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AR057331A1 - Serin- amidas sustituidas con heteroaroilo - Google Patents

Serin- amidas sustituidas con heteroaroilo

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Publication number
AR057331A1
AR057331A1 ARP060102179A ARP060102179A AR057331A1 AR 057331 A1 AR057331 A1 AR 057331A1 AR P060102179 A ARP060102179 A AR P060102179A AR P060102179 A ARP060102179 A AR P060102179A AR 057331 A1 AR057331 A1 AR 057331A1
Authority
AR
Argentina
Prior art keywords
alkyl
alkoxy
amino
phenyl
aminocarbonyl
Prior art date
Application number
ARP060102179A
Other languages
English (en)
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of AR057331A1 publication Critical patent/AR057331A1/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Furan Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

Procedimientos y productos intermediarios para su preparacion, así como el uso de esos compuestos o agentes que contienen estos compuestos, para el combate de plantas no deseadas. Reivindicacion 1: Serin-amidas sustituidas con heteroaroílo, caracterizadas porque tienen la formula en donde las variables tienen los siguientes significados: A es heteroarilo de 5 o 6 miembros con uno a cuatro átomos de N, o con uno a tres átomos de N y un átomo de O o S, o con un átomo de O o S, que puede estar parcial o totalmente halogenado y/o que puede llevar 1 a 3 radicales del grupo ciano, alquilo C1-6, cicloalquilo C3-6, halogenoalquilo C1-6, alcoxi C1-6, halogenoalcoxi C1-6 y alcoxi C1-6-alquilo C1-4; R1, R2 es H, hidroxi o alcoxi C1-6; R3 es alquilo C1-6, cianoalquilo C1-4 o halogenoalquilo C1-6; R4 es H, alquilo C1-6, cicloalquilo C3-6, alquenilo C3-6, alquinilo C3-6, halogenalquenilo C3-6, halogenalquinilo C3-6, formilo, alquil C1-6-carbonilo, cicloalquilcarbonilo C3-6, alquenilcarbonilo C2-6, alquinilcarbonilo C2-6, alcoxi C1-6-carbonilo, alqueniloxicarbonilo C3-6, alquinil C3-6-oxicarbonilo, alquil C1-6-aminocarbonilo, alquenilaminocarbonilo C3-6, alquinilaminocarbonilo C3-6, alquil C1-6-sulfonilaminocarbonilo, di(alquil C1-6)-aminocarbonilo, N-(alquenil C3-6)-N-(alquil C1-6)-aminocarbonilo, N-(alquinil C3-6)-N(alquilo C1-6)-aminocarbonilo, N-(alcoxi C1-6)-N-(alquil C1-6)-amino-carbonilo, N-(alquenil C3-6)-N-(alcoxi C1-6)-aminocarbonilo, N-(alquinil C3-6)- N-(alcoxi C1-6)-aminocarbonilo, di-(alquil C1-6)-aminotiocarbonilo, (alquil 1-6)cianoimino, (amino)cianoimino, [(alquil C1-6)amino]cianoimino, [di(alquil C1-6)amino]cianoimino, alquil C1-6-carbonil-alquilo C1-6, alcoxi C1-6-imino-alquilo C1-6, N- (alquil C1-6-amino)-imino-alquilo C1-6, N-(di-alquil C1-6-amino)-imino-alquilo C1-6, o tri-alquil C1-4-sililo, en donde los radicales alquilo, cicloalquilo y alcoxi mencionados pueden estar parcial o totalmente halogenados y/o pueden llevar 1 a 3 de los siguientes grupos: ciano, hidroxi, cicloalquilo C3-6, alcoxi C1-6-alquilo C1-4, alcoxi C1-4-alcoxi C1-4-alquilo C1-4, alcoxi C1-4, alquil C1-4-tio, di(alquil C1-4)-amino, alquilo C1-4-alcoxi C1-6-carbonilamino, alquil C1-4-carbonilo, hidroxicarbonilo, alcoxi C1-4-carbonilo, aminocarbonilo, alquil C1-4-aminocarbonilo, di(alquil C1-4)aminocarbonilo o alquil C1-4-carboniloxi; fenilo, fenil-alquilo C1-6, fenilcarbonilo, fenilcarbonil-alquilo C1-6, fenoxicarbonilo, fenilaminocarbonilo, fenilsulfonilaminocarbonilo, N-(alquilo C1-6)-N-(fenil)-aminocarbonilo, fenil-alquil C1-6-carbonilo, en donde el radical fenilo puede estar parcial o totalmente halogenado y/o puede llevar 1 a 3 de los siguientes grupos: nitro, ciano, alquilo C1-4, halogenalquilo C1-4, alcoxi C1-4 o halogenalcoxi C1-4, o SO2R7; R5 es H o alquilo C1-6; R6 es alquilo C1-6, alquenilo C2-6, alquinilo C2-6, halogenalquilo C1-6, halogenalquenilo C2-6, halogenalquinilo C2-6, cianoalquilo C1-6, cianoalquenilo C2-6, cianoalquinilo C2-6, hidroxialquilo C1-6, hidroxialquenilo C2-6, hidroxialquinilo C2-6, cicloalquilo C3-6, cicloalquenilo C3-6, heterociclilo de 3 a 6 miembros, heterociclil-alquilo C1-4 de 3 a 6 miembros, en donde los radicales cicloalquilo, cicloalquenilo o heterociclilo de 3 a 6 miembros antes mencionados peden estar parcial o totalmente halogenados y/o pueden llevar 1 a 3 radicales del grupo oxo, ciano, nitro, alquilo C1-6, halogenalquilo C1-6, hidroxi, alcoxi C1-6, halogenalcoxi C1-6, hidroxicarbonilo, alcoxi C1-6-carbonilo, hidroxicarbonil-alcoxi C1-6, alcoxi C1-6-carbonil-alcoxi C1-6, amino, alquil C1-6-amino, di(alquil C1-6)amino, alquil C1-6-sulfonilamino, halogenalquil C1-6-sulfonilamino, aminocarbonilamino, (alquil C1-6-amino)carbonilamino, di-(alquil C1-6)-aminocarbonilamino, arilo y aril(alquilo C1-6); alcoxi C1-6-alquilo C1-4, alquenil C2-6-oxi-alquilo C1-4, alquinil C2-6-oxi-alquilo C1-4, halogenalcoxi C1-6-alquilo C1-4, halogenalquenil C2-6-oxi-alquilo C1-4, halogenalquinil C2-6-oxi-alquilo C1-4, alcoxi C1-6-alcoxi C1-4-alquilo C1-4, alquil C1-6-tio-alquilo C1-4, alquenil C2-6-tio-alquilo C1-4, alquinil C2-6-tioalquilo C1-4, halogenalquil C1-6-tioalquilo C1-4, halogenalquenil C2-6-tioalquilo C1-4, halogenalquinil C2-6-tioalquilo C1-4, alquil C1-6-sulfinil-alquilo C1-4, halogenalquil C1-6-sulfinil-alquilo C1-4, alquil C1-4-sulfonil-alquilo C1-4, halogenalquil C1-6-sulfonil-alquilo C1-4, amino-alquilo C1-4, alquil C1-6-amino-alquilo C1-4, di-(alquil C1-6)amino-alquilo C1-4, alquil C1-6-sulfonilamino-alquilo C1-4, alquil C1-6-sulfonil-(alquil C1-6)-amino-alquilo C1-4, alquil C1-6-carbonilo, hidroxicarbonilo, alcoxi C1-6-carbonilo, aminocarbonilo, alquil C1-6-aminocarbonilo, di-(alquil C1-6)-aminocarbonilo, alquil C1-6-carbonil-alquilo C1-6, hidroxicarbonil-alquilo C1-4, alcoxi C1-6-carbonil-alquilo C1-4, halogenalcoxi C1-6-carbonil-alquilo C1-4, alquil C1-6-carboniloxi-alquilo C1-4, aminocarbonil- alquilo C1-4, alquil C1-6-aminocarbonil-alquilo C1-4, di(alquil C1-6)aminocarbonil-alquilo C1-4, formilamino-alquilo C1-4, alcoxi C1-6-carbonilamino-alquilo C1-4, alquil C1-6-carbonilamino-alquilo C1-4, alquil C1-6-carbonil-(alquil C1-6-amino)- alquilo C1-4, [(alquil C1-6)aminocarboniloxi]-alquilo C1-4, [di(-alquil C1-6)aminocarboniloxi]-alquilo C1-4, {di-[di-(alquil C1-6)amino]carboniloxi}-alquilo C1-4, [(alquil C1-6-amino)carbonilamino]-alquilo C1-4, [di-(alquil C1-6)aminocarbonilamino]- alquilo C1-4; fenil-alquilo C1-4, fenil-alquenilo C2-4, fenil-alquinilo C2-4, fenil-halogenalquilo C1-4, fenil-halogenalquenilo C2-4, fenil-halogenalquinilo C2-4, fenil-hidroxialquilo C1-4, fenil-hidroxialquenilo C2-4, fenil-hidroxialquinilo C2-4, fenilcarbonil-alquilo C1-4, fenilcarbonilamino-alquilo C1-4, fenilcarboniloxi-alquilo C1-4, fenilcarbonil-alquilo C1-4, feniloxi-alquilo C1-4, feniltio-alquilo C1-4, fenilsulfinil-alquilo C1-4, fenilsulfonil-alquilo C1-4, heteroaril-alquilo C1-4, heteroaril-alquenilo C2-4, heteroaril-alquinilo C2-4, heteroaril-halogenalquilo C1-4, heteroaril-halogenalquenilo C2-4, heteroaril-halogenalquinilo C2-4, heteroaril-hidroxialquilo C1-4, heteroaril-hidroxialquenilo C2-4, heteroaril-hidroxialquinilo C1-4, heteroarilcarbonil-alquilo C1-4, heteroarilcarboniloxi-alquilo C1-4, heteroariloxicarbonil-alquilo C1-4, heteroariloxi-alquilo C1-4, heteroariltio-alquilo C1-4, heteroarilsulfinil-alquilo C1-4, heteroarilsulfonil-alquilo C1-4, en donde los radicales fenilo y heteroarilo antes mencionados pueden estar parcial o totalmente halogenados y/o pueden llevar 1 a 3 radicales del grupo ciano, nitro, alquilo C1-6, halogenalquilo C1-6, hidroxi, alcoxi C1-6, halogenalcoxi C1-6, hidroxicarbonilo, alcoxi C1-6-carbonilo, hidroxicarbonil-alcoxi C1-6, alcoxi C1-6-carbonil-alcoxi C1-6, amino, alquil C1-6-amino, di-(alquil C1-6)amino, alquil C1-6-sulfonilamino, halogenalquil C1-6-sulfonilamino, (alquil C1-6-amino)carbonilamino, di-(alquil C1-6)- aminocarbonilamino, arilo y aril(alquilo C1-6); R7 alquilo C1-6, halogenalquilo C1-6 o fenilo; en donde el radical fenilo puede estar parcial o totalmente halogenado y/o puede llevar 1 a 3 de los siguientes grupos: alquilo C1-6, haloalquilo C1-6, o alcoxi C1-6; así como sus sales de utilidad en agricultura.
ARP060102179A 2005-05-25 2006-05-24 Serin- amidas sustituidas con heteroaroilo AR057331A1 (es)

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DE102005024599 2005-05-25

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US (1) US7879761B2 (es)
EP (1) EP1888532A1 (es)
JP (1) JP4981037B2 (es)
CN (1) CN101228133A (es)
AR (1) AR057331A1 (es)
AU (1) AU2006251302A1 (es)
BR (1) BRPI0611498B1 (es)
CA (1) CA2609243A1 (es)
EA (1) EA013636B1 (es)
IL (1) IL187502A0 (es)
MX (1) MX2007014490A (es)
PE (1) PE20070051A1 (es)
TW (1) TW200716558A (es)
UA (1) UA90720C2 (es)
UY (1) UY29565A1 (es)
WO (1) WO2006125687A1 (es)
ZA (1) ZA200711009B (es)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20060721A1 (es) * 2004-09-16 2006-08-24 Basf Ag Serinamidas sustituidas por heteroaroilo
BRPI0710930A2 (pt) * 2006-05-19 2012-02-14 Basf Se composto processo para preparar um composto, composição, processos para preparar composições e para combater vegetação indesejada, e, uso do composto
CN101578261B (zh) * 2007-01-11 2014-04-16 巴斯夫欧洲公司 杂芳酰基取代的丝氨酰胺
US8097712B2 (en) 2007-11-07 2012-01-17 Beelogics Inc. Compositions for conferring tolerance to viral disease in social insects, and the use thereof
RU2011121521A (ru) * 2008-10-31 2012-12-10 Басф Се Способ улучшения жизнеспособности растения
US8962584B2 (en) 2009-10-14 2015-02-24 Yissum Research Development Company Of The Hebrew University Of Jerusalem, Ltd. Compositions for controlling Varroa mites in bees
MX2012010479A (es) 2010-03-08 2012-10-09 Monsanto Technology Llc Moleculas polinucleotidicas para regulacion genetica en plantas.
CN103975068A (zh) 2011-09-13 2014-08-06 孟山都技术公司 用于杂草控制的方法和组合物
EP3296402B1 (en) 2011-09-13 2020-04-15 Monsanto Technology LLC Methods and compositions for weed control
US10760086B2 (en) 2011-09-13 2020-09-01 Monsanto Technology Llc Methods and compositions for weed control
CN110066794A (zh) 2011-09-13 2019-07-30 孟山都技术公司 用于杂草控制的方法和组合物
CA2848576A1 (en) 2011-09-13 2013-03-21 Monsanto Technology Llc Methods and compositions for weed control comprising topical application of 4-hydroxyphenyl-pyruvate-dioxygenase (hppd)-inhibiting polynucleotides
US10829828B2 (en) 2011-09-13 2020-11-10 Monsanto Technology Llc Methods and compositions for weed control
MX362810B (es) 2011-09-13 2019-02-13 Monsanto Technology Llc Metodos y composiciones para controlar malezas.
UA116092C2 (uk) 2011-09-13 2018-02-12 Монсанто Текнолоджи Ллс Спосіб та композиція для боротьби з бур'янами (варіанти)
US10806146B2 (en) 2011-09-13 2020-10-20 Monsanto Technology Llc Methods and compositions for weed control
MX362812B (es) 2011-09-13 2019-02-13 Monsanto Technology Llc Metodos y composiciones para el control de malezas.
WO2013175480A1 (en) 2012-05-24 2013-11-28 A.B. Seeds Ltd. Compositions and methods for silencing gene expression
US10683505B2 (en) 2013-01-01 2020-06-16 Monsanto Technology Llc Methods of introducing dsRNA to plant seeds for modulating gene expression
MX375327B (es) 2013-01-01 2025-03-06 A B Seeds Ltd Métodos para introducir dsrna en semillas de plantas para modular la expresión genética.
WO2014164797A2 (en) 2013-03-13 2014-10-09 Monsanto Technology Llc Methods and compositions for weed control
CN105074008A (zh) 2013-03-13 2015-11-18 孟山都技术有限公司 用于杂草控制的方法和组合物
US10568328B2 (en) 2013-03-15 2020-02-25 Monsanto Technology Llc Methods and compositions for weed control
US9850496B2 (en) 2013-07-19 2017-12-26 Monsanto Technology Llc Compositions and methods for controlling Leptinotarsa
CA2918387C (en) 2013-07-19 2021-11-02 Monsanto Technology Llc Compositions and methods for controlling leptinotarsa
NZ719544A (en) 2013-11-04 2022-09-30 Beeologics Inc Compositions and methods for controlling arthropod parasite and pest infestations
UA119253C2 (uk) 2013-12-10 2019-05-27 Біолоджикс, Інк. Спосіб боротьби із вірусом у кліща varroa та у бджіл
UA121462C2 (uk) 2014-01-15 2020-06-10 Монсанто Текнолоджі Елелсі Спосіб та композиція для боротьби із бур'янами з використанням полінуклеотидів epsps
EP3420809A1 (en) 2014-04-01 2019-01-02 Monsanto Technology LLC Compositions and methods for controlling insect pests
EP3158067B1 (en) 2014-06-23 2020-08-12 Monsanto Technology LLC Compositions and methods for regulating gene expression via rna interference
EP3161138A4 (en) 2014-06-25 2017-12-06 Monsanto Technology LLC Methods and compositions for delivering nucleic acids to plant cells and regulating gene expression
WO2016018887A1 (en) 2014-07-29 2016-02-04 Monsanto Technology Llc Compositions and methods for controlling insect pests
CN105801485B (zh) * 2014-12-29 2018-04-24 浙江省化工研究院有限公司 一类苯基连吡唑酰胺衍生物、其制备方法及应用
CA2974101A1 (en) 2015-01-22 2016-07-28 Monsanto Technology Llc Compositions and methods for controlling leptinotarsa
WO2016196738A1 (en) 2015-06-02 2016-12-08 Monsanto Technology Llc Compositions and methods for delivery of a polynucleotide into a plant
CN108024517A (zh) 2015-06-03 2018-05-11 孟山都技术公司 用于将核酸引入到植物中的方法和组合物
TN2017000544A1 (en) 2015-07-31 2019-04-12 Pfizer 1,1,1-trifluoro-3-hydroxypropan-2-yl carbamate derivatives and 1,1,1-trifluoro-4-hydroxybutan-2-yl carbamate derivatives as magl inhibitors
RU2720203C1 (ru) 2017-01-20 2020-04-27 Пфайзер Инк. 1,1,1-трифтор-3-гидроксипропан-2-илкарбаматные производные как ингибиторы magl
MX2019008690A (es) 2017-01-23 2019-09-18 Pfizer Compuestos espiro heterociclicos como inhibidores de magl.

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS63301868A (ja) 1987-06-01 1988-12-08 Nippon Kayaku Co Ltd Ｎ−（２−クロロイソニコチノイル）アミノ酸誘導体およびそれを有効成分とする農園芸用殺菌剤
US5346907A (en) * 1988-04-05 1994-09-13 Abbott Laboratories Amino acid analog CCK antagonists
JPH02172956A (ja) 1988-12-23 1990-07-04 Sumitomo Pharmaceut Co Ltd エリスロ―３―（３，４―ジヒドロキシフェニル）セリン誘導体の新規製造法
US4904674A (en) * 1989-08-16 1990-02-27 Hoechst-Roussel Pharmaceuticals Inc. 1-(Benzo[b]thienyl)-2-(thienyl)ethenes and related compounds useful as anti-inflammatory agents
JP2543771B2 (ja) * 1989-12-12 1996-10-16 四国化成工業株式会社 ４（５）―カルバモイル―イミダゾ―ル化合物の合成方法及び新規化合物
DE4011172A1 (de) * 1990-04-06 1991-10-10 Degussa Verbindungen zur bekaempfung von pflanzenkrankheiten
JPH03294253A (ja) 1990-04-12 1991-12-25 Shionogi & Co Ltd 消化管ホルモン拮抗物質
ES2021557A6 (es) 1990-07-23 1991-11-01 Aliana S A Procedimiento de obtencion de 4-hidroxi-metil-n-2-piridinil-2h-tieno (2,3 c)-1,2 tiazina-3 carboxamida 1,1 dioxido.
US5658885A (en) 1993-04-27 1997-08-19 The Dupont Merck Pharmaceutical Company Amidino and guanidino substituted boronic acid inhibitors of trypsin-like enzymes
JPH10101655A (ja) 1996-10-01 1998-04-21 Sumitomo Chem Co Ltd オキサゾリン類、その製造法およびそれを用いるスレオ−３−芳香族セリン類の製造法
JP3294253B2 (ja) 1996-10-11 2002-06-24 新東工業株式会社 鋳物砂の混練供給システム
JP4418043B2 (ja) * 1998-10-07 2010-02-17 大塚化学株式会社 β−ヒドロキシエステルの製造法
HUP0600103A2 (en) 2001-03-02 2006-06-28 Bristol Myers Squibb Co Co-administration of melanocortin receptor agonist and phosphodiesterase inhibitor for treatment of cyclic-amp associated disorders
BR0208956A (pt) 2001-04-16 2004-07-13 Tanabe Seiyaku Co Abridor de canais de k ativados por cálcio de grande condutância
CA2467665A1 (en) * 2001-11-29 2003-06-05 Basf Aktiengesellschaft 2,w-diaminocarboxylic acid compounds
DE10204951A1 (de) 2002-02-06 2003-08-14 Basf Ag Phenylalaninderivate als Herbizide
AR046792A1 (es) 2003-12-19 2005-12-21 Basf Ag Fenilalanina-amidas sustituidas por heteroaroilo, un procedimiento para su preparacion, utilizacion de las mismas como herbicidas y productos fitosa-nitarios que los contienen como principio activo
CN1894202A (zh) 2003-12-19 2007-01-10 巴斯福股份公司 苯甲酰基取代的苯基丙氨酸酰胺
US8202843B2 (en) * 2004-02-27 2012-06-19 Rib-X Pharmaceuticals, Inc. Macrocyclic compounds and methods of making and using the same
PE20060721A1 (es) * 2004-09-16 2006-08-24 Basf Ag Serinamidas sustituidas por heteroaroilo

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CA2609243A1 (en) 2006-11-30
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EA200702443A1 (ru) 2008-06-30
IL187502A0 (en) 2008-03-20
AU2006251302A1 (en) 2006-11-30
US7879761B2 (en) 2011-02-01
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BRPI0611498B1 (pt) 2015-10-13
UA90720C2 (en) 2010-05-25
US20080200338A1 (en) 2008-08-21
BRPI0611498A2 (pt) 2011-02-22
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EA013636B1 (ru) 2010-06-30
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