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AR130742A1 - Proceso para la preparación de derivados de aminopiridazina - Google Patents

Proceso para la preparación de derivados de aminopiridazina

Info

Publication number
AR130742A1
AR130742A1 ARP230102726A ARP230102726A AR130742A1 AR 130742 A1 AR130742 A1 AR 130742A1 AR P230102726 A ARP230102726 A AR P230102726A AR P230102726 A ARP230102726 A AR P230102726A AR 130742 A1 AR130742 A1 AR 130742A1
Authority
AR
Argentina
Prior art keywords
preparation
aminopyridazine derivatives
aminopyridazine
derivatives
formula
Prior art date
Application number
ARP230102726A
Other languages
English (en)
Inventor
Eran Fogler
Michael Grabarnick
Revanappa Vasantrao Galge
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of AR130742A1 publication Critical patent/AR130742A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16Halogen atoms or nitro radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Una composición que comprende un compuesto de fórmula (1) o una sal, N-óxido, tautómero o enantiómero de este, obtenido mediante el proceso de una cualquiera de las reivindicaciones 1 - 22, y al menos un compuesto adicional seleccionado entre: los compuestos del grupo de fórmulas (2), en donde: cada T es independientemente un grupo de la fórmula: (3).
ARP230102726A 2022-10-12 2023-10-12 Proceso para la preparación de derivados de aminopiridazina AR130742A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN202211058387 2022-10-12

Publications (1)

Publication Number Publication Date
AR130742A1 true AR130742A1 (es) 2025-01-15

Family

ID=88793001

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP230102726A AR130742A1 (es) 2022-10-12 2023-10-12 Proceso para la preparación de derivados de aminopiridazina

Country Status (9)

Country Link
US (1) US20250353832A1 (es)
EP (1) EP4602033A1 (es)
CN (1) CN120019046A (es)
AR (1) AR130742A1 (es)
CL (1) CL2025001083A1 (es)
CO (1) CO2025006035A2 (es)
MX (1) MX2025004369A (es)
PE (1) PE20251585A1 (es)
WO (1) WO2024079733A1 (es)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200633990A (en) * 2004-11-18 2006-10-01 Takeda Pharmaceuticals Co Amide compound
WO2013164730A1 (en) * 2012-05-04 2013-11-07 Pfizer Inc. Heterocyclic substituted hexahydropyrano [3,4-d] [1,3] thiazin- 2 -amine compounds as inhibitors of app, bace1 and bace 2.
WO2016128465A1 (en) * 2015-02-11 2016-08-18 Basilea Pharmaceutica Ag Substituted mono- and polyazanaphthalene derivatives and their use
WO2018082964A1 (en) 2016-11-04 2018-05-11 Basf Se Process for the production of pyridazinyl-amides in a one-pot synthesis
US10316021B2 (en) * 2016-11-28 2019-06-11 Pfizer Inc. Heteroarylphenoxy benzamide kappa opioid ligands

Also Published As

Publication number Publication date
CO2025006035A2 (es) 2025-07-28
MX2025004369A (es) 2025-05-02
US20250353832A1 (en) 2025-11-20
CL2025001083A1 (es) 2025-05-30
WO2024079733A1 (en) 2024-04-18
CN120019046A (zh) 2025-05-16
EP4602033A1 (en) 2025-08-20
PE20251585A1 (es) 2025-06-16

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