AR119218A1 - Oxadiazoles fungicidas - Google Patents
Oxadiazoles fungicidasInfo
- Publication number
- AR119218A1 AR119218A1 ARP200101757A ARP200101757A AR119218A1 AR 119218 A1 AR119218 A1 AR 119218A1 AR P200101757 A ARP200101757 A AR P200101757A AR P200101757 A ARP200101757 A AR P200101757A AR 119218 A1 AR119218 A1 AR 119218A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- haloalkyl
- aryl
- heteroaryl
- carbocyclyl
- Prior art date
Links
- 239000000417 fungicide Substances 0.000 title 1
- WCPAKWJPBJAGKN-UHFFFAOYSA-N oxadiazole Chemical compound C1=CON=N1 WCPAKWJPBJAGKN-UHFFFAOYSA-N 0.000 title 1
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 16
- -1 cyano, hydroxy, amino Chemical group 0.000 abstract 15
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 7
- 150000001875 compounds Chemical class 0.000 abstract 7
- 125000001072 heteroaryl group Chemical group 0.000 abstract 7
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 abstract 6
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 6
- 125000003118 aryl group Chemical group 0.000 abstract 6
- 229910052739 hydrogen Inorganic materials 0.000 abstract 6
- 239000001257 hydrogen Substances 0.000 abstract 6
- 125000001424 substituent group Chemical group 0.000 abstract 6
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 5
- 229910052736 halogen Inorganic materials 0.000 abstract 5
- 150000002367 halogens Chemical class 0.000 abstract 5
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 5
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 4
- 229910052731 fluorine Inorganic materials 0.000 abstract 4
- 239000011737 fluorine Substances 0.000 abstract 4
- 125000000623 heterocyclic group Chemical group 0.000 abstract 4
- LJXQPZWIHJMPQQ-UHFFFAOYSA-N pyrimidin-2-amine Chemical compound NC1=NC=CC=N1 LJXQPZWIHJMPQQ-UHFFFAOYSA-N 0.000 abstract 4
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 3
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 3
- KXDHJXZQYSOELW-UHFFFAOYSA-M Carbamate Chemical compound NC([O-])=O KXDHJXZQYSOELW-UHFFFAOYSA-M 0.000 abstract 3
- 125000002015 acyclic group Chemical group 0.000 abstract 3
- 125000004122 cyclic group Chemical group 0.000 abstract 3
- 125000001153 fluoro group Chemical group F* 0.000 abstract 3
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 3
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 abstract 2
- 125000004890 (C1-C6) alkylamino group Chemical group 0.000 abstract 2
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 abstract 2
- 125000006642 (C1-C6) cyanoalkyl group Chemical group 0.000 abstract 2
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 abstract 2
- SHQQYGVGAKIMEX-UHFFFAOYSA-N C1(=CC=CC=C1)C1(CC1)NC1=NC=C(C=N1)C1=NOC(=N1)C(F)(F)F Chemical compound C1(=CC=CC=C1)C1(CC1)NC1=NC=C(C=N1)C1=NOC(=N1)C(F)(F)F SHQQYGVGAKIMEX-UHFFFAOYSA-N 0.000 abstract 2
- 241000233866 Fungi Species 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 150000001204 N-oxides Chemical class 0.000 abstract 2
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 abstract 2
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 2
- 125000001995 cyclobutyl group Chemical group [H]C1([H])C([H])([H])C([H])(*)C1([H])[H] 0.000 abstract 2
- 150000002431 hydrogen Chemical class 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 230000003032 phytopathogenic effect Effects 0.000 abstract 2
- 239000012453 solvate Substances 0.000 abstract 2
- 125000003396 thiol group Chemical group [H]S* 0.000 abstract 2
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 abstract 1
- 125000004845 (C1-C6) alkylsulfonylamino group Chemical group 0.000 abstract 1
- 125000004740 (C1-C6) haloalkylsulfanyl group Chemical group 0.000 abstract 1
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 abstract 1
- 125000006648 (C1-C8) haloalkyl group Chemical group 0.000 abstract 1
- 125000006714 (C3-C10) heterocyclyl group Chemical group 0.000 abstract 1
- 125000006272 (C3-C7) cycloalkyl group Chemical group 0.000 abstract 1
- XDOXQQBUPUADQB-UHFFFAOYSA-N 5-(trifluoromethyl)-1,2,4-oxadiazole Chemical compound FC(F)(F)C1=NC=NO1 XDOXQQBUPUADQB-UHFFFAOYSA-N 0.000 abstract 1
- 125000006577 C1-C6 hydroxyalkyl group Chemical group 0.000 abstract 1
- 125000004648 C2-C8 alkenyl group Chemical group 0.000 abstract 1
- 125000004649 C2-C8 alkynyl group Chemical group 0.000 abstract 1
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical group [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical group FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
- 125000005153 alkyl sulfamoyl group Chemical group 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 229910052801 chlorine Chemical group 0.000 abstract 1
- 239000000460 chlorine Chemical group 0.000 abstract 1
- 235000013399 edible fruits Nutrition 0.000 abstract 1
- 125000005221 halo alkyl carbonyl amino group Chemical group 0.000 abstract 1
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 abstract 1
- OMPHAFHZEBBOGW-UHFFFAOYSA-N n-[1-(2-methylpyridin-4-yl)ethyl]-5-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]pyrimidin-2-amine Chemical compound C=1C=NC(C)=CC=1C(C)NC(N=C1)=NC=C1C1=NOC(C(F)(F)F)=N1 OMPHAFHZEBBOGW-UHFFFAOYSA-N 0.000 abstract 1
- 125000003170 phenylsulfonyl group Chemical group C1(=CC=CC=C1)S(=O)(=O)* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000002689 soil Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/82—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Reivindicación 1: Uso de un compuesto conforme a la fórmula (1) para controlar hongos fitopatogénicos en plantas, siendo que X es flúor o cloro; R¹, R² considerados en forma independiente se seleccionan a partir del conjunto que consiste en hidrógeno, ciano, C₁₋₈-alquilo, C₁₋₈-haloalquilo, C₂₋₈-alquenilo, C₂₋₈-haloalquenilo, C₂₋₈-alquinilo, C₂₋₈-haloalquinilo, C₃₋₇-carbociclilo, arilo, heterociclilo de 3 a 10 miembros, heteroarilo, aril-C₁₋₈-alquilo, heterociclilo de 3 a 10 miembros-C₁₋₈-alquilo, heteroaril-C₁₋₈-alquilo y C₃₋₇-carbociclil-C₁₋₈-alquilo, siendo que dichos R¹ y R² acíclicos pueden estar sustituidos con, respectivamente, uno o más sustituyentes R¹ᵃ y R²ᵃ y dichos R¹ y R² cíclicos pueden estar sustituidos con, respectivamente, uno o más sustituyentes R¹ᵇ y R²ᵇ, o R¹, R² pueden formar, junto con el átomo de carbono al que están unidos, un C₃₋₇-carbociclilo o un heterociclilo de 3 a 10 miembros, siendo que dicho C₃₋₇-carbociclilo o heterociclilo de 3 a 10 miembros puede estar sustituido con uno o más sustituyentes R¹ᵇ; Cy es arilo, heteroarilo, C₃₋₁₀-carbociclilo o heterociclilo de 3 a 10 miembros; n es 0, 1, 2, 3 ó 4; R³ considerado en forma independiente se selecciona a partir del conjunto que consiste en halógeno, ciano, hidroxi, amino, nitro, carboxilo, sulfanilo, pentafluoro-l⁶-sulfanilo, formilo, carbamoilo, carbamato, C₁₋₆-alquilo, C₁₋₆-cianoalquilo, C₁₋₆-haloalquilo, C₂₋₆-alquenilo, C₂₋₆-haloalquenilo, C₂₋₆-alquinilo, C₂₋₆-haloalquinilo, C₁₋₆-alcoxi, C₁₋₆-haloalcoxi, C₁₋₆-alcoxi-C₁₋₆-alquilo, C₁₋₆-alquilsulfanilo, C₁₋₆-haloalquilsulfanilo, C₁₋₈-alquilsulfinilo, C₁₋₈-haloalquilsulfinilo, C₁₋₈-alquilsulfonilo, C₁₋₈-haloalquilsulfonilo, C₃₋₇-carbociclilo, C₃₋₇-halocarbociclilo, C₁₋₆-hidroxialquilo, C₁₋₆-alquilamino, di-C₁₋₆-alquilamino, C₁₋₆-alquilcarbonilo, C₁₋₆-alcoxicarbonilo, C₁₋₆-haloalcoxicarbonilo, C₁₋₆-alquilcarbamoilo, di-C₁₋₆-alquilcarbamoilo, aminocarbonilo, C₁₋₈-alquilcarboniloxi, C₁₋₈-haloalquilcarboniloxi, C₁₋₈-alquilcarbonilamino, C₁₋₈-haloalquilcarbonilamino, C₁₋₆-alquilsulfonilamino, C₁₋₆-haloalquilsulfonilamino, sulfamoilo, C₁₋₈-alquilsulfamoilo, di-C₁₋₈-alquilsulfamoilo, arilo (por ejemplo fenilo), aril-C₁₋₆-alquilo y heteroarilo, siendo que dichos R³ acíclicos y cíclicos pueden estar sustituidos con uno o más sustituyentes, los cuales pueden ser el mismo o diferentes, a seleccionar a partir del conjunto que consiste en halógeno, C₁₋₆-alquilo, C₁₋₆-haloalquilo, C₁₋₆-alcoxi y C₁₋₆-haloalcoxi; R⁴ se selecciona a partir del conjunto que consiste en hidrógeno, hidroxi, formilo, C₁₋₆-alquilo, C₁₋₆-haloalquilo, C₂₋₆-alquenilo, C₂₋₆-haloalquenilo, C₂₋₆-alquinilo, C₂₋₆-haloalquinilo, -C(=O)-C₁₋₆-alquilo, -C(=O)-C₁₋₆-haloalquilo, -C(=S)-C₁₋₆-alquilo, -C(=S)-C₁₋₆-haloalquilo, -C(=O)-O-C₁₋₆-alquilo, -C(=O)-O-C₁₋₆-haloalquilo, C₁₋₆-alcoxi, C₁₋₆-haloalcoxi, C₁₋₆-alquilsulfonilo, C₁₋₆-haloalquilsulfonilo, fenilsulfonilo, C₃₋₁₀-carbociclilo, heterociclilo de 3 a 10 miembros, arilo (fenilo), heteroarilo, C₃₋₁₀-carbociclil-C₁₋₆-alquilo, C₃₋₁₀-carbociclil-C₁₋₆-haloalquilo, aril-C₁₋₆-alquilo, aril-C₁₋₆-haloalquilo, heteroaril-C₁₋₆-alquilo y heteroaril-C₁₋₆-haloalquilo, siendo que dichos R⁴ cíclicos y acíclicos pueden estar sustituidos con uno o más sustituyentes a seleccionar a partir del conjunto que consiste en halógeno, ciano, C₁₋₆-alquilo, C₁₋₆-haloalquilo, C₁₋₆-alcoxi y C₁₋₆-haloalcoxi; R⁵ es hidrógeno o flúor; R¹ᵃ, R²ᵃ considerados en forma independiente se seleccionan a partir del conjunto que consiste en nitro, hidroxilo, ciano, carboxilo, amino, sulfanilo, pentafluoro-l⁶-sulfanilo, formilo, carbamoilo, carbamato, C₃₋₇-cicloalquilo, C₃₋₇-halocicloalquilo, C₁₋₈-alquilamino, di-C₁₋₈-alquilamino, C₁₋₈-alcoxi, C₁₋₈-haloalcoxi, C₁₋₈-alquilsulfanilo, C₁₋₈-haloalquilsulfanilo, C₁₋₈-alquilcarbonilo, C₁₋₈-haloalquilcarbonilo, C₁₋₈-alquilcarbamoilo, di-C₁₋₈-alquilcarbamoilo, C₁₋₈-alcoxicarbonilo, C₁₋₈-haloalcoxicarbonilo, C₁₋₈-alquilcarboniloxi, C₁₋₈-haloalquilcarboniloxi, C₁₋₈-alquilcarbonilamino, C₁₋₈-haloalquilcarbonilamino, C₁₋₈-alquilsulfinilo, C₁₋₈-haloalquilsulfinilo, C₁₋₈-alquilsulfonilo, C₁₋₈-haloalquilsulfonilo, C₁₋₈-alquilsulfonilamino, C₁₋₈-haloalquilsulfonilamino, sulfamoilo, C₁₋₈-alquilsulfamoilo y di-C₁₋₈-alquilsulfamoilo; R¹ᵇ, R²ᵇ considerados en forma independiente se seleccionan a partir del conjunto que consiste en halógeno, ciano, hidroxi, amino, nitro, carboxilo, sulfanilo, pentafluoro-l⁶-sulfanilo, formilo, carbamoilo, carbamato, C₁₋₆-alquilo, C₁₋₆-cianoalquilo, C₁₋₆-haloalquilo, C₂₋₆-alquenilo, C₂₋₆-haloalquenilo, C₂₋₆-alquinilo, C₂₋₆-haloalquinilo, C₁₋₆-alcoxi, C₁₋₆-haloalcoxi, C₁₋₆-alcoxiC₁₋₆-alquilo, C₁₋₆-alquilsulfanilo, C₁₋₆-haloalquilsulfanilo, C₁₋₈-alquilsulfinilo, C₁₋₈-haloalquilsulfinilo, C₁₋₈-alquilsulfonilo, C₁₋₈-haloalquilsulfonilo, C₁₋₆-alquil-C(=O)-NH-, C₃₋₇-carbociclilo, C₃₋₇-halocarbociclilo, hidroxi-C₁₋₆-alquilo, C₁₋₆-alquilamino, di-C₁₋₆-alquilamino, C₁₋₆-alquilcarbonilo, C₁₋₆-alcoxicarbonilo, C₁₋₆-haloalcoxicarbonilo, C₁₋₆-alquilcarbamoilo, di-C₁₋₆-alquilcarbamoilo, aminocarbonilo, C₁₋₈-alquilcarboniloxi, C₁₋₈-haloalquilcarboniloxi, C₁₋₈-alquilcarbonilamino, C₁₋₈-haloalquilcarbonilamino, C₁₋₆-alquilsulfonilamino, C₁₋₆-haloalquilsulfonilamino, sulfamoilo, C₁₋₈-alquilsulfamoilo, di-C₁₋₈-alquilsulfamoilo, arilo (por ejemplo fenilo), aril-C₁₋₆-alquilo y heteroarilo, siendo que dicho arilo (fenilo) o heteroarilo opcionalmente está sustituido con uno o más sustituyentes, los cuales pueden ser el mismo o diferentes, a seleccionar a partir del conjunto que consiste en halógeno, C₁₋₆-alquilo, C₁₋₆-haloalquilo, C₁₋₆-alcoxi y C₁₋₆-haloalcoxi; o una sal N-óxido o solvato de dicha estructura; siendo que el compuesto conforme a la fórmula (1) no es: (a) N-[1-(piridin-2-il)ciclobutil)-5-[5-(trifluorometil)-1,2,4-oxadiazol-3-il]pirimidin-2-amina; (b) 5-{5-[cloro(difluoro)metil)-1,2,4-oxadiazol-3-il}-N-[1-(piridin-2-il)ciclobutil]pirimidin-2-amina; (c) N-(1-fenilciclopropil)-5-[5-(trifluorometil)-1,2,4-oxadiazol-3-il]pirimidin-2-amina; (d) 5-{5-[cloro(difluoro)metil)-1,2,4-oxadiazol-3-il}-N-(1-fenilciclopropil)pirimidin-2-amina. Reivindicación 13: Un método para controlar hongos fitopatogénicos que comprende el paso de aplicar al menos un compuesto conforme a la fórmula (1) conforme a una cualquiera de las reivindicaciones 1 a 12 a las plantas, las partes de planta, las semillas, las frutas o el suelo en el que crecen las plantas. Reivindicación 14: Un compuesto conforme a la fórmula (1) o un sal, N-óxido o solvato de dicha estructura; siendo que X, R¹, R², R³, R⁴, R⁵, Cy y n son tal como se definen en cualquiera de las reivindicaciones 1 a 12, siendo que cuando X es flúor y R⁴ es hidrógeno o C₁₋₆-alquilo, R¹ y R² no son ambos hidrógeno; siendo que se excluyen los compuestos en los que X es flúor, Cy es fenilo o heteroarilo de 6 miembros, n es 0 y R¹, R² y R⁴ se seleccionan, considerando cada uno en forma independiente, a partir de hidrógeno y C₁₋₃-alquilo; y siendo que el compuesto conforme a la fórmula (1) no es: (a) N-[1-(piridin-2-il)ciclobutil)-5-[5-(trifluorometil)-1,2,4-oxadiazol-3-il]pirimidin-2-amina; (b) 5-{5-[cloro(difluoro)metil)-1,2,4-oxadiazol-3-il}-N-[1-(piridin-2-il)ciclobutil]pirimidin-2-amina; (c) N-(1-fenilciclopropil)-5-[5-(trifluorometil)-1,2,4-oxadiazol-3-il]pirimidin-2-amina; (d) 5-{5-[cloro(difluoro)metil)-1,2,4-oxadiazol-3-il}-N-(1-fenilciclopropil)pirimidin-2-amina; (e) N-[1-(2-metilpiridin-4-il)etil)-5-[5-(trifluorometil)-1,2,4-oxadiazol-3-il]pirimidin-2-amina. Reivindicación 16: Una composición que comprende al menos un compuesto conforme a la fórmula (1) conforme a la reivindicación 14 ó 15 y al menos un vehículo apto para uso agrícola.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP19181819 | 2019-06-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR119218A1 true AR119218A1 (es) | 2021-12-01 |
Family
ID=67001713
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP200101757A AR119218A1 (es) | 2019-06-21 | 2020-06-19 | Oxadiazoles fungicidas |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP3986889A1 (es) |
| AR (1) | AR119218A1 (es) |
| BR (1) | BR112021025300A2 (es) |
| TW (1) | TW202115045A (es) |
| UY (1) | UY38761A (es) |
| WO (1) | WO2020254494A1 (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018165520A1 (en) | 2017-03-10 | 2018-09-13 | Vps-3, Inc. | Metalloenzyme inhibitor compounds |
| WO2021021979A2 (en) | 2019-07-30 | 2021-02-04 | Eikonizo Therapapeutics, Inc. | Hdac6 inhibitors and uses thereof |
| JP2023043197A (ja) * | 2020-03-04 | 2023-03-29 | 日本曹達株式会社 | アジニルアゾール化合物および有害生物防除剤（２） |
| WO2021255093A1 (en) * | 2020-06-19 | 2021-12-23 | Bayer Aktiengesellschaft | Active compound combination |
| UY39854A (es) | 2021-07-15 | 2022-11-30 | Kumiai Chemical Industry Co | Derivado de formamida y agente de control hortícola y agrícola para el control de enfermedades de la |
| WO2023107705A1 (en) | 2021-12-10 | 2023-06-15 | Incyte Corporation | Bicyclic amines as cdk12 inhibitors |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| DE3639877A1 (de) | 1986-11-21 | 1988-05-26 | Bayer Ag | Hetarylalkyl substituierte 5- und 6-ringheterocyclen |
| IL132533A0 (en) | 1997-05-09 | 2001-03-19 | Agraquest Inc | A novel strain of bacillus for controlling plant diseases and corn rootworm |
| US6245551B1 (en) | 1999-03-30 | 2001-06-12 | Agraquest, Inc. | Strain of Bacillus pumilus for controlling plant diseases caused by fungi |
| JP4071036B2 (ja) | 2001-11-26 | 2008-04-02 | クミアイ化学工業株式会社 | バシルスｓｐ．Ｄ７４７菌株およびそれを用いた植物病害防除剤および害虫防除剤 |
| GB0213715D0 (en) | 2002-06-14 | 2002-07-24 | Syngenta Ltd | Chemical compounds |
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-
2020
- 2020-06-18 EP EP20734340.1A patent/EP3986889A1/en active Pending
- 2020-06-18 BR BR112021025300A patent/BR112021025300A2/pt unknown
- 2020-06-18 WO PCT/EP2020/066947 patent/WO2020254494A1/en not_active Ceased
- 2020-06-19 AR ARP200101757A patent/AR119218A1/es unknown
- 2020-06-19 TW TW109120773A patent/TW202115045A/zh unknown
- 2020-06-22 UY UY0001038761A patent/UY38761A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EP3986889A1 (en) | 2022-04-27 |
| TW202115045A (zh) | 2021-04-16 |
| WO2020254494A1 (en) | 2020-12-24 |
| BR112021025300A2 (pt) | 2022-02-01 |
| UY38761A (es) | 2021-01-29 |
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