AR070653A1 - Derivados de imidazolina y su uso como agentes biocidas - Google Patents
Derivados de imidazolina y su uso como agentes biocidasInfo
- Publication number
- AR070653A1 AR070653A1 ARP080104058A ARP080104058A AR070653A1 AR 070653 A1 AR070653 A1 AR 070653A1 AR P080104058 A ARP080104058 A AR P080104058A AR P080104058 A ARP080104058 A AR P080104058A AR 070653 A1 AR070653 A1 AR 070653A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- optionally substituted
- alkoxy
- r14r15n
- r7r8n
- Prior art date
Links
- 150000002462 imidazolines Chemical class 0.000 title abstract 3
- 229940083254 peripheral vasodilators imidazoline derivative Drugs 0.000 title abstract 3
- 239000003139 biocide Substances 0.000 title 1
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 4
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
- 125000000623 heterocyclic group Chemical group 0.000 abstract 3
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 3
- 125000000008 (C1-C10) alkyl group Chemical group 0.000 abstract 2
- ZCYVEMRRCGMTRW-UHFFFAOYSA-N 7553-56-2 Chemical group [I] ZCYVEMRRCGMTRW-UHFFFAOYSA-N 0.000 abstract 2
- 230000000895 acaricidal effect Effects 0.000 abstract 2
- 125000000304 alkynyl group Chemical group 0.000 abstract 2
- 102220389089 c.33G>T Human genes 0.000 abstract 2
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 2
- 125000000392 cycloalkenyl group Chemical group 0.000 abstract 2
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 2
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 230000000749 insecticidal effect Effects 0.000 abstract 2
- 229910052740 iodine Chemical group 0.000 abstract 2
- 239000011630 iodine Chemical group 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 229910052717 sulfur Inorganic materials 0.000 abstract 2
- NJYFRQQXXXRJHK-UHFFFAOYSA-N (4-aminophenyl) thiocyanate Chemical compound NC1=CC=C(SC#N)C=C1 NJYFRQQXXXRJHK-UHFFFAOYSA-N 0.000 abstract 1
- 125000006583 (C1-C3) haloalkyl group Chemical group 0.000 abstract 1
- 125000006274 (C1-C3)alkoxy group Chemical group 0.000 abstract 1
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
- 125000006272 (C3-C7) cycloalkyl group Chemical group 0.000 abstract 1
- 241000238876 Acari Species 0.000 abstract 1
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
- 125000006577 C1-C6 hydroxyalkyl group Chemical group 0.000 abstract 1
- 125000006374 C2-C10 alkenyl group Chemical group 0.000 abstract 1
- 241000238631 Hexapoda Species 0.000 abstract 1
- 241000237852 Mollusca Species 0.000 abstract 1
- 150000001204 N-oxides Chemical class 0.000 abstract 1
- 241000244206 Nematoda Species 0.000 abstract 1
- 241000607479 Yersinia pestis Species 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Chemical group BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
- 229910052794 bromium Inorganic materials 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 239000000460 chlorine Substances 0.000 abstract 1
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- ATDGTVJJHBUTRL-UHFFFAOYSA-N cyanogen bromide Chemical compound BrC#N ATDGTVJJHBUTRL-UHFFFAOYSA-N 0.000 abstract 1
- 125000000262 haloalkenyl group Chemical group 0.000 abstract 1
- 125000001188 haloalkyl group Chemical group 0.000 abstract 1
- 125000004995 haloalkylthio group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical group 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 230000001069 nematicidal effect Effects 0.000 abstract 1
- 239000005645 nematicide Substances 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 102220315634 rs1196125127 Human genes 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000003107 substituted aryl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/06—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms
- C07D233/08—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms with alkyl radicals, containing more than four carbon atoms, directly attached to ring carbon atoms
- C07D233/12—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms with alkyl radicals, containing more than four carbon atoms, directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D233/16—Radicals substituted by nitrogen atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Derivados de imidazolina y su uso como agentes insecticidas, acaricidas, moluscidas y nematicidas, también se extiende a composiciones insecticidas, acaricidas, moluscidas y nematicidas que comprenden dichos derivados de imidazolina, y a los métodos de uso de dichos derivados y/o composiciones para combatir y controlar las plagas de insectos, ácaros, moluscos y nematodos. Reivindicacion 1: Un compuesto de formula (1) y las sales y N-oxidos del mismo, donde: R1 es alquilo C1-10; R2 es cloro, bromo o yodo; R3 es alquilo C2-5, haloalquilo C1-5, hidroxialquilo C1-6, alcoxi C1-5-alquilo C1-3, di-alcoxi C1-5-alquilo C1-3, alquiltio C1-5-alquilo C1-3; alquilsulfinilo C1-5-aIquiIo C1-3; alquenilo C2-5, haloalquenilo C1-5, alquinilo C2-5, cicloalquilo C3-6, cicloalquenilo C3-6, hidroxi, alcoxi C1-15, haloalcoxi C1-5, alquiltio C1-5, haloalquiltio C1-.5, formilo, ciano, bromo o yodo; Z es hidrogeno, hidroxi, nitro, ciano, rodano, formilo, G-, G-S-, G-S-S-, G-A, R7R8N-, R7R8N-S-, R7R8N-A-, G-O-A-, G-S-A-, (R10O)(R11O)P(X)-, (R10O)(R11S)P(X)-, (R10O)(R11)P(X)-, (R10S)(R11S)P(X)-, (R10O)(R14R15N)P(X)-, (R11)(R14R15N)P(X)-, (R14R15N)(R16R17N)P(X)-., G-N=CH-, G-O-N=CH-, N:::C- N=CH-, o Z es un grupo de formula (2) donde B es S-, S-S-, S(O)-, C(O)- o (CH2)n-; n es un numero entero de 1 a 6; y R1, R2 y R3 son segun se definio anteriormente; y G es alquilo C1-10 opcionalmente sustituido, alquenilo C2-10 opcionalmente sustituido, alquinilo C2-10 opcionalmente sustituido, cicloalquilo C3-7 opcionalmente sustituido, cicloalquenilo C3-7 opcionalmente sustituido, arilo opcionalmente sustituido, heteroarilo opcionalmente sustituido o heterociclilo opcionalmente sustituido; A es S(O), SO2, C(O) o C(S); R7 y R8 son cada uno independientemente hidrogeno o G; R7 y R8 junto con el átomo N al cual están unidos forman un grupo N=CR12R13; o R7 y R8 junto con el átomo N al cual están unidos forman un anillo heterocíclico de cinco, seis o siete miembros, dicho anillo heterocíclico opcionalmente contiene uno o dos heteroátomos adicionales seleccionados a partir de O, N o S, y está opcionalmente sustituido con uno o dos grupos alquilo C1-6; R10 y R11 son cada uno independientemente alquilo C1-6, bencilo o fenilo, donde el grupo fenilo está opcionalmente sustituido con halogeno, nitro, ciano, alquilo C1-3, haloalquilo C1-3, alcoxi C1-3, haloalcoxi C1-3; R12, R13, R14, R15, R16 y R17 son cada uno independientemente hidrogeno o alquilo C1-6; X es O o S.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0718196A GB0718196D0 (en) | 2007-09-18 | 2007-09-18 | Chemical compounds |
| GB0721772A GB0721772D0 (en) | 2007-11-06 | 2007-11-06 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR070653A1 true AR070653A1 (es) | 2010-04-28 |
Family
ID=40210429
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080104058A AR070653A1 (es) | 2007-09-18 | 2008-09-18 | Derivados de imidazolina y su uso como agentes biocidas |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8455663B2 (es) |
| EP (1) | EP2190823B1 (es) |
| JP (1) | JP2010539114A (es) |
| CN (1) | CN101835758A (es) |
| AR (1) | AR070653A1 (es) |
| CL (1) | CL2008002764A1 (es) |
| RU (1) | RU2010115182A (es) |
| TW (1) | TW200922472A (es) |
| UY (1) | UY31348A1 (es) |
| WO (1) | WO2009036909A1 (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1958507A1 (en) * | 2007-02-15 | 2008-08-20 | Syngeta Participations AG | Chemical compounds |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS51106739A (en) * | 1975-03-12 | 1976-09-21 | Takeda Chemical Industries Ltd | Satsuchu satsudanizai |
| US4226876A (en) * | 1976-12-20 | 1980-10-07 | Burroughs Wellcome Co. | Arthropodicidal imidazoline derivatives |
| GB1593276A (en) | 1976-12-20 | 1981-07-15 | Wellcome Found | Imidazoline derivatives and their use as pesticides |
| GB1592649A (en) | 1976-12-20 | 1981-07-08 | Wellcome Found | Imidazoline derivatives and their use as pesticides |
| DE2756638A1 (de) | 1976-12-20 | 1978-06-22 | Wellcome Found | Imidazoline, verfahren zu ihrer herstellung und ihre verwendung in schaedlingsbekaempfungsmitteln |
| AU3546478A (en) * | 1977-04-29 | 1979-11-01 | Ciba Geigy Ag | Ectoparasiticides |
| GB2023603B (en) | 1978-06-19 | 1982-10-20 | Wellcome Found | Pesticidal imidazolienes and their preparation and use |
| EP0008071B1 (de) | 1978-08-14 | 1982-01-20 | Ciba-Geigy Ag | 1-Iminomethylen-substituierte 2-(Phenoxy-alkyl)-2-imidazolinderivate, Verfahren zu ihrer Herstellung, Mittel, welche diese Derivate als aktive Komponente enthalten und ihre Verwendung zur Bekämpfung von Schädlingen |
| EP0008565A1 (de) * | 1978-08-28 | 1980-03-05 | Ciba-Geigy Ag | Bis-(phenoxy-alkyl-2-imidazolin)-1,1'-sulfide, Verfahren zu ihrer Herstellung, Mittel welche diese Sulfide als aktive Komponente enthalten und deren Verwendung zur Bekämpfung von Schädlingen |
| US4241075A (en) * | 1978-09-27 | 1980-12-23 | Ciba-Geigy Corporation | Acaricidal 1-alkylthio-substituted and 1-phenylthio substituted 2-(phenoxyalkyl)-2-imidazolines |
| DE2940167A1 (de) | 1978-10-06 | 1980-04-17 | Ciba Geigy Ag | 2-imidazolinderivate mit pestizider wirkung |
| DE2961710D1 (en) | 1978-10-09 | 1982-02-18 | Ciba Geigy Ag | 2-(alpha-phenoxy-alkyl)-imidazolines and their salts, their preparation and use, and agents against phytoparasitic and zooparasitic mites containing them |
| US4232011A (en) * | 1978-11-02 | 1980-11-04 | Ciba-Geigy Corporation | 1-Phosphorylated 2-(phenoxyalkyl)-2-imidazoline derivatives and their use in pest control |
| DE3038395A1 (de) | 1980-10-10 | 1982-05-19 | Bayer Ag, 5090 Leverkusen | 2-(2,3-dimethyl-phenoxymethyl)-2-imidazolin enthaltendes anthelmintikum |
| DE3842798A1 (de) * | 1988-12-20 | 1990-06-21 | Hoechst Ag | Imidazolinderivate enthaltende mittel zur wirtstiersystemischen bekaempfung von ektoparasiten sowie neue imidazolinderivate |
| EP1958507A1 (en) | 2007-02-15 | 2008-08-20 | Syngeta Participations AG | Chemical compounds |
| EP1958508A1 (en) | 2007-02-16 | 2008-08-20 | Syngeta Participations AG | Phenoxymethyl imidazoline derivatives and their use as pesticides |
-
2008
- 2008-09-09 WO PCT/EP2008/007363 patent/WO2009036909A1/en not_active Ceased
- 2008-09-09 CN CN200880113281A patent/CN101835758A/zh active Pending
- 2008-09-09 EP EP08801936A patent/EP2190823B1/en not_active Not-in-force
- 2008-09-09 JP JP2010524388A patent/JP2010539114A/ja active Pending
- 2008-09-09 RU RU2010115182/04A patent/RU2010115182A/ru not_active Application Discontinuation
- 2008-09-09 US US12/677,825 patent/US8455663B2/en not_active Expired - Fee Related
- 2008-09-09 TW TW097134497A patent/TW200922472A/zh unknown
- 2008-09-16 CL CL2008002764A patent/CL2008002764A1/es unknown
- 2008-09-18 UY UY31348A patent/UY31348A1/es unknown
- 2008-09-18 AR ARP080104058A patent/AR070653A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CN101835758A (zh) | 2010-09-15 |
| EP2190823A1 (en) | 2010-06-02 |
| TW200922472A (en) | 2009-06-01 |
| UY31348A1 (es) | 2009-04-30 |
| CL2008002764A1 (es) | 2009-07-17 |
| EP2190823B1 (en) | 2012-07-11 |
| US20100280088A1 (en) | 2010-11-04 |
| WO2009036909A1 (en) | 2009-03-26 |
| US8455663B2 (en) | 2013-06-04 |
| RU2010115182A (ru) | 2011-10-27 |
| JP2010539114A (ja) | 2010-12-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |