AR100404A1 - Polimorfos cristalinos de un derivado de piridina y método para producirlos - Google Patents
Polimorfos cristalinos de un derivado de piridina y método para producirlosInfo
- Publication number
- AR100404A1 AR100404A1 ARP150101454A ARP150101454A AR100404A1 AR 100404 A1 AR100404 A1 AR 100404A1 AR P150101454 A ARP150101454 A AR P150101454A AR P150101454 A ARP150101454 A AR P150101454A AR 100404 A1 AR100404 A1 AR 100404A1
- Authority
- AR
- Argentina
- Prior art keywords
- polymorphes
- producers
- crystalline
- pyridine derivative
- crystal
- Prior art date
Links
- JUJWROOIHBZHMG-UHFFFAOYSA-N Pyridine Chemical class C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 title 1
- 239000013078 crystal Substances 0.000 abstract 7
- XYCCPIZLKKAACR-UHFFFAOYSA-N 2-(5-chloropyridin-3-yl)-3-[(2,5-dichlorophenyl)methyl]-5-methylimidazole-4-carboxylic acid Chemical compound ClC=1C=C(C=NC1)C=1N(C(=C(N1)C)C(=O)O)CC1=C(C=CC(=C1)Cl)Cl XYCCPIZLKKAACR-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Hematology (AREA)
- Vascular Medicine (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
- Pyridine Compounds (AREA)
Abstract
Reivindicación 1: Un cristal del ácido 2-(5-cloropiridin-3-il)-1-(2,5-diclorobencil)-4-metil-1H-imidazol-5-carboxílico. Reivindicación 2: El cristal de acuerdo con la reivindicación 1, donde el cristal tiene una forma de cristal A. Reivindicación 10: El cristal de acuerdo con la reivindicación 1, donde el cristal tiene una forma de cristal B.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2014099678 | 2014-05-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR100404A1 true AR100404A1 (es) | 2016-10-05 |
Family
ID=54479948
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP150101454A AR100404A1 (es) | 2014-05-13 | 2015-05-12 | Polimorfos cristalinos de un derivado de piridina y método para producirlos |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20170144987A1 (es) |
| EP (1) | EP3144304A4 (es) |
| JP (1) | JP6289619B2 (es) |
| KR (1) | KR20170003569A (es) |
| CN (1) | CN106458970B (es) |
| AR (1) | AR100404A1 (es) |
| AU (1) | AU2015260294A1 (es) |
| CA (1) | CA2948792A1 (es) |
| IL (1) | IL248901A0 (es) |
| MX (1) | MX2016014692A (es) |
| PH (1) | PH12016502222A1 (es) |
| RU (1) | RU2016148736A (es) |
| SG (1) | SG11201609483YA (es) |
| TW (1) | TW201625580A (es) |
| WO (1) | WO2015174411A1 (es) |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK0513379T3 (da) * | 1990-11-30 | 1996-09-30 | Teijin Ltd | 2-Arylthiazolderivater og farmaceutisk præparat indeholdende sådanne |
| US8148542B2 (en) * | 2006-06-23 | 2012-04-03 | Teijin Pharma Limited | Method for producing crystal polymorphs of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazolecarboxylic acid |
| MX2010010366A (es) * | 2008-03-31 | 2010-11-30 | C & C Res Lab | Derivados heterociclicos. |
| CN102333765B (zh) * | 2009-02-27 | 2015-01-14 | 帝人制药株式会社 | 基于使用过渡金属催化剂的偶联法的苯基取代杂环衍生物的制造方法 |
| WO2011007895A1 (ja) * | 2009-07-15 | 2011-01-20 | 帝人ファーマ株式会社 | 貧溶媒添加法による2-(3-シアノ-4-イソブチルオキシフェニル)-4-メチル-5-チアゾールカルボン酸の結晶多形体の製造方法 |
| JP5519201B2 (ja) * | 2009-07-15 | 2014-06-11 | 光孝 北村 | 2−(3−シアノ−4−イソブチルオキシフェニル)−4−メチル−5−チアゾールカルボン酸の結晶多形体の製造方法 |
| KR101800054B1 (ko) * | 2010-08-27 | 2017-11-21 | 데이진 화-마 가부시키가이샤 | 팔라듐 화합물을 사용한 커플링법에 의한 페닐 치환 복소 고리 유도체의 제조법 |
| US9637469B2 (en) * | 2012-11-14 | 2017-05-02 | Teijin Pharma Limited | Pyridine derivative |
-
2015
- 2015-05-12 US US15/310,217 patent/US20170144987A1/en not_active Abandoned
- 2015-05-12 JP JP2016519263A patent/JP6289619B2/ja not_active Expired - Fee Related
- 2015-05-12 EP EP15792728.6A patent/EP3144304A4/en not_active Withdrawn
- 2015-05-12 AR ARP150101454A patent/AR100404A1/es unknown
- 2015-05-12 SG SG11201609483YA patent/SG11201609483YA/en unknown
- 2015-05-12 CA CA2948792A patent/CA2948792A1/en not_active Abandoned
- 2015-05-12 TW TW104115029A patent/TW201625580A/zh unknown
- 2015-05-12 KR KR1020167031454A patent/KR20170003569A/ko not_active Withdrawn
- 2015-05-12 WO PCT/JP2015/063632 patent/WO2015174411A1/ja not_active Ceased
- 2015-05-12 MX MX2016014692A patent/MX2016014692A/es unknown
- 2015-05-12 CN CN201580024742.0A patent/CN106458970B/zh not_active Expired - Fee Related
- 2015-05-12 RU RU2016148736A patent/RU2016148736A/ru not_active Application Discontinuation
- 2015-05-12 AU AU2015260294A patent/AU2015260294A1/en not_active Abandoned
-
2016
- 2016-11-09 PH PH12016502222A patent/PH12016502222A1/en unknown
- 2016-11-10 IL IL248901A patent/IL248901A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| SG11201609483YA (en) | 2016-12-29 |
| CN106458970B (zh) | 2019-09-13 |
| RU2016148736A3 (es) | 2018-06-14 |
| US20170144987A1 (en) | 2017-05-25 |
| CN106458970A (zh) | 2017-02-22 |
| MX2016014692A (es) | 2017-02-23 |
| EP3144304A1 (en) | 2017-03-22 |
| IL248901A0 (en) | 2017-01-31 |
| RU2016148736A (ru) | 2018-06-14 |
| AU2015260294A1 (en) | 2017-01-05 |
| JPWO2015174411A1 (ja) | 2017-04-20 |
| TW201625580A (zh) | 2016-07-16 |
| KR20170003569A (ko) | 2017-01-09 |
| EP3144304A4 (en) | 2017-10-25 |
| WO2015174411A1 (ja) | 2015-11-19 |
| PH12016502222A1 (en) | 2017-02-06 |
| JP6289619B2 (ja) | 2018-03-07 |
| CA2948792A1 (en) | 2015-11-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |