AR030258A1 - Proceso para la preparacion de derivados de tiazol y compuestos relacionados - Google Patents
Proceso para la preparacion de derivados de tiazol y compuestos relacionadosInfo
- Publication number
- AR030258A1 AR030258A1 ARP000104086A ARP000104086A AR030258A1 AR 030258 A1 AR030258 A1 AR 030258A1 AR P000104086 A ARP000104086 A AR P000104086A AR P000104086 A ARP000104086 A AR P000104086A AR 030258 A1 AR030258 A1 AR 030258A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparation
- related compounds
- tiazol
- derivatives
- chloro
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 239000002253 acid Substances 0.000 abstract 2
- PEOOQVDIOJQJHW-UHFFFAOYSA-N (2-chloro-1,3-thiazol-5-yl)methanol Chemical compound OCC1=CN=C(Cl)S1 PEOOQVDIOJQJHW-UHFFFAOYSA-N 0.000 abstract 1
- VRMUIVKEHJSADG-UHFFFAOYSA-N 2-chloro-5-(chloromethyl)-1,3-thiazole Chemical compound ClCC1=CN=C(Cl)S1 VRMUIVKEHJSADG-UHFFFAOYSA-N 0.000 abstract 1
- VEXZGXHMUGYJMC-UHFFFAOYSA-M Chloride anion Chemical compound [Cl-] VEXZGXHMUGYJMC-UHFFFAOYSA-M 0.000 abstract 1
- 150000001450 anions Chemical class 0.000 abstract 1
- 239000002917 insecticide Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 150000003557 thiazoles Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/34—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/50—Nitrogen atoms bound to hetero atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
Compuestos de tiazol intermediarios, (1) y (2) donde A- está definido en la memoria descriptiva. Un proceso para la preparacion del compuesto que tiene la formula (3) y sales de adicion de ácidodel mismo, el cual comprende el paso de hacer reaccionar 2-cloro-5-hidroximetiltiazol que tiene la formula (4) con una fuente de aniones de cloruro en la presencia de ácido. El compuesto 2-cloro-5-clorometil-tiazol es un intermediario conocido util para la preparacion de insecticidas.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/371,180 US6265553B1 (en) | 1999-08-10 | 1999-08-10 | Intermediate thiazoles and process for the preparation of 2-chloro-5-chloromethyl-thiazole |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR030258A1 true AR030258A1 (es) | 2003-08-20 |
Family
ID=23462834
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP000104086A AR030258A1 (es) | 1999-08-10 | 2000-08-08 | Proceso para la preparacion de derivados de tiazol y compuestos relacionados |
Country Status (19)
| Country | Link |
|---|---|
| US (4) | US6265553B1 (es) |
| EP (1) | EP1202979B1 (es) |
| JP (1) | JP2003506444A (es) |
| KR (1) | KR20020022796A (es) |
| CN (2) | CN1626525A (es) |
| AR (1) | AR030258A1 (es) |
| AT (1) | ATE294166T1 (es) |
| AU (1) | AU778367B2 (es) |
| BR (1) | BR0013235A (es) |
| CA (1) | CA2380838A1 (es) |
| CZ (1) | CZ2002483A3 (es) |
| DE (1) | DE60019763D1 (es) |
| ES (1) | ES2238029T3 (es) |
| HU (1) | HUP0202819A3 (es) |
| MX (1) | MXPA02001246A (es) |
| RU (1) | RU2002105516A (es) |
| TR (2) | TR200202474T2 (es) |
| WO (1) | WO2001010852A1 (es) |
| ZA (1) | ZA200201110B (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN100554249C (zh) | 2003-08-29 | 2009-10-28 | 三井化学株式会社 | 农园艺用杀虫剂及其使用方法 |
| BR112012020521B1 (pt) * | 2010-02-17 | 2017-12-26 | Syngenta Participations Ag | Derivative compounds of isoxazoline, its intermediaries and method for controlling insects, mites, nematodes, or molluscs |
| WO2011105632A1 (ja) * | 2010-02-26 | 2011-09-01 | 住友化学株式会社 | シクロプロパンカルボン酸エステル化合物の製造方法 |
| AU2012303664A1 (en) * | 2011-09-01 | 2014-04-10 | Biotelliga Holdings Limited | Insecticidal lipid agents isolated from entomopathogenic fungi and uses thereof |
| DE102015011861B4 (de) | 2015-09-10 | 2018-03-01 | Rudolf Schindler | Neue cyclische Carboxamide als NMDA NR2B Rezeptor Inhibitoren |
| CN106749086B (zh) * | 2016-12-27 | 2019-05-24 | 江苏振方生物化学有限公司 | 一种农药中间体2-氯-5-氯甲基噻唑的制备方法 |
| CN111036158A (zh) * | 2019-12-28 | 2020-04-21 | 邯郸市瑞田农药有限公司 | 一种2氯-5氯甲基噻唑合成反应系统 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3631538A1 (de) * | 1986-09-17 | 1988-03-24 | Bayer Ag | Verfahren zur herstellung von 2-chlor-5-chlormethylthiazol |
| DE69607293T2 (de) * | 1995-11-22 | 2000-12-14 | Kureha Chemical Industry Co., Ltd. | Verfahren zum Ersatz einer primären Aminogruppe durch Chlor und Verwendung dieses Verfahrens zur Herstellung von 2-Chlor-5-Chlormethylthiazol |
| JP2001508452A (ja) * | 1997-01-22 | 2001-06-26 | ノバルティス アクチェンゲゼルシャフト | チアゾール誘導体の製造方法 |
| US5773625A (en) * | 1997-10-02 | 1998-06-30 | Abbott Laboratories | Process for the preparation of disubstituted carbonates |
| US6407251B1 (en) * | 2000-12-28 | 2002-06-18 | Takeda Chemical Industries, Ltd. | Process for preparing 2-chloro-5-chloromethylthiazole |
-
1999
- 1999-08-10 US US09/371,180 patent/US6265553B1/en not_active Expired - Fee Related
-
2000
- 2000-08-08 AU AU68364/00A patent/AU778367B2/en not_active Ceased
- 2000-08-08 MX MXPA02001246A patent/MXPA02001246A/es unknown
- 2000-08-08 TR TR2002/02474T patent/TR200202474T2/xx unknown
- 2000-08-08 ES ES00956412T patent/ES2238029T3/es not_active Expired - Lifetime
- 2000-08-08 WO PCT/EP2000/007709 patent/WO2001010852A1/en not_active Ceased
- 2000-08-08 AT AT00956412T patent/ATE294166T1/de not_active IP Right Cessation
- 2000-08-08 CZ CZ2002483A patent/CZ2002483A3/cs unknown
- 2000-08-08 CN CNA2004100566415A patent/CN1626525A/zh active Pending
- 2000-08-08 KR KR1020027001623A patent/KR20020022796A/ko not_active Withdrawn
- 2000-08-08 US US10/049,073 patent/US6476230B1/en not_active Expired - Fee Related
- 2000-08-08 CN CNB008114455A patent/CN1169800C/zh not_active Expired - Fee Related
- 2000-08-08 BR BR0013235-7A patent/BR0013235A/pt not_active IP Right Cessation
- 2000-08-08 TR TR2002/00304T patent/TR200200304T2/xx unknown
- 2000-08-08 EP EP00956412A patent/EP1202979B1/en not_active Expired - Lifetime
- 2000-08-08 CA CA002380838A patent/CA2380838A1/en not_active Abandoned
- 2000-08-08 DE DE60019763T patent/DE60019763D1/de not_active Expired - Lifetime
- 2000-08-08 RU RU2002105516/04A patent/RU2002105516A/ru not_active Application Discontinuation
- 2000-08-08 JP JP2001515318A patent/JP2003506444A/ja active Pending
- 2000-08-08 HU HU0202819A patent/HUP0202819A3/hu not_active Application Discontinuation
- 2000-08-08 AR ARP000104086A patent/AR030258A1/es not_active Application Discontinuation
-
2002
- 2002-02-08 ZA ZA200201110A patent/ZA200201110B/en unknown
- 2002-09-16 US US10/244,236 patent/US6566530B2/en not_active Expired - Fee Related
-
2003
- 2003-05-07 US US10/431,100 patent/US6710182B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US6710182B2 (en) | 2004-03-23 |
| EP1202979B1 (en) | 2005-04-27 |
| US20030191321A1 (en) | 2003-10-09 |
| TR200200304T2 (tr) | 2002-06-21 |
| CN1169800C (zh) | 2004-10-06 |
| AU6836400A (en) | 2001-03-05 |
| RU2002105516A (ru) | 2003-09-20 |
| BR0013235A (pt) | 2002-04-23 |
| MXPA02001246A (es) | 2002-07-22 |
| EP1202979A1 (en) | 2002-05-08 |
| CZ2002483A3 (cs) | 2002-05-15 |
| US6476230B1 (en) | 2002-11-05 |
| CN1626525A (zh) | 2005-06-15 |
| US6265553B1 (en) | 2001-07-24 |
| HUP0202819A3 (en) | 2004-03-01 |
| WO2001010852A1 (en) | 2001-02-15 |
| KR20020022796A (ko) | 2002-03-27 |
| HUP0202819A2 (hu) | 2002-12-28 |
| CN1368966A (zh) | 2002-09-11 |
| ES2238029T3 (es) | 2005-08-16 |
| US6566530B2 (en) | 2003-05-20 |
| ATE294166T1 (de) | 2005-05-15 |
| ZA200201110B (en) | 2002-11-27 |
| TR200202474T2 (tr) | 2003-01-21 |
| JP2003506444A (ja) | 2003-02-18 |
| AU778367B2 (en) | 2004-12-02 |
| DE60019763D1 (de) | 2005-06-02 |
| US20030055229A1 (en) | 2003-03-20 |
| CA2380838A1 (en) | 2001-02-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |