AR070456A1 - Combinacion que comprende paclitaxel para el tratamiento de cancer de ovario y su uso - Google Patents
Combinacion que comprende paclitaxel para el tratamiento de cancer de ovario y su usoInfo
- Publication number
- AR070456A1 AR070456A1 ARP090100596A ARP090100596A AR070456A1 AR 070456 A1 AR070456 A1 AR 070456A1 AR P090100596 A ARP090100596 A AR P090100596A AR P090100596 A ARP090100596 A AR P090100596A AR 070456 A1 AR070456 A1 AR 070456A1
- Authority
- AR
- Argentina
- Prior art keywords
- treatment
- cancer
- ovary
- combination including
- including paclitaxel
- Prior art date
Links
- 206010033128 Ovarian cancer Diseases 0.000 title abstract 2
- 206010061535 Ovarian neoplasm Diseases 0.000 title abstract 2
- 229930012538 Paclitaxel Natural products 0.000 title abstract 2
- 229960001592 paclitaxel Drugs 0.000 title abstract 2
- RCINICONZNJXQF-MZXODVADSA-N taxol Chemical compound O([C@@H]1[C@@]2(C[C@@H](C(C)=C(C2(C)C)[C@H](C([C@]2(C)[C@@H](O)C[C@H]3OC[C@]3([C@H]21)OC(C)=O)=O)OC(=O)C)OC(=O)[C@H](O)[C@@H](NC(=O)C=1C=CC=CC=1)C=1C=CC=CC=1)O)C(=O)C1=CC=CC=C1 RCINICONZNJXQF-MZXODVADSA-N 0.000 title abstract 2
- 229940118365 Endothelin receptor antagonist Drugs 0.000 abstract 1
- 239000002308 endothelin receptor antagonist Substances 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Emergency Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Combinacion de un antagonista de receptor de endotelina de formula (1) con paclitaxel, para uso terapéutico, de manera simultánea, separada o durante un período de tiempo, en el tratamiento de cáncer de ovarios.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IB2008050607 | 2008-02-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR070456A1 true AR070456A1 (es) | 2010-04-07 |
Family
ID=40670930
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP090100596A AR070456A1 (es) | 2008-02-20 | 2009-02-20 | Combinacion que comprende paclitaxel para el tratamiento de cancer de ovario y su uso |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US8541433B2 (es) |
| EP (1) | EP2254570B1 (es) |
| JP (1) | JP5514123B2 (es) |
| KR (1) | KR20100132489A (es) |
| CN (1) | CN101939001B (es) |
| AR (1) | AR070456A1 (es) |
| AU (1) | AU2009215329B2 (es) |
| CA (1) | CA2714608A1 (es) |
| CY (1) | CY1115071T1 (es) |
| DK (1) | DK2254570T3 (es) |
| ES (1) | ES2446303T3 (es) |
| HR (1) | HRP20140215T1 (es) |
| MX (1) | MX2010008994A (es) |
| PL (1) | PL2254570T3 (es) |
| PT (1) | PT2254570E (es) |
| RU (1) | RU2494736C2 (es) |
| SI (1) | SI2254570T1 (es) |
| TW (1) | TWI441639B (es) |
| WO (1) | WO2009104149A1 (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2292209A3 (en) | 2005-09-12 | 2011-05-04 | Actelion Pharmaceuticals Ltd. | Stable pharmaceutical composition comprising a pyramidine-sulfamide |
| MX2010001837A (es) | 2007-08-17 | 2010-03-10 | Actelion Pharmaceuticals Ltd | Derivados de 4-pirimidinasulfamida. |
| PT2254570E (pt) * | 2008-02-20 | 2014-02-17 | Actelion Pharmaceuticals Ltd | Combinação que compreende paclitaxel para o tratamento de cancro de ovário |
| KR101678699B1 (ko) | 2008-08-13 | 2016-11-23 | 액테리온 파마슈티칼 리미티드 | 마시텐탄을 포함하는 치료 조성물 |
| PT2464218E (pt) | 2009-08-10 | 2015-09-16 | Univ Texas | Tratamento de metástases do cérebro com inibidores de recetores de endotelina, em combinação com um agente quimioterapêutico citotóxico |
| BR112013019680A2 (pt) * | 2011-02-04 | 2016-10-11 | Actelion Pharmaceuticals Ltd | combinações compreendendo macitentana para o tratamento de glioblastoma multiforme |
| CN103819411A (zh) * | 2014-03-14 | 2014-05-28 | 成都克莱蒙医药科技有限公司 | 一种马西替坦中间体新的制备方法 |
| KR102359214B1 (ko) | 2014-04-04 | 2022-02-07 | 델 마 파마슈티컬스 | 폐의 비소세포 암종 및 난소암을 치료하기 위한 디안하이드로갈락티톨 및 이의 유사체 또는 유도체 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW406020B (en) * | 1993-09-29 | 2000-09-21 | Bristol Myers Squibb Co | Stabilized pharmaceutical composition and its method for preparation and stabilizing solvent |
| ATE323079T1 (de) * | 2000-12-18 | 2006-04-15 | Actelion Pharmaceuticals Ltd | Neue sulfamiden und deren verwendung als endothelin-antagonisten |
| CA2502848C (en) | 2002-10-24 | 2012-10-02 | The Board Of Trustees Of The University Of Illinois | Use of irl-1620 and paclitaxel for preventing and treating breast tumors |
| US20040121971A1 (en) * | 2002-12-20 | 2004-06-24 | Gang Chen | Therapeutic use of tumor necrosis factor-alpha mutein |
| GB0425854D0 (en) | 2004-11-25 | 2004-12-29 | Astrazeneca Ab | Therapeutic treatment |
| EP2292209A3 (en) | 2005-09-12 | 2011-05-04 | Actelion Pharmaceuticals Ltd. | Stable pharmaceutical composition comprising a pyramidine-sulfamide |
| AR062501A1 (es) | 2006-08-29 | 2008-11-12 | Actelion Pharmaceuticals Ltd | Composiciones terapeuticas |
| PT2254570E (pt) * | 2008-02-20 | 2014-02-17 | Actelion Pharmaceuticals Ltd | Combinação que compreende paclitaxel para o tratamento de cancro de ovário |
| KR20100005486A (ko) * | 2008-07-07 | 2010-01-15 | 페어차일드코리아반도체 주식회사 | 스위치 제어 장치 및 이를 포함하는 컨버터 |
-
2009
- 2009-02-19 PT PT97123343T patent/PT2254570E/pt unknown
- 2009-02-19 DK DK09712334.3T patent/DK2254570T3/da active
- 2009-02-19 CA CA2714608A patent/CA2714608A1/en not_active Abandoned
- 2009-02-19 JP JP2010547291A patent/JP5514123B2/ja not_active Expired - Fee Related
- 2009-02-19 KR KR1020107018516A patent/KR20100132489A/ko not_active Abandoned
- 2009-02-19 PL PL09712334T patent/PL2254570T3/pl unknown
- 2009-02-19 WO PCT/IB2009/050677 patent/WO2009104149A1/en not_active Ceased
- 2009-02-19 SI SI200930849T patent/SI2254570T1/sl unknown
- 2009-02-19 EP EP09712334.3A patent/EP2254570B1/en not_active Not-in-force
- 2009-02-19 AU AU2009215329A patent/AU2009215329B2/en not_active Ceased
- 2009-02-19 CN CN2009801042583A patent/CN101939001B/zh not_active Expired - Fee Related
- 2009-02-19 US US12/867,939 patent/US8541433B2/en not_active Expired - Fee Related
- 2009-02-19 ES ES09712334.3T patent/ES2446303T3/es active Active
- 2009-02-19 MX MX2010008994A patent/MX2010008994A/es active IP Right Grant
- 2009-02-19 RU RU2010138650/15A patent/RU2494736C2/ru not_active IP Right Cessation
- 2009-02-19 HR HRP20140215AT patent/HRP20140215T1/hr unknown
- 2009-02-19 TW TW098105324A patent/TWI441639B/zh not_active IP Right Cessation
- 2009-02-20 AR ARP090100596A patent/AR070456A1/es unknown
-
2013
- 2013-08-01 US US13/957,126 patent/US20130317048A1/en not_active Abandoned
-
2014
- 2014-02-26 CY CY20141100152T patent/CY1115071T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK2254570T3 (da) | 2014-02-03 |
| TWI441639B (zh) | 2014-06-21 |
| ES2446303T3 (es) | 2014-03-07 |
| AU2009215329B2 (en) | 2014-08-21 |
| KR20100132489A (ko) | 2010-12-17 |
| EP2254570B1 (en) | 2013-12-18 |
| SI2254570T1 (sl) | 2014-03-31 |
| JP5514123B2 (ja) | 2014-06-04 |
| PL2254570T3 (pl) | 2014-05-30 |
| CY1115071T1 (el) | 2016-12-14 |
| HRP20140215T1 (hr) | 2014-04-11 |
| WO2009104149A1 (en) | 2009-08-27 |
| US20130317048A1 (en) | 2013-11-28 |
| TW200940062A (en) | 2009-10-01 |
| EP2254570A1 (en) | 2010-12-01 |
| RU2494736C2 (ru) | 2013-10-10 |
| CN101939001B (zh) | 2012-06-20 |
| MX2010008994A (es) | 2010-09-07 |
| US20100311774A1 (en) | 2010-12-09 |
| RU2010138650A (ru) | 2012-03-27 |
| PT2254570E (pt) | 2014-02-17 |
| JP2011512399A (ja) | 2011-04-21 |
| AU2009215329A1 (en) | 2009-08-27 |
| CA2714608A1 (en) | 2009-08-27 |
| CN101939001A (zh) | 2011-01-05 |
| US8541433B2 (en) | 2013-09-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |