AR114086A2 - Polvos para reconstitución - Google Patents
Polvos para reconstituciónInfo
- Publication number
- AR114086A2 AR114086A2 ARP190100128A ARP190100128A AR114086A2 AR 114086 A2 AR114086 A2 AR 114086A2 AR P190100128 A ARP190100128 A AR P190100128A AR P190100128 A ARP190100128 A AR P190100128A AR 114086 A2 AR114086 A2 AR 114086A2
- Authority
- AR
- Argentina
- Prior art keywords
- reconstitution
- powders
- refers
- water soluble
- soluble polymers
- Prior art date
Links
- 239000000843 powder Substances 0.000 title abstract 2
- 208000031886 HIV Infections Diseases 0.000 abstract 1
- 208000037357 HIV infectious disease Diseases 0.000 abstract 1
- 208000033519 human immunodeficiency virus infectious disease Diseases 0.000 abstract 1
- 239000002726 nonnucleoside reverse transcriptase inhibitor Substances 0.000 abstract 1
- YIBOMRUWOWDFLG-ONEGZZNKSA-N rilpivirine Chemical compound CC1=CC(\C=C\C#N)=CC(C)=C1NC1=CC=NC(NC=2C=CC(=CC=2)C#N)=N1 YIBOMRUWOWDFLG-ONEGZZNKSA-N 0.000 abstract 1
- 229920003169 water-soluble polymer Polymers 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Virology (AREA)
- Inorganic Chemistry (AREA)
- Oncology (AREA)
- AIDS & HIV (AREA)
- General Chemical & Material Sciences (AREA)
- Molecular Biology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Compositions Of Macromolecular Compounds (AREA)
Abstract
La presente se refiere a polvos para reconstitución que comprenden el NNRTI TMC278 disperso en ciertos polímeros solubles en agua, que puede aplicarse en el tratamiento contra la infección por HIV.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07104082 | 2007-03-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR114086A2 true AR114086A2 (es) | 2020-07-22 |
Family
ID=38055251
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080101032A AR065720A1 (es) | 2007-03-14 | 2008-03-13 | Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso. |
| ARP190100128A AR114086A2 (es) | 2007-03-14 | 2019-01-21 | Polvos para reconstitución |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080101032A AR065720A1 (es) | 2007-03-14 | 2008-03-13 | Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US8916558B2 (es) |
| EP (1) | EP2043608B1 (es) |
| JP (1) | JP5554571B2 (es) |
| KR (1) | KR101580297B1 (es) |
| CN (1) | CN101636149B (es) |
| AP (1) | AP2964A (es) |
| AR (2) | AR065720A1 (es) |
| AU (1) | AU2008225774B2 (es) |
| BR (1) | BRPI0808897B8 (es) |
| CA (1) | CA2676981C (es) |
| CL (1) | CL2008000746A1 (es) |
| ES (1) | ES2535162T3 (es) |
| IL (1) | IL199874A (es) |
| MX (1) | MX2009009743A (es) |
| RU (1) | RU2477133C2 (es) |
| TW (1) | TWI494133B (es) |
| WO (1) | WO2008110619A1 (es) |
| ZA (1) | ZA200906344B (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY169670A (en) | 2003-09-03 | 2019-05-08 | Tibotec Pharm Ltd | Combinations of a pyrimidine containing nnrti with rt inhibitors |
| AR065720A1 (es) | 2007-03-14 | 2009-06-24 | Tibotec Pharm Ltd | Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso. |
| HRP20201241T1 (hr) * | 2011-04-15 | 2020-11-27 | Janssen Pharmaceutica N.V. | Nanosuspenzije lijeka osušene zamrzavanjem |
| CN104684545B (zh) * | 2012-09-27 | 2018-04-03 | 巴斯夫欧洲公司 | 包含至少一种水溶性维生素e衍生物和至少一种亲水聚合物的储存稳定的无粉尘均质颗粒状配制剂 |
| CA3144534A1 (en) * | 2019-07-03 | 2021-01-07 | Janssen Sciences Ireland Unlimited Company | Methods of treating hiv in pediatric patients with rilpivirine |
| CN113440529B (zh) * | 2020-03-25 | 2023-11-14 | 江苏恒瑞医药股份有限公司 | 一种可注射的药物组合物及其制备方法 |
| CN114392241B (zh) * | 2022-01-10 | 2023-07-25 | 安徽贝克生物制药有限公司 | 一种利匹韦林片及其制备方法 |
| JP2025513501A (ja) * | 2022-04-22 | 2025-04-24 | ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー | 凍結乾燥組成物 |
Family Cites Families (47)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3089818A (en) * | 1960-06-02 | 1963-05-14 | Baxter Laboratories Inc | Water dispersible antibiotics |
| US5182111A (en) * | 1987-11-17 | 1993-01-26 | Boston University Research Foundation | In vivo delivery of active factors by co-cultured cell implants |
| US5368864A (en) * | 1988-11-25 | 1994-11-29 | Henning Berlin Gmbh Chemie- Und Pharmawerk | Formulation of oxypurinol and/or its alkali and alkaline earth salts |
| WO1992001453A1 (fr) | 1990-07-19 | 1992-02-06 | Otsuka Pharmaceutical Co., Ltd. | Preparation solide |
| US5145684A (en) | 1991-01-25 | 1992-09-08 | Sterling Drug Inc. | Surface modified drug nanoparticles |
| AU3124793A (en) * | 1991-10-29 | 1993-06-07 | Clover Consolidated, Limited | Crosslinkable polysaccharides, polycations and lipids useful for encapsulation and drug release |
| DK0639971T3 (da) | 1992-05-13 | 2000-03-20 | Wellcome Found | Terapeutiske kombinationer |
| JPH06316524A (ja) | 1992-09-11 | 1994-11-15 | Naoyuki Inoue | 抗エイズウイルス剤 |
| TW401303B (en) | 1994-07-01 | 2000-08-11 | Janssen Pharmaceutica Nv | Anti-HIV triple combination |
| US6045829A (en) * | 1997-02-13 | 2000-04-04 | Elan Pharma International Limited | Nanocrystalline formulations of human immunodeficiency virus (HIV) protease inhibitors using cellulosic surface stabilizers |
| JP2003509453A (ja) | 1999-09-21 | 2003-03-11 | アールティーピー・ファーマ・インコーポレーテッド | 生物学的に活性な物質の、表面改質された粒状組成物 |
| WO2001022938A1 (en) * | 1999-09-24 | 2001-04-05 | Janssen Pharmaceutica N.V. | Antiviral compositions |
| US6743446B2 (en) * | 1999-12-15 | 2004-06-01 | The Ohio State University Research Foundation | Methods for stabilizing biologically active agents encapsulated in biodegradable controlled-release polymers |
| TWI284048B (en) * | 2000-01-27 | 2007-07-21 | Zentaris Ag | Compressed microparticles for dry injection |
| HUP0302631A2 (hu) | 2000-03-30 | 2003-11-28 | Bristol-Myers Squibb Co. | Stavudint tartalmazó elnyújtott hatóanyag-kibocsátású szemcsék |
| US20040115268A1 (en) * | 2000-04-26 | 2004-06-17 | Control Delivery Systems, Inc. | Systemic delivery of antiviral agents |
| DE10050199A1 (de) | 2000-10-11 | 2002-04-25 | Ethicon Gmbh | Flächiges Implantat mit im Ultraschall detektierbaren Elementen |
| EP1350792A1 (en) | 2000-12-11 | 2003-10-08 | Takeda Chemical Industries, Ltd. | Medicinal compositions improved in solublity in water |
| CA2450957A1 (en) * | 2001-06-22 | 2003-01-03 | Pfizer Products Inc. | Pharmaceutical compositions of dispersions of drugs and neutral polymers |
| JO3429B1 (ar) * | 2001-08-13 | 2019-10-20 | Janssen Pharmaceutica Nv | مشتقات برميدينات مثبطة فيروس الايدز |
| MY169670A (en) | 2003-09-03 | 2019-05-08 | Tibotec Pharm Ltd | Combinations of a pyrimidine containing nnrti with rt inhibitors |
| AU2002364701B8 (en) | 2001-11-20 | 2006-06-22 | Alkermes, Inc. | Compositions for sustained action product delivery |
| ES2422196T3 (es) | 2002-08-09 | 2013-09-09 | Janssen Pharmaceutica Nv | Procesos para la preparación de 4-4-4-(2-cianoetenil)-2,6-dimetilfenil)amino)-2-pirimidinil)aminobenzonitrilo |
| WO2004022033A1 (en) * | 2002-09-04 | 2004-03-18 | Microchips, Inc. | Method and device for the controlled delivery of parathyroid hormone |
| ATE361059T1 (de) | 2002-11-08 | 2007-05-15 | Glaxo Group Ltd | Antivirale zusammensetzungen |
| KR20050084621A (ko) | 2002-11-15 | 2005-08-26 | 티보텍 파마슈티칼즈 리미티드 | 항감염성 화합물로서의 치환된 인돌피리디늄 |
| WO2004050068A1 (en) * | 2002-11-29 | 2004-06-17 | Janssen Pharmaceutica N.V. | Pharmaceutical compositions comprising a basic respectively acidic drug compound, a surfactant and a physiologically tolerable water-soluble acid respectively base |
| CL2004000192A1 (es) | 2003-02-07 | 2005-03-18 | Janssen Pharmaceutica Nv | Uso de compuestos derivados de 2-aminopirimidina para preparar un medicamento para la prevencion de una infeccion por vih relaciones sexuales o un contacto intimo en la pareja. |
| KR100629771B1 (ko) * | 2004-01-27 | 2006-09-28 | 씨제이 주식회사 | 결정성이 감소되거나 무정형화된 올티프라즈의 제조방법 |
| BRPI0511900A (pt) * | 2004-06-08 | 2008-01-22 | Vertex Pharma | composições farmacêuticas |
| MY191349A (en) | 2004-08-27 | 2022-06-17 | Bayer Pharmaceuticals Corp | New pharmaceutical compositions for the treatment of hyper-proliferative disorders |
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| PL1632232T6 (pl) | 2004-09-02 | 2022-06-27 | Janssen Pharmaceutica Nv | Sól 4-[[4-[[4-(2-cyjanoetenylo)-2,6-dimetylofenylo]amino]-2-pirymidynylo]amino]benzonitrylu |
| ES2526092T3 (es) | 2004-11-16 | 2015-01-05 | Alkermes Pharma Ireland Limited | Formulaciones de olanzapina en nanopartículas inyectables |
| TWI457136B (zh) | 2005-04-04 | 2014-10-21 | Tibotec Pharm Ltd | Hiv-感染之預防 |
| AR056652A1 (es) * | 2005-04-11 | 2007-10-17 | Tibotec Pharm Ltd | Derivados de (1,10-b dihidro-2-(aminoalquil-fenil) -5h-pirazolo (1,5-c) (1,3)benzoxazin-5-il) fenilmetanona y su uso en la fabricacion de un medicamento |
| WO2006110889A2 (en) * | 2005-04-11 | 2006-10-19 | The Board Of Trustees Of The Leland Stanford Junior University | Multi-layer structure having a predetermined layer pattern including an agent |
| US20090142401A1 (en) | 2005-06-07 | 2009-06-04 | Leah Elizabeth Appel | Multiparticulates comprising low-solubility drugs and carriers that result in rapid drug release |
| US20070026073A1 (en) | 2005-07-28 | 2007-02-01 | Doney John A | Amorphous efavirenz and the production thereof |
| RS52821B2 (sr) | 2006-01-20 | 2021-07-30 | Janssen Sciences Ireland Unlimited Co | Dugotrajno tretiranje hiv-infekcije sa tcm278 |
| ES2372983T3 (es) | 2006-06-06 | 2012-01-30 | Tibotec Pharmaceuticals | Proceso para preparar formulaciones secadas por aspersión de tmc125. |
| HUE038797T2 (hu) | 2006-06-23 | 2018-11-28 | Janssen Sciences Ireland Uc | TMC278 vizes szuszpenziói |
| WO2008060360A2 (en) * | 2006-09-28 | 2008-05-22 | Surmodics, Inc. | Implantable medical device with apertures for delivery of bioactive agents |
| AR065720A1 (es) | 2007-03-14 | 2009-06-24 | Tibotec Pharm Ltd | Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso. |
| ES2437331T3 (es) | 2007-07-12 | 2014-01-10 | Janssen R&D Ireland | Forma cristalina de 4-[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]amino]-2-pirimidinil]amino]benzonitrilo |
| WO2009046299A2 (en) | 2007-10-04 | 2009-04-09 | Boston Scientific Scimed, Inc | Implantable drug depot for intrathecal drug delivery system for pain management |
| WO2010047819A1 (en) * | 2008-10-24 | 2010-04-29 | Concert Pharmaceuticals, Inc. | Hydroxyethylamino sulfonamide derivatives |
-
2008
- 2008-03-13 AR ARP080101032A patent/AR065720A1/es not_active Application Discontinuation
- 2008-03-13 TW TW097108780A patent/TWI494133B/zh active
- 2008-03-13 CL CL200800746A patent/CL2008000746A1/es unknown
- 2008-03-14 WO PCT/EP2008/053056 patent/WO2008110619A1/en not_active Ceased
- 2008-03-14 MX MX2009009743A patent/MX2009009743A/es active IP Right Grant
- 2008-03-14 CN CN200880008342.0A patent/CN101636149B/zh active Active
- 2008-03-14 JP JP2009553156A patent/JP5554571B2/ja active Active
- 2008-03-14 BR BRPI0808897A patent/BRPI0808897B8/pt not_active IP Right Cessation
- 2008-03-14 KR KR1020097017592A patent/KR101580297B1/ko not_active Expired - Fee Related
- 2008-03-14 AP AP2009004969A patent/AP2964A/xx active
- 2008-03-14 US US12/530,665 patent/US8916558B2/en active Active
- 2008-03-14 ES ES08717800.0T patent/ES2535162T3/es active Active
- 2008-03-14 CA CA2676981A patent/CA2676981C/en active Active
- 2008-03-14 AU AU2008225774A patent/AU2008225774B2/en not_active Ceased
- 2008-03-14 RU RU2009137911/15A patent/RU2477133C2/ru active
- 2008-03-14 EP EP08717800.0A patent/EP2043608B1/en active Active
-
2009
- 2009-07-15 IL IL199874A patent/IL199874A/en active IP Right Grant
- 2009-09-11 ZA ZA2009/06344A patent/ZA200906344B/en unknown
-
2019
- 2019-01-21 AR ARP190100128A patent/AR114086A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CN101636149A (zh) | 2010-01-27 |
| IL199874A0 (en) | 2010-04-15 |
| AR065720A1 (es) | 2009-06-24 |
| EP2043608A1 (en) | 2009-04-08 |
| BRPI0808897A2 (pt) | 2014-09-02 |
| CL2008000746A1 (es) | 2008-09-22 |
| AP2964A (en) | 2014-09-30 |
| JP5554571B2 (ja) | 2014-07-23 |
| US20100120795A1 (en) | 2010-05-13 |
| ES2535162T3 (es) | 2015-05-05 |
| CN101636149B (zh) | 2014-08-06 |
| IL199874A (en) | 2016-02-29 |
| US8916558B2 (en) | 2014-12-23 |
| BRPI0808897B8 (pt) | 2021-05-25 |
| CA2676981C (en) | 2015-01-13 |
| AP2009004969A0 (en) | 2009-10-31 |
| WO2008110619A1 (en) | 2008-09-18 |
| EP2043608B1 (en) | 2015-01-21 |
| KR101580297B1 (ko) | 2015-12-24 |
| JP2010520918A (ja) | 2010-06-17 |
| RU2477133C2 (ru) | 2013-03-10 |
| TW200911303A (en) | 2009-03-16 |
| RU2009137911A (ru) | 2011-04-20 |
| KR20090119964A (ko) | 2009-11-23 |
| BRPI0808897B1 (pt) | 2020-10-20 |
| AU2008225774A1 (en) | 2008-09-18 |
| ZA200906344B (en) | 2015-04-29 |
| TWI494133B (zh) | 2015-08-01 |
| CA2676981A1 (en) | 2008-09-18 |
| MX2009009743A (es) | 2009-09-23 |
| AU2008225774B2 (en) | 2014-04-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC | Refusal |