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AR064832A1 - Utilizacion de ivabradina para la obtencion de medicamentos destinados al tratamiento de la disfuncion endotelial - Google Patents

Utilizacion de ivabradina para la obtencion de medicamentos destinados al tratamiento de la disfuncion endotelial

Info

Publication number
AR064832A1
AR064832A1 ARP080100090A ARP080100090A AR064832A1 AR 064832 A1 AR064832 A1 AR 064832A1 AR P080100090 A ARP080100090 A AR P080100090A AR P080100090 A ARP080100090 A AR P080100090A AR 064832 A1 AR064832 A1 AR 064832A1
Authority
AR
Argentina
Prior art keywords
ivabradine
treatment
dysfunction
endotelial
medicines
Prior art date
Application number
ARP080100090A
Other languages
English (en)
Inventor
Vidal Benatar
Guy Lerebours-Pigeonniere
Jean-Claude Tardif
Eric Thorin
Eric Rheaume
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of AR064832A1 publication Critical patent/AR064832A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Utilizacion de ivabradina o 3-{3-[{[(7S)-3,4-dimetoxibiciclo[4.2.0]octa-1,3,5-trien-7-il]-metil}-(metil)-amino]-propil} -7,8-dimetoxi-1,3,4,5-tetrahidro-2H-3-benzazepin-2-ona, de sus sales de adicion a un ácido aceptable farmacéuticamente y de sus hidratos, para la obtencion de un medicamento destinado al tratamiento de la disfuncion endotelial, y sus composiciones farmacéuticas.
ARP080100090A 2007-01-11 2008-01-10 Utilizacion de ivabradina para la obtencion de medicamentos destinados al tratamiento de la disfuncion endotelial AR064832A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0700189A FR2911279B1 (fr) 2007-01-11 2007-01-11 Utilisation de l'ivabradine pour l'obtention de medicaments destines au traitement de la dysfonction endotheliale

Publications (1)

Publication Number Publication Date
AR064832A1 true AR064832A1 (es) 2009-04-29

Family

ID=38123876

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080100090A AR064832A1 (es) 2007-01-11 2008-01-10 Utilizacion de ivabradina para la obtencion de medicamentos destinados al tratamiento de la disfuncion endotelial

Country Status (20)

Country Link
US (2) US20080200450A1 (es)
EP (1) EP1944031A1 (es)
JP (1) JP2008169213A (es)
KR (2) KR20080066613A (es)
CN (1) CN101480398B (es)
AR (1) AR064832A1 (es)
AU (1) AU2008200123B2 (es)
BR (1) BRPI0800001A2 (es)
CA (1) CA2617363C (es)
EA (1) EA015398B1 (es)
FR (1) FR2911279B1 (es)
GE (1) GEP20115158B (es)
MA (1) MA29720B1 (es)
MX (1) MX2008000023A (es)
MY (1) MY148650A (es)
NZ (1) NZ564997A (es)
SG (1) SG144832A1 (es)
UA (1) UA96574C2 (es)
WO (1) WO2008099091A2 (es)
ZA (1) ZA200800358B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2938194B1 (fr) * 2008-11-07 2012-08-31 Servier Lab Utilisation de l'ivabradine comme agent de diagnostic dans la methode d'angiographie coronaire par tomodensitometrie multicoupe
FR2961105B1 (fr) * 2010-06-15 2013-02-08 Servier Lab Utilisation de l'association d'un inhibiteur du courant if sinusal et d'un inhibiteur de l'enzyme de conversion de l'angiotensine pour le traitement de l'insuffisance cardiaque
CN102908327B (zh) * 2011-08-05 2015-03-11 江苏恒瑞医药股份有限公司 伊伐布雷定或其可药用盐的缓释制剂
GB201312386D0 (en) * 2013-07-10 2013-08-21 Isis Innovation Pharmaceutical compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2681862B1 (fr) 1991-09-27 1993-11-12 Adir Cie Nouvelles (benzocycloalkyl)alkylamines, leur procede de preparation, et les compositions pharmaceutiques qui les contiennent.
BR0109966A (pt) * 2000-04-12 2003-08-05 Novartis Ag Combinação de compostos orgânicos
FR2834896B1 (fr) * 2002-01-23 2004-02-27 Servier Lab Composition pharmaceutique orodispersible d'ivabradine
FR2882553B1 (fr) * 2005-02-28 2007-05-04 Servier Lab Forme cristalline beta du chlorhydrate de l'ivabradine, son procede de preparation, et les compositions pharmaceutiques qui la contiennent

Also Published As

Publication number Publication date
AU2008200123A1 (en) 2008-07-31
CN101480398B (zh) 2011-07-27
MY148650A (en) 2013-05-15
NZ564997A (en) 2009-09-25
KR20100112540A (ko) 2010-10-19
ZA200800358B (en) 2008-11-26
EA200800022A2 (ru) 2008-08-29
FR2911279A1 (fr) 2008-07-18
EA015398B1 (ru) 2011-08-30
MX2008000023A (es) 2009-02-23
CA2617363C (fr) 2012-12-04
AU2008200123B2 (en) 2012-08-16
CN101480398A (zh) 2009-07-15
WO2008099091A2 (fr) 2008-08-21
GEP20115158B (en) 2011-02-10
US20110288072A1 (en) 2011-11-24
EP1944031A1 (fr) 2008-07-16
US20080200450A1 (en) 2008-08-21
HK1130686A1 (en) 2010-01-08
MA29720B1 (fr) 2008-09-01
KR20080066613A (ko) 2008-07-16
KR101359936B1 (ko) 2014-02-10
WO2008099091A3 (fr) 2008-10-02
SG144832A1 (en) 2008-08-28
JP2008169213A (ja) 2008-07-24
FR2911279B1 (fr) 2009-03-06
EA200800022A3 (ru) 2008-12-30
CA2617363A1 (fr) 2008-07-11
UA96574C2 (ru) 2011-11-25
BRPI0800001A2 (pt) 2010-02-23

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