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AR065096A1 - Preparacion solida - Google Patents

Preparacion solida

Info

Publication number
AR065096A1
AR065096A1 ARP080100380A ARP080100380A AR065096A1 AR 065096 A1 AR065096 A1 AR 065096A1 AR P080100380 A ARP080100380 A AR P080100380A AR P080100380 A ARP080100380 A AR P080100380A AR 065096 A1 AR065096 A1 AR 065096A1
Authority
AR
Argentina
Prior art keywords
tablet
compression
solid preparation
pharmaceutical use
cellulose
Prior art date
Application number
ARP080100380A
Other languages
English (en)
Inventor
Shigeyuki Marunaka
Makoto Fukuta
Akihiko Ono
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39156227&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR065096(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of AR065096A1 publication Critical patent/AR065096A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Comprimido que no origina un problema en la compresion, el cual es superior en la formacion del comprimido, la propiedad de disolucion del principio activo para uso farmacéutico y similares. Reivindicacion 1: Un comprimido caracterizado porque contiene los siguiente (A) y (B): (A) un gránulo que comprende un principio activo para uso farmacéutico que induce fácilmente a un problema en la compresion y celulosa macrocristalina; (B) un auxiliar de compresion que contiene estearato de magnesio y celulosa microcristalina.
ARP080100380A 2007-02-01 2008-01-30 Preparacion solida AR065096A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2007023584 2007-02-01

Publications (1)

Publication Number Publication Date
AR065096A1 true AR065096A1 (es) 2009-05-13

Family

ID=39156227

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080100380A AR065096A1 (es) 2007-02-01 2008-01-30 Preparacion solida

Country Status (11)

Country Link
US (1) US8697125B2 (es)
EP (1) EP2124901B1 (es)
JP (1) JP5284967B2 (es)
AR (1) AR065096A1 (es)
CA (1) CA2677193C (es)
CL (1) CL2008000280A1 (es)
ES (1) ES2639854T3 (es)
HR (1) HRP20171518T1 (es)
PE (1) PE20081734A1 (es)
TW (1) TW200836774A (es)
WO (1) WO2008093878A1 (es)

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CN102256976A (zh) 2008-12-23 2011-11-23 贝林格尔.英格海姆国际有限公司 有机化合物的盐形式
TW201036975A (en) 2009-01-07 2010-10-16 Boehringer Ingelheim Int Treatment for diabetes in patients with inadequate glycemic control despite metformin therapy
CN102387795A (zh) * 2009-02-13 2012-03-21 贝林格尔.英格海姆国际有限公司 包含dpp-4抑制剂(利拉列汀)任选地组合其它抗糖尿病药的抗糖尿病药物
JP5685550B2 (ja) 2009-02-13 2015-03-18 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｓｇｌｔ２阻害剤、ｄｐｐ−ｉｖ阻害剤、更に必要により抗糖尿病薬を含む医薬組成物及びその使用
KR20190128004A (ko) 2009-04-06 2019-11-13 와이어쓰 엘엘씨 네라티닙을 이용한 유방암의 치료법
JP5732394B2 (ja) * 2009-07-28 2015-06-10 武田薬品工業株式会社 錠剤
EP3566697B1 (en) * 2009-11-09 2024-09-11 Wyeth LLC Tablet formulations of neratinib maleate
CN107115530A (zh) 2009-11-27 2017-09-01 勃林格殷格翰国际有限公司 基因型糖尿病患者利用dpp‑iv抑制剂例如利拉利汀的治疗
JP5775463B2 (ja) * 2009-12-18 2015-09-09 田辺三菱製薬株式会社 溶出安定性製剤
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AR083878A1 (es) 2010-11-15 2013-03-27 Boehringer Ingelheim Int Terapia antidiabetica vasoprotectora y cardioprotectora, linagliptina, metodo de tratamiento
UY33937A (es) 2011-03-07 2012-09-28 Boehringer Ingelheim Int Composiciones farmacéuticas que contienen inhibidores de dpp-4 y/o sglt-2 y metformina
JP5874545B2 (ja) * 2011-06-20 2016-03-02 アステラス製薬株式会社 経口投与用医薬組成物
HUE061596T2 (hu) 2011-07-15 2023-07-28 Boehringer Ingelheim Int Szubsztituált dimer kinazolin származék, annak elõállítása és alkalmazása az I. és II. típusú cukorbetegség kezelésére szolgáló gyógyszerkészítményekben
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EP3685839A1 (en) 2012-05-14 2020-07-29 Boehringer Ingelheim International GmbH Linagliptin for use in the treatment of albuminuria and kidney related diseases
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WO2013174767A1 (en) 2012-05-24 2013-11-28 Boehringer Ingelheim International Gmbh A xanthine derivative as dpp -4 inhibitor for use in modifying food intake and regulating food preference
JP6309895B2 (ja) * 2012-09-27 2018-04-11 株式会社三和化学研究所 アナグリプチン含有製剤
CN103877054B (zh) * 2012-12-21 2016-05-25 北大方正集团有限公司 一种苯甲酸阿格列汀片剂及其制备方法
CN103610661B (zh) * 2013-11-22 2017-09-12 威海迪素制药有限公司 一种组合物
CN104721188A (zh) * 2013-12-20 2015-06-24 中美华世通生物医药科技（武汉）有限公司 一种稳定的含苯甲酸阿格列汀的组合物
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Also Published As

Publication number Publication date
EP2124901B1 (en) 2017-07-19
ES2639854T3 (es) 2017-10-30
WO2008093878A1 (en) 2008-08-07
JP2010517936A (ja) 2010-05-27
JP5284967B2 (ja) 2013-09-11
CA2677193A1 (en) 2008-08-07
CA2677193C (en) 2015-06-30
TW200836774A (en) 2008-09-16
US20090318482A1 (en) 2009-12-24
PE20081734A1 (es) 2009-01-19
HRP20171518T1 (hr) 2017-11-17
EP2124901A1 (en) 2009-12-02
US8697125B2 (en) 2014-04-15
CL2008000280A1 (es) 2008-08-18

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