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AR124286A1 - Proteínas de unión a il-7 y su uso en tratamientos médicos - Google Patents

Proteínas de unión a il-7 y su uso en tratamientos médicos

Info

Publication number
AR124286A1
AR124286A1 ARP210103301A ARP210103301A AR124286A1 AR 124286 A1 AR124286 A1 AR 124286A1 AR P210103301 A ARP210103301 A AR P210103301A AR P210103301 A ARP210103301 A AR P210103301A AR 124286 A1 AR124286 A1 AR 124286A1
Authority
AR
Argentina
Prior art keywords
seq
set forth
binding
binding protein
binding proteins
Prior art date
Application number
ARP210103301A
Other languages
English (en)
Inventor
Gerben Bouma
Edward Thomas Coulstock
David Dixon
Stephanie Hopley
Alan Peter Lewis
Jessica Lynn Neisen
Original Assignee
Glaxosmithkline Ip Dev Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Ip Dev Ltd filed Critical Glaxosmithkline Ip Dev Ltd
Publication of AR124286A1 publication Critical patent/AR124286A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/24Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against cytokines, lymphokines or interferons
    • C07K16/244Interleukins [IL]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/30Immunoglobulins specific features characterized by aspects of specificity or valency
    • C07K2317/33Crossreactivity, e.g. for species or epitope, or lack of said crossreactivity
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/30Immunoglobulins specific features characterized by aspects of specificity or valency
    • C07K2317/34Identification of a linear epitope shorter than 20 amino acid residues or of a conformational epitope defined by amino acid residues
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/73Inducing cell death, e.g. apoptosis, necrosis or inhibition of cell proliferation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/75Agonist effect on antigen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/76Antagonist effect on antigen, e.g. neutralization or inhibition of binding
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/90Immunoglobulins specific features characterized by (pharmaco)kinetic aspects or by stability of the immunoglobulin
    • C07K2317/92Affinity (KD), association rate (Ka), dissociation rate (Kd) or EC50 value
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/90Immunoglobulins specific features characterized by (pharmaco)kinetic aspects or by stability of the immunoglobulin
    • C07K2317/94Stability, e.g. half-life, pH, temperature or enzyme-resistance

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Immunology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Apparatus Associated With Microorganisms And Enzymes (AREA)

Abstract

En el presente documento se proporcionan proteínas de unión a interleucina 7 (IL-7), composiciones farmacéuticas y su uso en el tratamiento o prevención de una enfermedad o afección. Reivindicación 1: Una proteína de unión a IL-7 que se une a uno o más residuos de aminoácidos dentro de la secuencia de aminoácidos establecida en la SEQ ID Nº 12 de IL-7 humana. Reivindicación 4: Una proteína de unión a IL-7 caracterizada porque se une a IL-7 humana adyacente a un sitio de unión a IL-7Ra, con una KD de aproximadamente 100 nM o menos medida por ensayo de resonancia de plasmón de superficie. Reivindicación 7: Una proteína de unión a IL-7 caracterizada porque comprende CDRH1 como se establece en la SEQ ID Nº 6, CDRH2 como se indica en la SEQ ID Nº 7, CDRH3 como se indica en la SEQ ID Nº 8, CDRL1 como se indica en la SEQ ID Nº 9, CDRL2 como se establece en la SEQ ID Nº 10 y CDRL3 como se establece en la SEQ ID Nº 11. Reivindicación 27: Una composición farmacéutica, caracterizada porque comprende un transportador o excipiente farmacéuticamente aceptable y una proteína de unión a IL-7 que exhibe unión para IL-7 en un epítopo que comprende al menos 5 aminoácidos contiguos de una secuencia establecida en la SEQ ID Nº 12 o la SEQ ID Nº 16.
ARP210103301A 2020-12-02 2021-11-30 Proteínas de unión a il-7 y su uso en tratamientos médicos AR124286A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US202063120564P 2020-12-02 2020-12-02

Publications (1)

Publication Number Publication Date
AR124286A1 true AR124286A1 (es) 2023-03-15

Family

ID=78844686

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP210103301A AR124286A1 (es) 2020-12-02 2021-11-30 Proteínas de unión a il-7 y su uso en tratamientos médicos

Country Status (15)

Country Link
US (3) US11802150B2 (es)
EP (1) EP4255928A1 (es)
JP (1) JP2023551935A (es)
KR (1) KR20230098288A (es)
CN (1) CN116547002A (es)
AR (1) AR124286A1 (es)
AU (1) AU2021391493B2 (es)
CA (1) CA3199648A1 (es)
CL (1) CL2023001556A1 (es)
CO (1) CO2023007851A2 (es)
IL (1) IL303134A (es)
MX (1) MX2023006294A (es)
PH (1) PH12023551170A1 (es)
TW (1) TWI821804B (es)
WO (1) WO2022117526A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR129445A1 (es) * 2022-05-27 2024-08-28 Glaxosmithkline Ip Dev Ltd USO DE PROTEÍNAS DE UNIÓN A TNF-a Y PROTEÍNAS DE UNIÓN A IL-7 EN EL TRATAMIENTO MÉDICO

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57106673A (en) 1980-12-24 1982-07-02 Chugai Pharmaceut Co Ltd Dibenzo(b,f)(1,4)oxazepin derivative
GB8607679D0 (en) 1986-03-27 1986-04-30 Winter G P Recombinant dna product
DE3883899T3 (de) 1987-03-18 1999-04-22 Sb2, Inc., Danville, Calif. Geänderte antikörper.
IL127127A0 (en) 1998-11-18 1999-09-22 Peptor Ltd Small functional units of antibody heavy chain variable regions
US6737056B1 (en) 1999-01-15 2004-05-18 Genentech, Inc. Polypeptide variants with altered effector function
AU7950400A (en) 1999-10-19 2001-04-30 Kyowa Hakko Kogyo Co. Ltd. Process for producing polypeptide
US20050089932A1 (en) 2001-04-26 2005-04-28 Avidia Research Institute Novel proteins with targeted binding
US20050053973A1 (en) 2001-04-26 2005-03-10 Avidia Research Institute Novel proteins with targeted binding
MXPA04001072A (es) 2001-08-03 2005-02-17 Glycart Biotechnology Ag Variantes de glicosilacion de anticuerpos que tienen citotoxicidad celulares dependiente de anticuerpos incrementada.
ES2562177T3 (es) 2002-09-27 2016-03-02 Xencor Inc. Variantes de Fc optimizadas y métodos para su generación
EP2368578A1 (en) 2003-01-09 2011-09-28 Macrogenics, Inc. Identification and engineering of antibodies with variant Fc regions and methods of using same
US20050164301A1 (en) 2003-10-24 2005-07-28 Avidia Research Institute LDL receptor class A and EGF domain monomers and multimers
CA2573745A1 (en) 2004-07-21 2007-01-12 Glycofi, Inc. Immunoglobulins comprising predominantly a glcnac2man3glcnac2 glycoform
TW201018482A (en) 2008-08-08 2010-05-16 Glaxo Wellcome Mfg Pte Ltd Novel treatment
HRP20161542T1 (hr) * 2009-11-30 2016-12-30 Janssen Biotech, Inc. MUTIRANA Fc ANTITIJELA SA UKLONJENOM EFEKTORSKOM FUNKCIJOM

Also Published As

Publication number Publication date
TWI821804B (zh) 2023-11-11
US12122828B2 (en) 2024-10-22
CL2023001556A1 (es) 2023-11-10
US20240025988A1 (en) 2024-01-25
US11802150B2 (en) 2023-10-31
JP2023551935A (ja) 2023-12-13
WO2022117526A1 (en) 2022-06-09
CO2023007851A2 (es) 2023-06-30
US20220169717A1 (en) 2022-06-02
TW202237183A (zh) 2022-10-01
AU2021391493A1 (en) 2023-06-08
MX2023006294A (es) 2023-06-13
AU2021391493B2 (en) 2025-10-30
US20240425581A1 (en) 2024-12-26
CA3199648A1 (en) 2022-06-09
IL303134A (en) 2023-07-01
EP4255928A1 (en) 2023-10-11
KR20230098288A (ko) 2023-07-03
AU2021391493A9 (en) 2024-05-23
CN116547002A (zh) 2023-08-04
PH12023551170A1 (en) 2024-01-22

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