AR130742A1 - Proceso para la preparación de derivados de aminopiridazina - Google Patents
Proceso para la preparación de derivados de aminopiridazinaInfo
- Publication number
- AR130742A1 AR130742A1 ARP230102726A ARP230102726A AR130742A1 AR 130742 A1 AR130742 A1 AR 130742A1 AR P230102726 A ARP230102726 A AR P230102726A AR P230102726 A ARP230102726 A AR P230102726A AR 130742 A1 AR130742 A1 AR 130742A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparation
- aminopyridazine derivatives
- aminopyridazine
- derivatives
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/20—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Una composición que comprende un compuesto de fórmula (1) o una sal, N-óxido, tautómero o enantiómero de este, obtenido mediante el proceso de una cualquiera de las reivindicaciones 1 - 22, y al menos un compuesto adicional seleccionado entre: los compuestos del grupo de fórmulas (2), en donde: cada T es independientemente un grupo de la fórmula: (3).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN202211058387 | 2022-10-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR130742A1 true AR130742A1 (es) | 2025-01-15 |
Family
ID=88793001
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP230102726A AR130742A1 (es) | 2022-10-12 | 2023-10-12 | Proceso para la preparación de derivados de aminopiridazina |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20250353832A1 (es) |
| EP (1) | EP4602033A1 (es) |
| CN (1) | CN120019046A (es) |
| AR (1) | AR130742A1 (es) |
| CL (1) | CL2025001083A1 (es) |
| CO (1) | CO2025006035A2 (es) |
| MX (1) | MX2025004369A (es) |
| PE (1) | PE20251585A1 (es) |
| WO (1) | WO2024079733A1 (es) |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200633990A (en) * | 2004-11-18 | 2006-10-01 | Takeda Pharmaceuticals Co | Amide compound |
| WO2013164730A1 (en) * | 2012-05-04 | 2013-11-07 | Pfizer Inc. | Heterocyclic substituted hexahydropyrano [3,4-d] [1,3] thiazin- 2 -amine compounds as inhibitors of app, bace1 and bace 2. |
| WO2016128465A1 (en) * | 2015-02-11 | 2016-08-18 | Basilea Pharmaceutica Ag | Substituted mono- and polyazanaphthalene derivatives and their use |
| WO2018082964A1 (en) | 2016-11-04 | 2018-05-11 | Basf Se | Process for the production of pyridazinyl-amides in a one-pot synthesis |
| US10316021B2 (en) * | 2016-11-28 | 2019-06-11 | Pfizer Inc. | Heteroarylphenoxy benzamide kappa opioid ligands |
-
2023
- 2023-10-12 AR ARP230102726A patent/AR130742A1/es unknown
- 2023-10-12 PE PE2025000773A patent/PE20251585A1/es unknown
- 2023-10-12 US US19/119,542 patent/US20250353832A1/en active Pending
- 2023-10-12 WO PCT/IL2023/051070 patent/WO2024079733A1/en not_active Ceased
- 2023-10-12 EP EP23805699.8A patent/EP4602033A1/en active Pending
- 2023-10-12 CN CN202380072340.2A patent/CN120019046A/zh active Pending
-
2025
- 2025-04-10 CL CL2025001083A patent/CL2025001083A1/es unknown
- 2025-04-11 MX MX2025004369A patent/MX2025004369A/es unknown
- 2025-05-09 CO CONC2025/0006035A patent/CO2025006035A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CO2025006035A2 (es) | 2025-07-28 |
| MX2025004369A (es) | 2025-05-02 |
| US20250353832A1 (en) | 2025-11-20 |
| CL2025001083A1 (es) | 2025-05-30 |
| WO2024079733A1 (en) | 2024-04-18 |
| CN120019046A (zh) | 2025-05-16 |
| EP4602033A1 (en) | 2025-08-20 |
| PE20251585A1 (es) | 2025-06-16 |
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