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AR089020A1 - Agentes de reversion anticoagulante - Google Patents

Agentes de reversion anticoagulante

Info

Publication number
AR089020A1
AR089020A1 ARP120104474A ARP120104474A AR089020A1 AR 089020 A1 AR089020 A1 AR 089020A1 AR P120104474 A ARP120104474 A AR P120104474A AR P120104474 A ARP120104474 A AR P120104474A AR 089020 A1 AR089020 A1 AR 089020A1
Authority
AR
Argentina
Prior art keywords
different
same
compound
anticoagulating
absent
Prior art date
Application number
ARP120104474A
Other languages
English (en)
Inventor
E Laulicht Bryan
H Bakhru Sasha
Mathiowitz Edith
S Steiner Solomon
Original Assignee
Perosphere Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47430065&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR089020(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Perosphere Inc filed Critical Perosphere Inc
Publication of AR089020A1 publication Critical patent/AR089020A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/12Ketones
    • A61K31/122Ketones having the oxygen directly attached to a ring, e.g. quinones, vitamin K1, anthralin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Vascular Medicine (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Reivindicación 1: Un compuesto de la fórmula (1): Y-M-X-L-A-L-X-M-Y (1) o una sal farmacéuticamente aceptable de la misma, donde: A es un anillo carbocíclico o heterocíclico, aromático o no aromático, sustituido o no sustituido o un resto lineal; L y L son iguales o diferentes y son enlaces; X y X son iguales o diferentes y están ausentes o son un grupo funcional que une el enlace L a M y el enlace L a M, respectivamente; M y M son iguales o diferentes y están ausentes o son un enlace que une X a Y y X a Y, respectivamente; e Y e Y son iguales o diferentes y son un resto que contiene uno o más átomos o grupos catiónicos o uno o más grupos que se vuelven catiónicos en condiciones fisiológicas. Reivindicación 6: El compuesto de la reivindicación 1, donde el compuesto está representado por la fórmula (2) o una sal farmacéuticamente aceptable de este.
ARP120104474A 2011-11-29 2012-11-29 Agentes de reversion anticoagulante AR089020A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201161564559P 2011-11-29 2011-11-29
US201261614292P 2012-03-22 2012-03-22
US201261641698P 2012-05-02 2012-05-02
US201261666291P 2012-06-29 2012-06-29

Publications (1)

Publication Number Publication Date
AR089020A1 true AR089020A1 (es) 2014-07-23

Family

ID=47430065

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP120104474A AR089020A1 (es) 2011-11-29 2012-11-29 Agentes de reversion anticoagulante

Country Status (34)

Country Link
US (5) US9522892B2 (es)
EP (1) EP2785700B1 (es)
JP (1) JP6134731B2 (es)
KR (1) KR101892330B1 (es)
CN (1) CN104080772B (es)
AP (1) AP2014007662A0 (es)
AR (1) AR089020A1 (es)
AU (1) AU2012345975B2 (es)
BR (1) BR112014012892B1 (es)
CA (1) CA2856540C (es)
CL (1) CL2014001399A1 (es)
CO (1) CO6990738A2 (es)
CR (1) CR20140310A (es)
CY (1) CY1117414T1 (es)
DK (1) DK2785700T3 (es)
EA (1) EA027603B1 (es)
EC (1) ECSP14006696A (es)
ES (1) ES2569674T3 (es)
HR (1) HRP20160513T1 (es)
HU (1) HUE027452T2 (es)
IL (1) IL232788B (es)
ME (1) ME02424B (es)
MX (1) MX349514B (es)
PE (1) PE20141295A1 (es)
PH (1) PH12014501176A1 (es)
PL (1) PL2785700T3 (es)
PT (1) PT2785700E (es)
RS (1) RS54738B1 (es)
SG (1) SG11201402713WA (es)
SI (1) SI2785700T1 (es)
SM (1) SMT201600161B (es)
UA (1) UA116336C2 (es)
WO (1) WO2013082210A1 (es)
ZA (1) ZA201404793B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015069844A1 (en) * 2013-11-08 2015-05-14 Perosphere Inc. Labeled compounds and methods of imaging, diagnosing cartilage disorders and diseases, and monitoring cartilage health using labeled and unlabeled compounds
HUE064656T2 (hu) 2016-03-28 2024-04-28 Incyte Corp Pirrolotriazin vegyületek mint TAM inhibitorok
KR102739325B1 (ko) 2017-09-27 2024-12-09 인사이트 코포레이션 Tam 억제제로서 유용한 피롤로트리아진 유도체의 염
AU2018365257B2 (en) * 2017-11-13 2021-05-13 Maximum Fidelity Surgical Simulations, Inc. Reconstitution of post mortem circulation, specialized methods and procedures
ES3031110T3 (en) 2018-06-29 2025-07-04 Incyte Corp Formulations of an axl/mer inhibitor
US11716989B2 (en) 2019-04-16 2023-08-08 Maximum Fidelity Surgical Simulations, LLC Cadaver preservation systems and methods
WO2020232402A1 (en) 2019-05-15 2020-11-19 Maximum Fidelity Surgical Simulations, LLC Cadaverous heart model
CN112010930B (zh) * 2019-05-28 2022-08-02 首都医科大学 Rgd修饰的五环哌嗪二酮及其制备和应用
AU2021230385A1 (en) 2020-03-06 2022-09-22 Incyte Corporation Combination therapy comprising AXL/MER and PD-1/PD-L1 inhibitors
CN118684672A (zh) 2023-03-24 2024-09-24 陕西麦科奥特科技有限公司 一种抗凝逆转剂及其制备方法和应用
CN117624137A (zh) * 2023-12-04 2024-03-01 中国药科大学 三嗪骨架小分子肝素逆转剂及其制备方法与用途
US20250389737A1 (en) * 2024-06-20 2025-12-25 Instrumentation Laboratory Company FACTOR Xa REAGENT
EP4667582A1 (en) * 2024-06-20 2025-12-24 Instrumentation Laboratory Company Factor xa reagent

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IL115420A0 (en) * 1994-09-26 1995-12-31 Zeneca Ltd Aminoheterocyclic derivatives
US6069232A (en) * 1995-10-02 2000-05-30 Hoechst Marion Roussel, Inc. Polyfluoroalkyl tryptophan tripeptide thrombin inhibitors
US6080852A (en) 1996-06-27 2000-06-27 The Perkin-Elmer Corporation 4,7-dichlororhodamine dyes
AU743735B2 (en) 1996-10-11 2002-02-07 Millennium Pharmaceuticals, Inc. Selective factor Xa inhibitors
SI20115A (sl) * 1997-04-07 2000-06-30 Axys Pharmaceuticals, Inc. Spojine in sestavki za zdravljenje bolezni, povezanih z aktivnostjo serinskih proteaz, zlasti triptaze
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KR20010113969A (ko) 1999-05-19 2001-12-28 추후보정 항응고제로서의 치환된 폴리시클릭 아릴 및 헤테로아릴우라실
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Also Published As

Publication number Publication date
CO6990738A2 (es) 2014-07-10
AU2012345975A1 (en) 2014-05-29
ES2569674T3 (es) 2016-05-12
RS54738B1 (sr) 2016-10-31
AU2012345975B2 (en) 2016-12-15
DK2785700T3 (en) 2016-06-13
HRP20160513T1 (hr) 2016-07-15
EP2785700B1 (en) 2016-03-09
PT2785700E (pt) 2016-06-02
BR112014012892B1 (pt) 2022-12-20
EA027603B1 (ru) 2017-08-31
BR112014012892A2 (pt) 2017-06-13
KR101892330B1 (ko) 2018-08-27
UA116336C2 (uk) 2018-03-12
US20240366592A1 (en) 2024-11-07
US20130137702A1 (en) 2013-05-30
PH12014501176B1 (en) 2014-09-01
HUE027452T2 (en) 2016-09-28
US20210169874A1 (en) 2021-06-10
EA201490823A1 (ru) 2015-01-30
IL232788A0 (en) 2014-08-03
CY1117414T1 (el) 2017-04-26
IL232788B (en) 2018-05-31
CA2856540C (en) 2018-04-03
PH12014501176A1 (en) 2014-09-01
US9522892B2 (en) 2016-12-20
CN104080772A (zh) 2014-10-01
HK1202858A1 (en) 2015-10-09
NZ625337A (en) 2016-11-25
CL2014001399A1 (es) 2014-11-03
US20180207152A1 (en) 2018-07-26
BR112014012892A8 (pt) 2021-06-08
KR20140107259A (ko) 2014-09-04
EP2785700A1 (en) 2014-10-08
US9877961B2 (en) 2018-01-30
SG11201402713WA (en) 2014-06-27
SI2785700T1 (sl) 2016-09-30
PL2785700T3 (pl) 2016-09-30
WO2013082210A1 (en) 2013-06-06
ME02424B (me) 2016-09-20
ZA201404793B (en) 2015-04-29
MX349514B (es) 2017-08-02
CN104080772B (zh) 2016-10-05
JP2014534270A (ja) 2014-12-18
CR20140310A (es) 2014-08-20
MX2014006349A (es) 2014-09-04
AP2014007662A0 (en) 2014-05-31
ECSP14006696A (es) 2015-06-30
US20170056396A1 (en) 2017-03-02
SMT201600161B (it) 2016-07-01
CA2856540A1 (en) 2013-06-06
JP6134731B2 (ja) 2017-05-24
PE20141295A1 (es) 2014-10-01

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