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AR095260A1 - Composiciones de anfetaminas transdérmicas estables y métodos de fabricación - Google Patents

Composiciones de anfetaminas transdérmicas estables y métodos de fabricación

Info

Publication number
AR095260A1
AR095260A1 ARP140100872A ARP140100872A AR095260A1 AR 095260 A1 AR095260 A1 AR 095260A1 AR P140100872 A ARP140100872 A AR P140100872A AR P140100872 A ARP140100872 A AR P140100872A AR 095260 A1 AR095260 A1 AR 095260A1
Authority
AR
Argentina
Prior art keywords
amphetamine
compositions
composition
polymer
group
Prior art date
Application number
ARP140100872A
Other languages
English (en)
Inventor
Patel Prashant
Nguyen Viet
Liao Jun
Original Assignee
Noven Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Noven Pharma filed Critical Noven Pharma
Publication of AR095260A1 publication Critical patent/AR095260A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7007Drug-containing films, membranes or sheets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61LMETHODS OR APPARATUS FOR STERILISING MATERIALS OR OBJECTS IN GENERAL; DISINFECTION, STERILISATION OR DEODORISATION OF AIR; CHEMICAL ASPECTS OF BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES; MATERIALS FOR BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES
    • A61L31/00Materials for other surgical articles, e.g. stents, stent-grafts, shunts, surgical drapes, guide wires, materials for adhesion prevention, occluding devices, surgical gloves, tissue fixation devices
    • A61L31/12Composite materials, i.e. containing one material dispersed in a matrix of the same or different material
    • A61L31/125Composite materials, i.e. containing one material dispersed in a matrix of the same or different material having a macromolecular matrix
    • A61L31/129Composite materials, i.e. containing one material dispersed in a matrix of the same or different material having a macromolecular matrix containing macromolecular fillers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061Polyacrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Vascular Medicine (AREA)
  • Surgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Materials Engineering (AREA)
  • Composite Materials (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Composiciones de fármacos que comprenden anfetamina para administración transdérmica, métodos para preparar composiciones de fármacos que comprenden anfetamina para administración transdérmica, y métodos terapéuticos para utilizarlos. En formas de realización específicas, las composiciones están libres de componentes con unidades que reaccionan con la anfetamina. En formas de realización no específicas, las composiciones se fabrican usando solventes libres de componentes con unidades que reaccionan con la anfetamina. También se describen métodos terapéuticos usando las composiciones. Reivindicación 1: Una composición para la administración transdérmica de anfetamina en la forma de un sistema finito flexible para aplicación tópica, que comprende una matriz de polímero que comprende anfetamina o una sal farmacéuticamente aceptable o una prodroga de la misma, donde la matriz de polímero comprende un polímero que está libre de unidades de acetato de vinilo. Reivindicación 2: La composición de la reivindicación 1, en donde el polímero se selecciona entre el grupo formado por los polímeros de acrílico que están libres de unidades de acetato de vinilo, polímeros a base de gomas, y mezclas de los mismos. Reivindicación 3: La composición de la reivindicación 2, en donde el polímero comprende un polímero de acrílico formado a partir de uno o más monómeros que se seleccionan entre el grupo que consiste en acrilato de butilo, acrilato de metilo, metacrilato de metilo, ácido acrílico, acrilato de etil hexilo, y acrilato de hidroxietilo. Reivindicación 9: La composición de la reivindicación 7, en donde el antioxidante se selecciona entre el grupo formado por hidroxitolueno butilado (BHT), hidroxianisol butilado (BHA), y mezclas de los mismos. Reivindicación 10: La composición de cualquiera de las reivindicaciones 1 - 6, en donde la matriz de polímero comprende además un componente que se selecciona entre el grupo que consiste en dióxido de silicio, resinas de hidrocarburo hidrogenado, y copolímeros de bloques estireno-isobutileno-estireno.
ARP140100872A 2013-03-15 2014-03-12 Composiciones de anfetaminas transdérmicas estables y métodos de fabricación AR095260A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361790077P 2013-03-15 2013-03-15

Publications (1)

Publication Number Publication Date
AR095260A1 true AR095260A1 (es) 2015-09-30

Family

ID=50391537

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP140100872A AR095260A1 (es) 2013-03-15 2014-03-12 Composiciones de anfetaminas transdérmicas estables y métodos de fabricación

Country Status (9)

Country Link
US (3) US20140322298A1 (es)
EP (1) EP2968198B1 (es)
AR (1) AR095260A1 (es)
AU (1) AU2014235057B2 (es)
CA (1) CA2905907C (es)
ES (1) ES2702879T3 (es)
MX (1) MX375186B (es)
TW (1) TWI677341B (es)
WO (1) WO2014151387A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014106014A1 (en) 2012-12-28 2014-07-03 Noven Pharmaceuticals, Inc Transdermal drug delivery systems for levonorgestrel and ethinyl estradiol
AR095260A1 (es) 2013-03-15 2015-09-30 Noven Pharma Composiciones de anfetaminas transdérmicas estables y métodos de fabricación
AU2015296807A1 (en) 2014-07-31 2017-03-09 Noven Pharmaceuticals, Inc. Silicone-containing acrylic polymers for transdermal drug delivery compositions
US10406116B2 (en) 2015-02-06 2019-09-10 Noven Pharmaceuticals, Inc. Pressure-sensitive adhesives for transdermal drug delivery
CA2975452C (en) 2015-02-06 2024-03-12 Noven Pharmaceuticals, Inc. Pressure-sensitive adhesives for transdermal drug delivery
CN116997330A (zh) 2021-01-07 2023-11-03 诺芬药品公司 具有低水平氨基甲酸盐的透皮安非他命组合物
WO2022150431A2 (en) 2021-01-07 2022-07-14 Noven Pharmaceuticals, Inc. Amphetamine carbamate compounds and methods

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US5234957A (en) 1991-02-27 1993-08-10 Noven Pharmaceuticals, Inc. Compositions and methods for topical administration of pharmaceutically active agents
US5446070A (en) 1991-02-27 1995-08-29 Nover Pharmaceuticals, Inc. Compositions and methods for topical administration of pharmaceutically active agents
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US5719197A (en) 1988-03-04 1998-02-17 Noven Pharmaceuticals, Inc. Compositions and methods for topical administration of pharmaceutically active agents
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CA2331264C (en) 1999-01-14 2008-09-23 Noven Pharmaceuticals, Inc. Compositions and methods for drug delivery
US20030104041A1 (en) * 1999-12-16 2003-06-05 Tsung-Min Hsu Transdermal and topical administration of drugs using basic permeation enhancers
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ME00114B (me) 2003-10-28 2011-02-10 Noven Pharma Kompozicije i postupci za kontrolisanje gubitka i oslobađanja lijeka u transdermalnim sistemima oslobađanja lijeka
TW200616589A (en) 2004-10-08 2006-06-01 Noven Pharma Transdermal delivery of drugs based on crystal size
WO2006041907A2 (en) 2004-10-08 2006-04-20 Noven Pharmaceuticals, Inc. Transdermal delivery of estradiol
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MX2008010934A (es) * 2006-02-27 2008-10-30 Noven Pharma Sistema terapeutico transdermico que contiene escopolamina.
AU2007317629A1 (en) 2006-10-27 2008-05-15 Noven Pharmaceuticals, Inc. Transdermal delivery of ketoprofen polar derivatives
AU2008335809A1 (en) * 2007-12-06 2009-06-18 Durect Corporation Methods useful for the treatment of pain, arthritic conditions, or inflammation associated with a chronic condition
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AR095258A1 (es) 2013-03-14 2015-09-30 Noven Pharma Composiciones transdérmicas de metilfenidato con adhesivos a base de goma
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AR095260A1 (es) 2013-03-15 2015-09-30 Noven Pharma Composiciones de anfetaminas transdérmicas estables y métodos de fabricación
AR095259A1 (es) 2013-03-15 2015-09-30 Noven Pharma Composiciones y métodos para la administración transdérmica de fármacos de amina terciaria

Also Published As

Publication number Publication date
WO2014151387A1 (en) 2014-09-25
AU2014235057A1 (en) 2015-10-08
AU2014235057B2 (en) 2019-01-03
US20140322298A1 (en) 2014-10-30
EP2968198B1 (en) 2018-11-21
MX375186B (es) 2025-03-06
US11376327B2 (en) 2022-07-05
US20180207280A1 (en) 2018-07-26
US20220370619A1 (en) 2022-11-24
CA2905907C (en) 2021-05-11
ES2702879T3 (es) 2019-03-06
MX2015013187A (es) 2016-04-04
TW201521715A (zh) 2015-06-16
EP2968198A1 (en) 2016-01-20
HK1220608A1 (en) 2017-05-12
TWI677341B (zh) 2019-11-21
CA2905907A1 (en) 2014-09-25

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