AR070179A1 - DERIVADOS DE PIRIDAZINA, PROCESOS PARA PREPARARLOS, COMPOSICIONES FUNGICIDAS Y FARMACÉUTICAS QUE LOS COMPRENDEN Y SU USO EN MÉTODOS DE PREVENCIoN DE INFESTACIoN DE CULTIVOS Y EN MEDICAMENTOS CONTRA EL CANCER. - Google Patents
DERIVADOS DE PIRIDAZINA, PROCESOS PARA PREPARARLOS, COMPOSICIONES FUNGICIDAS Y FARMACÉUTICAS QUE LOS COMPRENDEN Y SU USO EN MÉTODOS DE PREVENCIoN DE INFESTACIoN DE CULTIVOS Y EN MEDICAMENTOS CONTRA EL CANCER.Info
- Publication number
- AR070179A1 AR070179A1 ARP090100124A ARP090100124A AR070179A1 AR 070179 A1 AR070179 A1 AR 070179A1 AR P090100124 A ARP090100124 A AR P090100124A AR P090100124 A ARP090100124 A AR P090100124A AR 070179 A1 AR070179 A1 AR 070179A1
- Authority
- AR
- Argentina
- Prior art keywords
- derivatives
- fluorine
- piridazine
- fungicide
- prepare
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- 206010028980 Neoplasm Diseases 0.000 title abstract 2
- 201000011510 cancer Diseases 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title abstract 2
- 229940079593 drug Drugs 0.000 title abstract 2
- 230000000855 fungicidal effect Effects 0.000 title abstract 2
- 206010061217 Infestation Diseases 0.000 title 1
- 239000000417 fungicide Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 230000002265 prevention Effects 0.000 title 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical group FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 5
- 229910052731 fluorine Inorganic materials 0.000 abstract 5
- 239000011737 fluorine Chemical group 0.000 abstract 5
- 229910052801 chlorine Inorganic materials 0.000 abstract 4
- 239000000460 chlorine Substances 0.000 abstract 4
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 1
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000003905 agrochemical Substances 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Chemical group BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
- 229910052794 bromium Chemical group 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
- 238000002483 medication Methods 0.000 abstract 1
- 230000003641 microbiacidal effect Effects 0.000 abstract 1
- 150000004892 pyridazines Chemical class 0.000 abstract 1
- 150000003839 salts Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Derivados de piridazina de formula (1) como ingredientes activos los cuales poseen actividad microbicida, en particular actividad fungicida y procedimientos para su obtencion. Estos compuestos son utilizables en agroquímica y en medicamentos para el cáncer. Reivindicacion 1: Un compuesto de formula (1) donde R1 es metilo, etilo o isopropilo; R2 es cloro, fluor, hidroxi o alcoxi C1-2; R3 es H, cloro, fluor, metoxi o alquilo C1-3; R4 es cloro, fluor o bromo; y R5 es H, fluor o metoxi; o su forma de sal utilizable en agroquímica; con la condicion de que cuando R1 es metilo, R2 es cloro y R3 es H, entonces R4 o R5 es diferente de fluor.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0800762.7A GB0800762D0 (en) | 2008-01-16 | 2008-01-16 | Novel pyridazine derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR070179A1 true AR070179A1 (es) | 2010-03-17 |
Family
ID=39165850
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP090100124A AR070179A1 (es) | 2008-01-16 | 2009-01-15 | DERIVADOS DE PIRIDAZINA, PROCESOS PARA PREPARARLOS, COMPOSICIONES FUNGICIDAS Y FARMACÉUTICAS QUE LOS COMPRENDEN Y SU USO EN MÉTODOS DE PREVENCIoN DE INFESTACIoN DE CULTIVOS Y EN MEDICAMENTOS CONTRA EL CANCER. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8410026B2 (es) |
| EP (1) | EP2231637B1 (es) |
| JP (1) | JP2011509960A (es) |
| CN (1) | CN101910149A (es) |
| AR (1) | AR070179A1 (es) |
| AU (1) | AU2009204981A1 (es) |
| CA (1) | CA2711514A1 (es) |
| CL (1) | CL2009000076A1 (es) |
| GB (1) | GB0800762D0 (es) |
| GT (1) | GT200900006A (es) |
| TW (1) | TW200932238A (es) |
| WO (1) | WO2009090039A1 (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0714872A2 (pt) * | 2006-07-17 | 2013-03-19 | Syngenta Participations Ag | derivados de piridazina |
| WO2011095459A1 (en) * | 2010-02-04 | 2011-08-11 | Syngenta Participations Ag | Pyridazine derivatives, process for their preparation and their use as fungicides |
| TWI507381B (zh) | 2010-09-08 | 2015-11-11 | Sumitomo Chemical Co | 製造嗒酮化合物的方法及其中間物 |
| JP2012236875A (ja) * | 2011-05-10 | 2012-12-06 | Dic Corp | 熱硬化性樹脂組成物およびプリント配線板用層間接着フィルム |
| JPWO2012161133A1 (ja) * | 2011-05-20 | 2014-07-31 | 日産化学工業株式会社 | 置換ピリダジン化合物及び農園芸用殺菌剤 |
| AU2018334290A1 (en) | 2017-09-18 | 2020-04-02 | Goldfinch Bio, Inc. | Pyridazinones and methods of use thereof |
| WO2021081923A1 (zh) * | 2019-10-31 | 2021-05-06 | 江苏中旗科技股份有限公司 | 用作杀真菌剂的2-吡啶胺衍生物 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1340685C (en) | 1988-07-29 | 1999-07-27 | Frederick Meins | Dna sequences encoding polypeptides having beta-1,3-glucanase activity |
| EP0392225B1 (en) | 1989-03-24 | 2003-05-28 | Syngenta Participations AG | Disease-resistant transgenic plants |
| US5639949A (en) | 1990-08-20 | 1997-06-17 | Ciba-Geigy Corporation | Genes for the synthesis of antipathogenic substances |
| EA001148B1 (ru) | 1996-03-11 | 2000-10-30 | Новартис Аг | Производные пиримидин-4-она |
| TWI252231B (en) | 1997-04-14 | 2006-04-01 | American Cyanamid Co | Fungicidal trifluorophenyl-triazolopyrimidines |
| DE10215292A1 (de) | 2002-02-19 | 2003-08-28 | Bayer Cropscience Ag | Disubstitutierte Pyrazolylcarbocanilide |
| BR0308230B1 (pt) | 2002-03-05 | 2014-05-20 | Syngenta Participations Ag | O-ciclopropil-carboxanilida, composição e método de controle ou prevenção de infestação de plantas cultivadas por microorganismos fitopatogênicos |
| WO2004016088A2 (en) | 2002-08-12 | 2004-02-26 | Bayer Cropscience S.A. | Novel 2-pyridylethylbenzamide derivative |
| GB0224316D0 (en) | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
| WO2005121104A1 (ja) | 2004-06-09 | 2005-12-22 | Sumitomo Chemical Company, Limited | ピリダジン化合物及びその用途 |
| ATE488506T1 (de) | 2004-06-28 | 2010-12-15 | Sumitomo Chemical Co | Pyridazinverbindung und deren verwendung |
| GB0422401D0 (en) | 2004-10-08 | 2004-11-10 | Syngenta Participations Ag | Fungicidal compositions |
| RU2416609C2 (ru) | 2005-12-07 | 2011-04-20 | Сумитомо Кемикал Компани, Лимитед | Соединение пиридазина и его применение |
| GB0614153D0 (en) | 2006-07-17 | 2006-08-23 | Syngenta Participations Ag | Novel pyridazine derivatives |
-
2008
- 2008-01-16 GB GBGB0800762.7A patent/GB0800762D0/en not_active Ceased
-
2009
- 2009-01-12 GT GT200900006A patent/GT200900006A/es unknown
- 2009-01-14 AU AU2009204981A patent/AU2009204981A1/en not_active Abandoned
- 2009-01-14 CA CA2711514A patent/CA2711514A1/en not_active Abandoned
- 2009-01-14 US US12/863,377 patent/US8410026B2/en not_active Expired - Fee Related
- 2009-01-14 CN CN2009801024547A patent/CN101910149A/zh active Pending
- 2009-01-14 TW TW098101156A patent/TW200932238A/zh unknown
- 2009-01-14 WO PCT/EP2009/000166 patent/WO2009090039A1/en not_active Ceased
- 2009-01-14 EP EP09701980A patent/EP2231637B1/en not_active Not-in-force
- 2009-01-14 JP JP2010542575A patent/JP2011509960A/ja not_active Withdrawn
- 2009-01-15 CL CL2009000076A patent/CL2009000076A1/es unknown
- 2009-01-15 AR ARP090100124A patent/AR070179A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CA2711514A1 (en) | 2009-07-23 |
| CL2009000076A1 (es) | 2009-05-22 |
| TW200932238A (en) | 2009-08-01 |
| US8410026B2 (en) | 2013-04-02 |
| GB0800762D0 (en) | 2008-02-27 |
| CN101910149A (zh) | 2010-12-08 |
| WO2009090039A1 (en) | 2009-07-23 |
| AU2009204981A1 (en) | 2009-07-23 |
| EP2231637A1 (en) | 2010-09-29 |
| EP2231637B1 (en) | 2012-12-19 |
| JP2011509960A (ja) | 2011-03-31 |
| GT200900006A (es) | 2010-04-20 |
| US20110112108A1 (en) | 2011-05-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |