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AR058078A1 - Maleato de tegaserod y procesos de obtencion - Google Patents

Maleato de tegaserod y procesos de obtencion

Info

Publication number
AR058078A1
AR058078A1 ARP060104386A ARP060104386A AR058078A1 AR 058078 A1 AR058078 A1 AR 058078A1 AR P060104386 A ARP060104386 A AR P060104386A AR P060104386 A ARP060104386 A AR P060104386A AR 058078 A1 AR058078 A1 AR 058078A1
Authority
AR
Argentina
Prior art keywords
iodhydrate
tegaserod
pentylcarbazimidamide
ylmethylene
indole
Prior art date
Application number
ARP060104386A
Other languages
English (en)
Inventor
Montero Ma Carmen Burgarolas
Original Assignee
Medichem Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Medichem Sa filed Critical Medichem Sa
Publication of AR058078A1 publication Critical patent/AR058078A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)

Abstract

La presente provee un proceso para preparar maleato ácido de 3-(5-metoxi-1H-indol-3- ilmetilen)-N-pentilcarbazimidamida (es decir, maleato de tegaserod). Este proceso incluye hacer reaccionar 5-metoxiindol-3-carbaldehído con iodhidrato de N-pentil- N'-aminoguanidina y aislar el iodhidrato de 3-(5-metoxi-1H-indol-3-ilmetilen)-N-pentilcarbazimidamida (es decir, iodhidrato de tegaserod) solido. Reivindicacion 1: Un compuesto, caracterizado porque es iodhidrato de 3-(5-metoxi-1H-indol-3- ilmetilen)-N-pentilcarbazimidamida (iodhidrato de tegaserod).
ARP060104386A 2005-10-06 2006-10-05 Maleato de tegaserod y procesos de obtencion AR058078A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US72396205P 2005-10-06 2005-10-06
US72528205P 2005-10-12 2005-10-12
US80896006P 2006-05-30 2006-05-30

Publications (1)

Publication Number Publication Date
AR058078A1 true AR058078A1 (es) 2008-01-23

Family

ID=38514208

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060104386A AR058078A1 (es) 2005-10-06 2006-10-05 Maleato de tegaserod y procesos de obtencion

Country Status (2)

Country Link
AR (1) AR058078A1 (es)
WO (1) WO2007119109A2 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010015794A1 (en) * 2008-08-07 2010-02-11 Generics [Uk] Limited Novel polymorphic forms of tegaserod

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY137386A (en) * 2003-07-24 2009-01-30 Novartis Ag Stable modifications of tegaserod hydrogen maleate
WO2006116953A1 (en) * 2005-05-02 2006-11-09 Zentiva, A.S. A method for the preparation of tegaserod and slected salts thereof

Also Published As

Publication number Publication date
WO2007119109A3 (en) 2008-06-12
WO2007119109A2 (en) 2007-10-25

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Legal Events

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