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AR123593A1 - Un proceso para la síntesis de compuestos antranílicos de ácido / amida e intermedios de los mismos - Google Patents

Un proceso para la síntesis de compuestos antranílicos de ácido / amida e intermedios de los mismos

Info

Publication number
AR123593A1
AR123593A1 ARP210102654A ARP210102654A AR123593A1 AR 123593 A1 AR123593 A1 AR 123593A1 AR P210102654 A ARP210102654 A AR P210102654A AR P210102654 A ARP210102654 A AR P210102654A AR 123593 A1 AR123593 A1 AR 123593A1
Authority
AR
Argentina
Prior art keywords
synthesis
intermediates
anthranilic acid
amide compounds
compound
Prior art date
Application number
ARP210102654A
Other languages
English (en)
Inventor
Suresh Kumar Sythana
Pramod Nagle
Vijay Kumar Salvi
Shrikant Bhausaheb Kanawade
Tukaram Nivrutti Chandre
Vinayak Kisan Thube
Pradeep Prakash Patil
Shalini Shukla
Kantilal Balu Shende
Pranab Kumar Patra
Alexander G M Klausener
Original Assignee
Pi Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pi Industries Ltd filed Critical Pi Industries Ltd
Publication of AR123593A1 publication Critical patent/AR123593A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32—Oxygen atoms
    • C07D209/38—Oxygen atoms in positions 2 and 3, e.g. isatin
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J27/00—Catalysts comprising the elements or compounds of halogens, sulfur, selenium, tellurium, phosphorus or nitrogen; Catalysts comprising carbon compounds
    • B01J27/02—Sulfur, selenium or tellurium; Compounds thereof
    • B01J27/057—Selenium or tellurium; Compounds thereof
    • B01J27/0573—Selenium; Compounds thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
    • C07C227/18—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions involving amino or carboxyl groups, e.g. hydrolysis of esters or amides, by formation of halides, salts or esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C229/26—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having more than one amino group bound to the carbon skeleton, e.g. lysine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/12—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
    • C07C233/15—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/56—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having carbon atoms of carboxamide groups bound to carbon atoms of carboxyl groups, e.g. oxamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/28—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton
    • C07C237/30—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having the nitrogen atom of the carboxamide group bound to hydrogen atoms or to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C249/00—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C249/04—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of oximes
    • C07C249/06—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of oximes by nitrosation of hydrocarbons or substituted hydrocarbons
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/36—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atoms of the oxyimino groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C251/40—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atoms of the oxyimino groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/20—Preparation of carboxylic acid nitriles by dehydration of carboxylic acid amides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C291/00—Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención divulga un proceso para la síntesis de compuesto de fórmula (2) o una sal del mismo, en donde, R, R¹, R², R³, R⁴ᵃ y R⁴ᵇ son como se definen en la descripción detallada. El proceso comprende adicionalmente la síntesis de un compuesto antranílico de diamida de fórmula (1).
ARP210102654A 2020-09-26 2021-09-24 Un proceso para la síntesis de compuestos antranílicos de ácido / amida e intermedios de los mismos AR123593A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN202011041843 2020-09-26

Publications (1)

Publication Number Publication Date
AR123593A1 true AR123593A1 (es) 2022-12-21

Family

ID=78599050

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP210102654A AR123593A1 (es) 2020-09-26 2021-09-24 Un proceso para la síntesis de compuestos antranílicos de ácido / amida e intermedios de los mismos

Country Status (11)

Country Link
US (1) US20230339906A1 (es)
EP (1) EP4217339A1 (es)
KR (1) KR20230074164A (es)
CN (1) CN116547266A (es)
AR (1) AR123593A1 (es)
BR (1) BR112023005509A2 (es)
CA (1) CA3191922A1 (es)
IL (1) IL301294A (es)
MX (1) MX2023003496A (es)
TW (1) TW202222162A (es)
WO (1) WO2022064454A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2024105700A1 (en) * 2022-11-18 2024-05-23 Pi Industries Ltd. A method for the synthesis of anthranilic amide compounds and intermediates thereof
CN116751151B (zh) * 2023-05-10 2025-10-10 瑞弘(天津)科技有限公司 一种5-氯-7-甲基靛红的一锅法制备方法
CN116836103A (zh) * 2023-07-06 2023-10-03 青岛科技大学 一种k胺中间体7-甲基靛红的制备方法
WO2025057193A1 (en) * 2023-09-13 2025-03-20 Pi Industries Ltd. A method for the synthesis of substituted anthranilic amide compounds, intermediates and salts thereof
TW202542105A (zh) * 2023-12-19 2025-11-01 印度商皮埃企業有限公司 經取代的鄰胺基苯甲醯胺化合物、其中間產物及其鹽的合成方法

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JP3184345B2 (ja) * 1992-12-16 2001-07-09 日清製粉株式会社 ５−クロロオキシインドールの製造方法
TWI325302B (en) 2001-08-13 2010-06-01 Du Pont Benzoxazinone compounds
AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
TWI326283B (en) 2002-07-31 2010-06-21 Du Pont Method for preparing fused oxazinones
EP1599463B1 (en) 2003-01-28 2013-06-05 E.I. Du Pont De Nemours And Company Cyano anthranilamide insecticides
EP1631564A1 (en) 2003-06-12 2006-03-08 E.I. Dupont De Nemours And Company Method for preparing fused oxazinones
WO2005021005A2 (en) * 2003-08-28 2005-03-10 Ranbaxy Laboratories Limited Process for the preparation of 1,4-benzodiazepine derivatives
SI1717237T1 (sl) 2004-02-18 2011-03-31 Ishihara Sangyo Kaisha Antranilamidi, postopek za njihovo proizvodnjo in sredstva za zatiranje škodljivcev, ki jih vsebujejo
TWI363756B (en) * 2004-12-07 2012-05-11 Du Pont Method for preparing n-phenylpyrazole-1-carboxamides
CN100361974C (zh) * 2005-12-31 2008-01-16 渤海大学 一种合成2-吲哚酮的方法
EP2394983B1 (en) 2006-07-19 2014-09-24 E.I. Du Pont De Nemours And Company Process for making 3-substituted 2-amino-5-halobenzamides
TWI395728B (zh) 2006-12-06 2013-05-11 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
TWI415827B (zh) 2006-12-21 2013-11-21 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
TWI430980B (zh) 2007-06-29 2014-03-21 Du Pont 製備２－胺基－5－氰基苯甲酸衍生物之方法
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TWI432421B (zh) 2007-12-19 2014-04-01 Du Pont 製備２－胺基－５－氰基苯甲酸衍生物之方法
WO2010069502A2 (de) 2008-12-18 2010-06-24 Bayer Cropscience Ag Tetrazolsubstituierte anthranilsäureamide als pestizide
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KR20140006007A (ko) 2011-01-28 2014-01-15 이 아이 듀폰 디 네모아 앤드 캄파니 2-아미노벤즈아미드 유도체의 제조 방법
TWI554507B (zh) 2011-08-26 2016-10-21 拜耳智慧財產有限公司 藉由苯并酮與胺反應製備經四唑取代之鄰胺苯甲酸二醯胺衍生物的方法
WO2019224678A1 (en) * 2018-05-21 2019-11-28 Pi Industries Ltd. A novel process for the preparation of anthranilic diamides
HUE069962T2 (hu) * 2019-02-18 2025-04-28 Pi Industries Ltd Eljárás antranil-diamidok és intermedierjeik elõállítására

Also Published As

Publication number Publication date
BR112023005509A2 (pt) 2023-04-25
CN116547266A (zh) 2023-08-04
KR20230074164A (ko) 2023-05-26
US20230339906A1 (en) 2023-10-26
IL301294A (en) 2023-05-01
EP4217339A1 (en) 2023-08-02
TW202222162A (zh) 2022-06-16
WO2022064454A1 (en) 2022-03-31
CA3191922A1 (en) 2022-03-31
MX2023003496A (es) 2023-04-14

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