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AR059126A1 - Uso de sales de tiotropio en el tratamiento del asma persistente moderada - Google Patents

Uso de sales de tiotropio en el tratamiento del asma persistente moderada

Info

Publication number
AR059126A1
AR059126A1 ARP070100019A ARP070100019A AR059126A1 AR 059126 A1 AR059126 A1 AR 059126A1 AR P070100019 A ARP070100019 A AR P070100019A AR P070100019 A ARP070100019 A AR P070100019A AR 059126 A1 AR059126 A1 AR 059126A1
Authority
AR
Argentina
Prior art keywords
treatment
salts
tiotrope
moderate asthma
persistent moderate
Prior art date
Application number
ARP070100019A
Other languages
English (en)
Inventor
Michael Engel
Stefan Heinrichs
Original Assignee
Boehringer Ingelheim Vetmed
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35695896&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR059126(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Vetmed filed Critical Boehringer Ingelheim Vetmed
Publication of AR059126A1 publication Critical patent/AR059126A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Uso de sales de tiotropio para la preparacion de un medicamento destinado al tratamiento de pacientes que padecen asma persistente moderada. Reivindicacion 1: Uso de sales de tiotropio (1) en la que X- indica un anion con una sola carga negativa, preferiblemente un anion que se selecciona entre cloruro, bromuro, yoduro, sulfato, fosfato, metansulfonato, nitrato, maleato, acetato, citrato, fumarato, tartrato, oxalato, succinato, benzoato y p-toluensulfonato, opcionalmente en forma de los hidratos y/o solvatos de los mismos, para la preparacion de un medicamento destinado al tratamiento del asma persistente moderada
ARP070100019A 2006-01-04 2007-01-03 Uso de sales de tiotropio en el tratamiento del asma persistente moderada AR059126A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06100055 2006-01-04

Publications (1)

Publication Number Publication Date
AR059126A1 true AR059126A1 (es) 2008-03-12

Family

ID=35695896

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070100019A AR059126A1 (es) 2006-01-04 2007-01-03 Uso de sales de tiotropio en el tratamiento del asma persistente moderada

Country Status (30)

Country Link
US (2) US20070155773A1 (es)
EP (1) EP1971332B1 (es)
JP (1) JP2009525950A (es)
KR (1) KR20080083060A (es)
CN (1) CN101355937A (es)
AR (1) AR059126A1 (es)
AT (1) ATE500825T1 (es)
AU (1) AU2006334367B2 (es)
BR (1) BRPI0620886A2 (es)
CA (1) CA2634984C (es)
CY (1) CY1111534T1 (es)
DE (1) DE602006020620D1 (es)
DK (1) DK1971332T3 (es)
EA (1) EA015353B1 (es)
EC (1) ECSP088588A (es)
ES (1) ES2362306T3 (es)
HR (1) HRP20110200T1 (es)
IL (1) IL192602A (es)
ME (1) ME01205B (es)
MY (1) MY146362A (es)
NO (1) NO20082439L (es)
NZ (1) NZ570162A (es)
PL (1) PL1971332T3 (es)
PT (1) PT1971332E (es)
RS (1) RS51703B (es)
SI (1) SI1971332T1 (es)
TW (1) TW200731976A (es)
UA (1) UA95271C2 (es)
WO (1) WO2007077162A1 (es)
ZA (1) ZA200804436B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2617717C (en) 2005-08-06 2014-02-11 Boehringer Ingelheim International Gmbh Use of tiotropium salts in the treatment of severe persistant asthma
WO2015065222A1 (ru) * 2013-10-28 2015-05-07 Шолекс Девелопмент Гмбх Фармацевтический ингаляционный препарат для лечения бронхиальной астмы и хронической обструктивной болезни легких, содержащий в качестве активного вещества микронизированный тиотропия бромид, и способ его получения
GB201321717D0 (en) 2013-12-09 2014-01-22 Pharmachemie Bv Inhalable Medicaments
CN110876720A (zh) * 2018-09-06 2020-03-13 天津金耀集团有限公司 依地酸盐恰当改变噻托溴铵喷雾剂表面张力的应用
CN110876721A (zh) * 2018-09-06 2020-03-13 天津金耀集团有限公司 一种含有表面活性剂的噻托溴铵喷雾剂

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2425539A (en) * 1942-10-31 1947-08-12 Aro Equipment Corp Coupling
US5610163A (en) * 1989-09-16 1997-03-11 Boehringer Ingelheim Gmbh Esters of thienyl carboxylic acids and amino alcohols and their quaternization products
DE3931041C2 (de) * 1989-09-16 2000-04-06 Boehringer Ingelheim Kg Ester von Thienylcarbonsäuren mit Aminoalkoholen, ihre Quaternierungsprodukte, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
US6156503A (en) * 1997-03-03 2000-12-05 The Regents Of The University Of California Diagnosing asthma patients predisposed to adverse β-agonist reactions
GB9902689D0 (en) * 1999-02-08 1999-03-31 Novartis Ag Organic compounds
GB0009583D0 (en) * 2000-04-18 2000-06-07 Glaxo Group Ltd Respiratory formulations
EP1326862B1 (de) * 2000-10-12 2004-09-15 BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG Kristallines monohydrat von tiotropiumbromid, verfahren zu dessen herstellung und dessen verwendung zur herstellung eines arzneimittels
US6908928B2 (en) * 2000-10-12 2005-06-21 Bi Pharma Kg. Crystalline tiotropium bromide monohydrate, processes for the preparation thereof, and pharmaceutical compositions
US6608055B2 (en) * 2001-06-22 2003-08-19 Boehringer Ingelheim Pharma Kg Crystalline anticholinergic, processes for preparing it and its use for preparing a pharmaceutical composition
US6919325B2 (en) * 2001-09-14 2005-07-19 Boehringer Ingelheim Pharma Kg Pharmaceutical compositions containing tiotropium salts and low-solubility salmeterol salts
US7951557B2 (en) * 2003-04-27 2011-05-31 Protalix Ltd. Human lysosomal proteins from plant cell culture
US7968717B2 (en) * 2003-11-03 2011-06-28 Boehringer Ingelhein International Gmbh Crystalline anhydrate with anticholinergic efficacy
US8686148B2 (en) * 2003-11-03 2014-04-01 Boehringer Ingelheim International Gmbh Process for preparing new tiotropium salts, new tiotropium salts as such and pharmaceutical compositions thereof
JP4553902B2 (ja) * 2003-11-03 2010-09-29 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 抗コリン作用を有する新規結晶性無水物
SE0303570L (sv) * 2003-12-03 2005-06-04 Microdrug Ag Fukt-känslig medicinsk produkt
SE0303571D0 (sv) * 2003-12-03 2003-12-22 Microdrug Ag Medical product for moisture-sensitive medicaments
US20060269946A1 (en) * 2005-05-10 2006-11-30 Young Robert P Methods and compositions for assessment of pulmonary function and disorders
US7933722B2 (en) * 2005-05-20 2011-04-26 Synergenz Bioscience Limited Methods of analysis of polymorphisms and uses thereof
CA2617717C (en) * 2005-08-06 2014-02-11 Boehringer Ingelheim International Gmbh Use of tiotropium salts in the treatment of severe persistant asthma
US20070167480A1 (en) * 2005-12-19 2007-07-19 Sicor Inc. Pure and stable tiotropium bromide

Also Published As

Publication number Publication date
MY146362A (en) 2012-08-15
ATE500825T1 (de) 2011-03-15
SI1971332T1 (sl) 2011-05-31
AU2006334367A1 (en) 2007-07-12
DE602006020620D1 (de) 2011-04-21
KR20080083060A (ko) 2008-09-12
US20070155773A1 (en) 2007-07-05
ECSP088588A (es) 2008-07-30
US20150224090A1 (en) 2015-08-13
EA015353B1 (ru) 2011-06-30
ZA200804436B (en) 2008-12-31
NO20082439L (no) 2008-08-04
DK1971332T3 (da) 2011-04-18
EP1971332A1 (en) 2008-09-24
PL1971332T3 (pl) 2011-08-31
ES2362306T3 (es) 2011-07-01
AU2006334367B2 (en) 2012-11-08
HRP20110200T1 (hr) 2011-04-30
EP1971332B1 (en) 2011-03-09
NZ570162A (en) 2011-09-30
ME01205B (me) 2013-03-20
CA2634984A1 (en) 2007-07-12
EA200801629A1 (ru) 2008-12-30
IL192602A0 (en) 2009-09-22
TW200731976A (en) 2007-09-01
UA95271C2 (ru) 2011-07-25
PT1971332E (pt) 2011-03-18
IL192602A (en) 2013-06-27
CN101355937A (zh) 2009-01-28
RS51703B (sr) 2011-10-31
CA2634984C (en) 2014-05-06
WO2007077162A1 (en) 2007-07-12
CY1111534T1 (el) 2015-08-05
BRPI0620886A2 (pt) 2011-11-29
JP2009525950A (ja) 2009-07-16

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