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AR054790A1 - Metodos para el tratamiento de disfuncion sexual - Google Patents

Metodos para el tratamiento de disfuncion sexual

Info

Publication number
AR054790A1
AR054790A1 ARP060102653A ARP060102653A AR054790A1 AR 054790 A1 AR054790 A1 AR 054790A1 AR P060102653 A ARP060102653 A AR P060102653A AR P060102653 A ARP060102653 A AR P060102653A AR 054790 A1 AR054790 A1 AR 054790A1
Authority
AR
Argentina
Prior art keywords
hydrogen
group
compound
treatment
sexual dysfunction
Prior art date
Application number
ARP060102653A
Other languages
English (en)
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of AR054790A1 publication Critical patent/AR054790A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Reproductive Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Método para el tratamiento de la disfuncion sexual en un sujeto, que comprende la etapa de la administracion de una cantidad terapéuticamente eficaz de un compuesto de la formula (1), o una sal aceptable para uso farmacéutico de dicho compuesto, o su éster; donde: Rx es un miembro seleccionado del grupo que consiste en hidrogeno, alquilo inferior C1-8, halogeno seleccionado de F, Cl, Br e I, alcoxi C1-3, nitro, hidroxi, trifluormetilo y tioalcoxi C1-3; x es un entero de 1 a 3, con la condicion de que R puede ser igual o diferente cuando x es 2 o 3; R1 y R2 pueden ser iguales o diferentes entre sí, y se seleccionan de manera independiente del grupo que consiste en hidrogeno, alquilo inferior C1-8, arilo, arilalquilo, cicloalquilo C3-7; R1 y R2 pueden unirse para formar un heterociclo de 5 a 7 miembros sustituido con un miembro seleccionado del grupo que consiste en hidrogeno, grupos alquilo y arilo; donde el compuesto cíclico puede comprender 1 a 2 átomos de nitrogeno y 0 a 1 átomo de oxígeno; donde los átomos de nitrogeno no están conectados directamente entre sí o con el átomo de oxígeno.
ARP060102653A 2005-06-22 2006-06-21 Metodos para el tratamiento de disfuncion sexual AR054790A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US69280905P 2005-06-22 2005-06-22

Publications (1)

Publication Number Publication Date
AR054790A1 true AR054790A1 (es) 2007-07-18

Family

ID=37067408

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060102653A AR054790A1 (es) 2005-06-22 2006-06-21 Metodos para el tratamiento de disfuncion sexual

Country Status (12)

Country Link
US (1) US8552060B2 (es)
EP (1) EP1893291B1 (es)
JP (1) JP5298334B2 (es)
KR (1) KR101335942B1 (es)
AR (1) AR054790A1 (es)
AT (1) ATE459393T1 (es)
CA (1) CA2612672C (es)
DE (1) DE602006012670D1 (es)
ES (1) ES2344469T3 (es)
MY (1) MY145066A (es)
TW (1) TWI387452B (es)
WO (1) WO2007001841A1 (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI419681B (zh) 2005-06-08 2013-12-21 Sk生物製藥股份有限公司 胺基甲酸酯用於製造供治療白天過度嗜睡(eds)的藥物之用途
JP6095366B2 (ja) 2009-06-22 2017-03-15 エスケー バイオファーマシューティカルズ カンパニー リミテッド 疲労を治療又は予防するための方法
CN102762201B (zh) 2009-11-06 2013-12-18 爱思开生物制药株式会社 注意力缺陷/多动症的治疗方法
EP2496227B1 (en) 2009-11-06 2019-05-22 SK Biopharmaceuticals Co., Ltd. Methods for treating fibromyalgia syndrome
US9610274B2 (en) 2010-06-30 2017-04-04 Sk Biopharmaceuticals Co., Ltd. Methods for treating bipolar disorder
PT2968208T (pt) 2013-03-13 2022-10-28 Aerial Biopharma Llc Tratamento da cataplexia
EP3021838B1 (en) 2013-07-18 2020-05-27 Jazz Pharmaceuticals Ireland Limited Treatment for obesity
TWI655179B (zh) 2014-02-28 2019-04-01 南韓商愛思開生物製藥股份有限公司 胺基羰基胺基甲酸酯化合物
US10888542B2 (en) 2014-02-28 2021-01-12 Sk Biopharmaceuticals Co., Ltd. Aminocarbonylcarbamate compounds
JP6466792B2 (ja) * 2015-07-03 2019-02-06 エスケー バイオファーマスティカルズ カンパニー リミテッド 注意欠陥/多動性障害(adhd)の治療方法
ES2970887T3 (es) 2016-09-06 2024-05-31 Axsome Malta Ltd Forma de solvato de carbamato de (R)-2-amino-3-fenilpropilo
US10195151B2 (en) 2016-09-06 2019-02-05 Jazz Pharmaceuticals International Iii Limited Formulations of (R)-2-amino-3-phenylpropyl carbamate
WO2018067971A1 (en) 2016-10-06 2018-04-12 Jazz Pharmaceuticals International Iii Limited Carbamoyl phenylalaninol compounds and uses therof
EP3630072A4 (en) 2017-06-02 2021-03-10 Jazz Pharmaceuticals Ireland Limited METHODS AND COMPOSITIONS FOR TREATMENT OF EXCESSIVE Drowsiness
RU2020108634A (ru) 2017-07-31 2021-09-02 Джаз Фармасьютикалз Айрлэнд Лимитед Аналоги карбамоилфенилаланинола и способы их применения
US10940133B1 (en) 2020-03-19 2021-03-09 Jazz Pharmaceuticals Ireland Limited Methods of providing solriamfetol therapy to subjects with impaired renal function
AU2024308064A1 (en) 2023-06-29 2026-01-22 Axsome Therapeutics, Inc. Methods of administering solriamfetol to lactating women

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ314570A (en) * 1993-06-10 2000-11-24 Lilly Co Eli Treatment of emesis using tetrahydrobenz[cd]indole-6-carboxamides
KR100197892B1 (ko) * 1994-09-09 1999-06-15 남창우 신규한 페닐알킬아미노 카바메이트 화합물과 그의 제조방법
KR0173862B1 (ko) 1995-02-11 1999-04-01 조규향 O-카바모일-(d)-페닐알라닌올 화합물과 그의 약제학적으로 유용한 염 및 이들의 제조방법
US6228864B1 (en) * 1997-10-28 2001-05-08 Vivus, Inc. Administration of 5-HT receptor agonists and antagonists, to treat premature ejaculation
US20050203130A1 (en) * 2003-12-02 2005-09-15 Erik Buntinx Use of D4 and 5-HT2A antagonists, inverse agonists or partial agonists
CA2587481A1 (en) 2004-10-28 2006-05-11 Sk Corporation Phenylalkylamino carbamates adjunctive therapy for depression
TWI419681B (zh) * 2005-06-08 2013-12-21 Sk生物製藥股份有限公司 胺基甲酸酯用於製造供治療白天過度嗜睡(eds)的藥物之用途

Also Published As

Publication number Publication date
JP2008546778A (ja) 2008-12-25
MY145066A (en) 2011-12-15
US20090221553A1 (en) 2009-09-03
CA2612672A1 (en) 2007-01-04
WO2007001841A1 (en) 2007-01-04
ATE459393T1 (de) 2010-03-15
KR101335942B1 (ko) 2013-12-04
TW200727893A (en) 2007-08-01
CA2612672C (en) 2014-10-14
JP5298334B2 (ja) 2013-09-25
ES2344469T3 (es) 2010-08-27
US8552060B2 (en) 2013-10-08
KR20080028445A (ko) 2008-03-31
TWI387452B (zh) 2013-03-01
EP1893291A1 (en) 2008-03-05
DE602006012670D1 (de) 2010-04-15
EP1893291B1 (en) 2010-03-03

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