A (es) 2025-10-01
CN120958028A (zh) 2025-11-14
CO2025013921A2 (es) 2025-10-20
AU2024237990A1 (en) 2025-09-25
TW202438527A (zh) 2024-10-01
WO2024193450A9 (en) 2025-10-09
KR20250160360A (ko) 2025-11-12
WO2024193450A1 (en) 2024-09-26
EP4680643A1 (en) 2026-01-21

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