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AR078950A1 - Peptido agonista de la guanilato ciclasa c (gc-c) util para tratamientos de trastornos gastrointestinales - Google Patents

Peptido agonista de la guanilato ciclasa c (gc-c) util para tratamientos de trastornos gastrointestinales

Info

Publication number
AR078950A1
AR078950A1 ARP100104153A ARP100104153A AR078950A1 AR 078950 A1 AR078950 A1 AR 078950A1 AR P100104153 A ARP100104153 A AR P100104153A AR P100104153 A ARP100104153 A AR P100104153A AR 078950 A1 AR078950 A1 AR 078950A1
Authority
AR
Argentina
Prior art keywords
acid
cys
asp
glu
carboxylated
Prior art date
Application number
ARP100104153A
Other languages
English (en)
Original Assignee
Ironwood Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43503086&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR078950(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ironwood Pharmaceuticals Inc filed Critical Ironwood Pharmaceuticals Inc
Publication of AR078950A1 publication Critical patent/AR078950A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/10Peptides having 12 to 20 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C07K14/4701Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
    • C07K14/4702Regulators; Modulating activity
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/08Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Epidemiology (AREA)
  • Zoology (AREA)
  • Toxicology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Nutrition Science (AREA)
  • Neurosurgery (AREA)
  • Obesity (AREA)
  • Neurology (AREA)

Abstract

La presente también provee composiciones y métodos para tratar trastornos gastrointestinales y composiciones farmacéuticas para llevar a cabo dicho métodos. En algunas formas de realizacion, estas composiciones farmacéuticas incluyen formas de dosis orales. Reivindicacion 1: Un péptido o una sal farmacéuticamente aceptable del mismo, en donde el péptido comprende la secuencia de aminoácidos Xaa1 Xaa2 Xaa3 Xaa4 Cys5 Xaa6 Xaa7 Xaa8 Cys9 Asn10 Pro11 Ala12 Cys13 Xaa14 Gly15 Xaa16 Xaa17, o una sal farmacéuticamente aceptable de los mismos; en donde Xaa1 es Asn, D-Asn, Gln, D-Gln, Pro, Ala, Beta-Ala, D-Ala, Val, D-Val, Gly, Thr, D-Thr, Asp, D-Asp, Asp Gama-carboxilado, Glu, D-Glu, Glu Gama-carboxilado, ácido alfa-aminosubérico (Asu), ácido alfa-aminoadípico (Aad), ácido alfa-aminopimélico (Apm), o se halla ausente; Xaa2 es Asp, Asp Gama-carboxilado, Glu, Glu Gama-carboxilado, Asu, Aad, Apm, o se halla ausente; Xaa3 es Asp, Asp Gama-carboxilado, Glu, Glu Gama-carboxilado, Asu, Aad, Apm, o se halla ausente; Xaa4 es Cys o D-Cys; Xaa6 es P-Ser, P-Thr, P-homo-Ser, fosfato de 4-hidroxivalina, P-homo-Thr, P-Cys o P-Tyr; Xaa7 es Tyr, Leu, Phe o Ile; Xaa8 es Cys o D-Cys; Xaa14 es Thr, Ala o Phe; Xaa16 es Cys o D-Cys; y Xaa17 es Tyr, D-Tyr, o se halla ausente; en donde: si Xaa1 se halla presente, Xaa1 puede ser modificado sobre su grupo amino por metilo, ácido etanodioico, ácido propanodioico, ácido butanodioico, ácido pentanodioico, ácido hexanodioico, ácido heptanodioico o ácido octanodioico; si Xaa1 se hallaba ausente y Xaa2 se halla presente, entonces Xaa2 puede ser modificado sobre su grupo amino por metilo, ácido etanodioico, ácido propanodioico, ácido butanodioico, ácido pentanodioico, ácido hexanodioico, ácido heptanodioico o ácido octanodioico; o si tanto Xaa1 como Xaa2 están ausentes, entonces Xaa3 puede ser modificado sobre su grupo amino por metilo, ácido etanodioico, ácido propanodioico, ácido butanodioico, ácido pentanodioico, ácido hexanodioico, ácido heptanodioico o ácido octanodioico.
ARP100104153A 2009-11-09 2010-11-09 Peptido agonista de la guanilato ciclasa c (gc-c) util para tratamientos de trastornos gastrointestinales AR078950A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US25926409P 2009-11-09 2009-11-09

Publications (1)

Publication Number Publication Date
AR078950A1 true AR078950A1 (es) 2011-12-14

Family

ID=43503086

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP100104153A AR078950A1 (es) 2009-11-09 2010-11-09 Peptido agonista de la guanilato ciclasa c (gc-c) util para tratamientos de trastornos gastrointestinales

Country Status (26)

Country Link
US (3) US8507447B2 (es)
EP (1) EP2499154B1 (es)
JP (1) JP5913115B2 (es)
KR (1) KR20120115495A (es)
CN (1) CN102812038B (es)
AR (1) AR078950A1 (es)
AU (1) AU2010314866B2 (es)
BR (1) BR112012011730A2 (es)
CA (1) CA2779482A1 (es)
CL (1) CL2012001186A1 (es)
CO (1) CO6551683A2 (es)
CR (1) CR20120303A (es)
EA (1) EA022817B1 (es)
EC (1) ECSP12011962A (es)
ES (1) ES2620153T3 (es)
GE (1) GEP20166435B (es)
IL (1) IL219596A0 (es)
MX (2) MX350046B (es)
NZ (1) NZ599751A (es)
PH (1) PH12012500916B1 (es)
SG (1) SG10201407403UA (es)
TW (1) TWI482626B (es)
UA (1) UA114274C2 (es)
UY (2) UY33018A (es)
WO (1) WO2011057272A1 (es)
ZA (1) ZA201203342B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2170930B3 (en) 2007-06-04 2013-10-02 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
JP2011522828A (ja) 2008-06-04 2011-08-04 シナジー ファーマシューティカルズ インコーポレイテッド 胃腸障害、炎症、癌、およびその他の障害の治療のために有用なグアニル酸シクラーゼのアゴニスト
EP2321341B1 (en) 2008-07-16 2017-02-22 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders
WO2010065524A2 (en) * 2008-12-02 2010-06-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of fluid retention disorders
AU2010314866B2 (en) * 2009-11-09 2014-10-30 Ironwood Pharmaceuticals, Inc. Treatments for gastrointestinal disorders
US8735360B2 (en) * 2009-12-07 2014-05-27 Ironwood Pharmaceuticals, Inc. Treatments for gastrointestinal disorders
CA2835624A1 (en) 2011-05-11 2012-11-15 Ironwood Pharmaceuticals, Inc. Treatments for gastrointestinal disorders
WO2012155114A1 (en) 2011-05-11 2012-11-15 Ironwood Pharmaceuticals, Inc. Peptides derived from uroguanylin and their use in gastrointestinal disorders
WO2012155108A1 (en) * 2011-05-11 2012-11-15 Ironwood Pharmaceuticals, Inc. Treatments for disorders using guanylate cyclase c agonists
US9617305B2 (en) 2011-06-08 2017-04-11 Ironwood Pharmaceuticals, Inc. Treatments for gastrointestinal disorders
US9527887B2 (en) 2011-06-08 2016-12-27 Ironwood Pharmaceutical, Inc. Treatments for gastrointestinal disorders
DK2776055T3 (en) * 2011-08-17 2017-03-06 Ironwood Pharmaceuticals Inc TREATMENTS FOR GASTROINTESTINAL DISORDERS
WO2014088623A1 (en) * 2012-07-12 2014-06-12 Forest Laboratories Holdings Limited Linaclotide compositions
US9708367B2 (en) 2013-03-15 2017-07-18 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase and their uses
CN114404588A (zh) 2013-08-09 2022-04-29 阿德利克斯公司 用于抑制磷酸盐转运的化合物和方法
AU2014331812B2 (en) * 2013-10-09 2019-01-17 Bausch Health Ireland Limited Agonists of guanylate cyclase useful for downregulation of pro-inflammatory cytokines
WO2016015055A1 (en) * 2014-07-25 2016-01-28 Ironwood Pharmaceuticals, Inc. Colon cleansing compositions
WO2020237096A1 (en) 2019-05-21 2020-11-26 Ardelyx, Inc. Combination for lowering serum phosphate in a patient

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB290795A (en) 1927-04-08 1928-05-24 British Colour Printing Compan Improvements in or relating to advertising or display devices
ES2216004T3 (es) * 1993-10-26 2004-10-16 Thomas Jefferson University Composiciones que se unen especificamente a celulas cancerosas colorectales y procedimientos de uso de las mismas.
US5962220A (en) * 1993-10-26 1999-10-05 Thomas Jefferson University Compositions that specifically bind to colorectal cells and methods of using the same
US5601990A (en) * 1994-09-13 1997-02-11 Thomas Jefferson University Methods of diagnosing colorectal tumors and metastasis thereof
US5518888A (en) * 1993-10-26 1996-05-21 Thomas Jefferson University ST receptor binding compounds and methods of using the same
US5879656A (en) * 1993-10-26 1999-03-09 Thomas Jefferson University Methods of treating metastatic colorectal cancer with ST receptor binding compounds
CH689139A5 (de) 1995-04-03 1998-10-30 Cerbios Pharma Sa Verfahren zur Herstellung einer liposomalen, in Wasser dispergierbaren, oral zu verabreichenden, festen, trockenen therapeutischen Formulierung.
US5912014A (en) 1996-03-15 1999-06-15 Unigene Laboratories, Inc. Oral salmon calcitonin pharmaceutical products
AU2001256315A1 (en) * 2000-04-22 2001-11-07 Ipf Pharmaceuticals Gmbh Use of guanylate cyclase-c (gc-c) agonists as insulinotropic factors for treating diabetes type 2
US7371727B2 (en) * 2003-01-28 2008-05-13 Microbia, Inc. Methods and compositions for the treatment of gastrointestinal disorders
WO2004069165A2 (en) * 2003-01-28 2004-08-19 Microbia, Inc. Methods and compositions for the treatment of gastrointestinal disorders
US7304036B2 (en) * 2003-01-28 2007-12-04 Microbia, Inc. Methods and compositions for the treatment of gastrointestinal disorders
US7772188B2 (en) * 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
US20090253634A1 (en) * 2005-08-19 2009-10-08 Microbia, Inc. Methods and Compositions for the Treatment of Gastrointestinal Disorders
EP2170930B3 (en) * 2007-06-04 2013-10-02 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
PT2328601T (pt) * 2008-08-15 2020-04-30 Ironwood Pharmaceuticals Inc Formulação sólida estável de um polipéptido agonista do recetor gc-c adequado para administração oral
WO2010027405A2 (en) * 2008-09-04 2010-03-11 Ironwood Pharmaceuticals, Inc. Stable solid formulations of gc-c receptor agonist polypeptides suitable for oral administration
AU2010314866B2 (en) * 2009-11-09 2014-10-30 Ironwood Pharmaceuticals, Inc. Treatments for gastrointestinal disorders
WO2011156453A2 (en) 2010-06-09 2011-12-15 Combimab, Inc. Therapeutic peptides

Also Published As

Publication number Publication date
NZ599751A (en) 2014-08-29
JP5913115B2 (ja) 2016-05-11
BR112012011730A2 (pt) 2016-03-08
US20140179607A9 (en) 2014-06-26
EP2499154A1 (en) 2012-09-19
MX350046B (es) 2017-08-24
IL219596A0 (en) 2012-06-28
ZA201203342B (en) 2013-01-30
CL2012001186A1 (es) 2013-07-12
US20140024593A1 (en) 2014-01-23
UY33018A (es) 2011-01-31
AU2010314866A1 (en) 2012-05-31
US20130085107A1 (en) 2013-04-04
MX2012005368A (es) 2012-06-13
US20110118184A1 (en) 2011-05-19
US8507447B2 (en) 2013-08-13
ES2620153T3 (es) 2017-06-27
TWI482626B (zh) 2015-05-01
PH12012500916B1 (en) 2018-03-23
EA201290322A1 (ru) 2013-01-30
CR20120303A (es) 2012-08-08
UY33017A (es) 2011-06-30
TW201116291A (en) 2011-05-16
EA022817B1 (ru) 2016-03-31
AU2010314866B2 (en) 2014-10-30
JP2013510182A (ja) 2013-03-21
GEP20166435B (en) 2016-02-25
EP2499154B1 (en) 2016-12-21
SG10201407403UA (en) 2014-12-30
PH12012500916A1 (en) 2018-01-29
WO2011057272A1 (en) 2011-05-12
UA114274C2 (uk) 2017-05-25
KR20120115495A (ko) 2012-10-18
US8946158B2 (en) 2015-02-03
CO6551683A2 (es) 2012-10-31
CA2779482A1 (en) 2011-05-12
ECSP12011962A (es) 2012-07-31
CN102812038A (zh) 2012-12-05
CN102812038B (zh) 2016-05-18

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