AR130477A1 - Antagonistas de c5ar1 y sus usos - Google Patents
Antagonistas de c5ar1 y sus usosInfo
- Publication number
- AR130477A1 AR130477A1 ARP230102436A ARP230102436A AR130477A1 AR 130477 A1 AR130477 A1 AR 130477A1 AR P230102436 A ARP230102436 A AR P230102436A AR P230102436 A ARP230102436 A AR P230102436A AR 130477 A1 AR130477 A1 AR 130477A1
- Authority
- AR
- Argentina
- Prior art keywords
- c5ar1
- compounds
- antagonists
- receptor
- antagonize
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D475/00—Heterocyclic compounds containing pteridine ring systems
- C07D475/02—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
En la presente memoria se proporcionan compuestos que modulan (por ejemplo, antagonizan) el receptor para el componente 5a del complemento 1 (C5aR1), un receptor acoplado a la proteína G para C5a que se asocia con trastornos autoinmunitarios, inflamatorios y neurodegenerativos. Además, se proporcionan composiciones farmacéuticas y kits que comprenden los compuestos y los métodos para tratar enfermedades y trastornos relacionados con el C5aR1 con los compuestos en un sujeto, mediante la administración de los compuestos y/o las composiciones que se describen en la presente memoria. Un compuesto con la fórmula (1).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202263406501P | 2022-09-14 | 2022-09-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR130477A1 true AR130477A1 (es) | 2024-12-11 |
Family
ID=90275968
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP230102436A AR130477A1 (es) | 2022-09-14 | 2023-09-13 | Antagonistas de c5ar1 y sus usos |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP4587014A2 (es) |
| AR (1) | AR130477A1 (es) |
| TW (1) | TW202425978A (es) |
| WO (1) | WO2024059096A2 (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2025176748A1 (en) * | 2024-02-22 | 2025-08-28 | F. Hoffmann-La Roche Ag | Condensed pyrazines or pyrimidines als trem2 agoonists |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK1357111T3 (da) * | 2000-12-28 | 2009-11-02 | Shionogi & Co | 2-pyridonderivater med affinitet for cannabinoid type 2-receptor |
| KR20180026774A (ko) * | 2015-07-17 | 2018-03-13 | 후지필름 가부시키가이샤 | 질소-함유 헤테로시클릭 화합물 |
| CN113924296B (zh) * | 2019-05-31 | 2024-09-17 | 株式会社钟根堂 | 作为组蛋白脱乙酰酶6抑制剂的1,3,4-噁二唑衍生化合物及包含其的药物组合物 |
-
2023
- 2023-09-13 AR ARP230102436A patent/AR130477A1/es unknown
- 2023-09-13 EP EP23866136.7A patent/EP4587014A2/en active Pending
- 2023-09-13 TW TW112134871A patent/TW202425978A/zh unknown
- 2023-09-13 WO PCT/US2023/032581 patent/WO2024059096A2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| TW202425978A (zh) | 2024-07-01 |
| WO2024059096A2 (en) | 2024-03-21 |
| WO2024059096A3 (en) | 2024-04-25 |
| EP4587014A2 (en) | 2025-07-23 |
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