AR048958A1 - Medicamento en forma de pelicula para administracion por via oral, que contiene estriol - Google Patents
Medicamento en forma de pelicula para administracion por via oral, que contiene estriolInfo
- Publication number
- AR048958A1 AR048958A1 ARP050101957A ARP050101957A AR048958A1 AR 048958 A1 AR048958 A1 AR 048958A1 AR P050101957 A ARP050101957 A AR P050101957A AR P050101957 A ARP050101957 A AR P050101957A AR 048958 A1 AR048958 A1 AR 048958A1
- Authority
- AR
- Argentina
- Prior art keywords
- film
- medication
- estriol
- administration via
- via oral
- Prior art date
Links
- PROQIPRRNZUXQM-UHFFFAOYSA-N (16alpha,17betaOH)-Estra-1,3,5(10)-triene-3,16,17-triol Natural products OC1=CC=C2C3CCC(C)(C(C(O)C4)O)C4C3CCC2=C1 PROQIPRRNZUXQM-UHFFFAOYSA-N 0.000 title abstract 3
- 229940079593 drug Drugs 0.000 title abstract 3
- 239000003814 drug Substances 0.000 title abstract 3
- PROQIPRRNZUXQM-ZXXIGWHRSA-N estriol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@H]([C@H](O)C4)O)[C@@H]4[C@@H]3CCC2=C1 PROQIPRRNZUXQM-ZXXIGWHRSA-N 0.000 title abstract 3
- 229960001348 estriol Drugs 0.000 title abstract 3
- 238000002483 medication Methods 0.000 abstract 2
- 239000013543 active substance Substances 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Endocrinology (AREA)
- Physiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nutrition Science (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente se refiere a medicamentos en forma de película para administracion por vía oral, en particular por vía bucal, indicados para el tratamiento de los trastornos climatéricos, por cuanto los medicamentos contienen como sustancias activas estriol y/o al menos un éster de estriol farmacologicamente aceptable, solo o combinado al menos con un gestogeno.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004023984A DE102004023984A1 (de) | 2004-05-14 | 2004-05-14 | Filmförmiges, oral zu verabreichendes Arzneimittel, enthaltend Estriol |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR048958A1 true AR048958A1 (es) | 2006-06-14 |
Family
ID=34977101
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP050101957A AR048958A1 (es) | 2004-05-14 | 2005-05-13 | Medicamento en forma de pelicula para administracion por via oral, que contiene estriol |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20070243217A1 (es) |
| EP (1) | EP1761242A2 (es) |
| JP (1) | JP2007537178A (es) |
| KR (1) | KR20070040753A (es) |
| CN (1) | CN1997349A (es) |
| AR (1) | AR048958A1 (es) |
| AU (1) | AU2005244409A1 (es) |
| BR (1) | BRPI0510855A (es) |
| CA (1) | CA2566325A1 (es) |
| DE (1) | DE102004023984A1 (es) |
| IL (1) | IL179014A0 (es) |
| MX (1) | MXPA06012890A (es) |
| NO (1) | NO20065657L (es) |
| RU (1) | RU2006140649A (es) |
| TW (1) | TW200536547A (es) |
| WO (1) | WO2005110358A2 (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2252261A2 (en) * | 2008-02-13 | 2010-11-24 | Bayer Schering Pharma Aktiengesellschaft | Drug delivery system with stabilising effect |
| MX2010008940A (es) * | 2008-02-13 | 2010-10-05 | Bayer Schering Pharma Ag | Sistemas de administracion de drogas que contienen estradiol. |
| US20090269403A1 (en) * | 2008-04-24 | 2009-10-29 | Shaked Ze Ev | Oral contraceptive dosage forms and methods of making such dosage forms |
| WO2010033832A2 (en) * | 2008-09-19 | 2010-03-25 | Evestra, Inc. | Estriol formulations |
| DE102009007771B4 (de) * | 2009-02-05 | 2012-02-16 | Bayer Schering Pharma Aktiengesellschaft | Bukkales Applikationssystem, 17α-Estradiol enthaltend |
| KR102044515B1 (ko) * | 2019-08-20 | 2019-11-14 | 이영환 | 구강점막 부착력이 우수한 서방형 구강붕해용 필름 및 이의 제조방법 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE209919T1 (de) * | 1987-09-24 | 2001-12-15 | Jencap Res Ltd | Oestrogen und progestin enthaltende verhütungspackungen |
| DK0630248T3 (da) * | 1992-03-21 | 1999-06-23 | Entec | Anvendelse af estriol til fremstilling af et transdermalt terapeutisk system til behandling af klimakteriel osteoporosis |
| DE19701949A1 (de) * | 1997-01-13 | 1998-07-16 | Jenapharm Gmbh | Transdermales therapeutisches System |
| DE19832169A1 (de) * | 1998-07-17 | 2000-01-27 | Jenapharm Gmbh | Lokal anwendbare pharmazeutische Präparate zur Prophylaxe und Therapie atrophischer Erscheinungen in der Mundhöhle |
| US6117446A (en) * | 1999-01-26 | 2000-09-12 | Place; Virgil A. | Drug dosage unit for buccal administration of steroidal active agents |
| DE19932603A1 (de) * | 1999-07-13 | 2001-01-25 | Gruenenthal Gmbh | Wirkstoffhaltiger Mehrschichtfilm aus in situ vernetzten hydrophilen Polymeren |
| RS52149B (sr) * | 2000-01-18 | 2012-08-31 | Bayer Schering Pharma Aktiengesellschaft | Farmaceutska kombinacija mikronizovanog drospirenona i estrogena za terapiju zamene hormona |
-
2004
- 2004-05-14 DE DE102004023984A patent/DE102004023984A1/de not_active Ceased
-
2005
- 2005-05-04 TW TW094114391A patent/TW200536547A/zh unknown
- 2005-05-06 JP JP2007512026A patent/JP2007537178A/ja active Pending
- 2005-05-06 EP EP05747659A patent/EP1761242A2/de not_active Withdrawn
- 2005-05-06 WO PCT/EP2005/004894 patent/WO2005110358A2/de not_active Ceased
- 2005-05-06 AU AU2005244409A patent/AU2005244409A1/en not_active Abandoned
- 2005-05-06 CN CNA2005800140311A patent/CN1997349A/zh active Pending
- 2005-05-06 KR KR1020067023835A patent/KR20070040753A/ko not_active Withdrawn
- 2005-05-06 BR BRPI0510855-1A patent/BRPI0510855A/pt not_active Application Discontinuation
- 2005-05-06 US US11/596,239 patent/US20070243217A1/en not_active Abandoned
- 2005-05-06 RU RU2006140649/15A patent/RU2006140649A/ru not_active Application Discontinuation
- 2005-05-06 MX MXPA06012890A patent/MXPA06012890A/es unknown
- 2005-05-06 CA CA002566325A patent/CA2566325A1/en not_active Abandoned
- 2005-05-13 AR ARP050101957A patent/AR048958A1/es unknown
-
2006
- 2006-11-02 IL IL179014A patent/IL179014A0/en unknown
- 2006-12-07 NO NO20065657A patent/NO20065657L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO20065657L (no) | 2006-12-07 |
| AU2005244409A1 (en) | 2005-11-24 |
| CA2566325A1 (en) | 2005-11-24 |
| EP1761242A2 (de) | 2007-03-14 |
| IL179014A0 (en) | 2007-03-08 |
| US20070243217A1 (en) | 2007-10-18 |
| TW200536547A (en) | 2005-11-16 |
| DE102004023984A1 (de) | 2005-12-08 |
| WO2005110358A2 (de) | 2005-11-24 |
| JP2007537178A (ja) | 2007-12-20 |
| CN1997349A (zh) | 2007-07-11 |
| MXPA06012890A (es) | 2007-07-19 |
| BRPI0510855A (pt) | 2007-12-26 |
| KR20070040753A (ko) | 2007-04-17 |
| RU2006140649A (ru) | 2008-05-27 |
| WO2005110358A3 (de) | 2007-03-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |