AR039028A1 - Piridinil amidas biciclicas fusionadas y composiciones ventajosas de las mismas como fungicidas - Google Patents
Piridinil amidas biciclicas fusionadas y composiciones ventajosas de las mismas como fungicidasInfo
- Publication number
- AR039028A1 AR039028A1 ARP030100969A ARP030100969A AR039028A1 AR 039028 A1 AR039028 A1 AR 039028A1 AR P030100969 A ARP030100969 A AR P030100969A AR P030100969 A ARP030100969 A AR P030100969A AR 039028 A1 AR039028 A1 AR 039028A1
- Authority
- AR
- Argentina
- Prior art keywords
- fused
- ring
- atoms
- alkyl
- alkylamino
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- 239000000417 fungicide Substances 0.000 title 1
- 125000003282 alkyl amino group Chemical group 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 4
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 abstract 3
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 abstract 3
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 abstract 3
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 3
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 3
- JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical compound O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 3
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 3
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 abstract 3
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 3
- 125000004414 alkyl thio group Chemical group 0.000 abstract 3
- 125000004429 atom Chemical group 0.000 abstract 3
- 125000004432 carbon atom Chemical group C* 0.000 abstract 3
- 125000006310 cycloalkyl amino group Chemical group 0.000 abstract 3
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 3
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 abstract 3
- 125000000262 haloalkenyl group Chemical group 0.000 abstract 3
- 125000000232 haloalkynyl group Chemical group 0.000 abstract 3
- 125000005347 halocycloalkyl group Chemical group 0.000 abstract 3
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 150000002367 halogens Chemical class 0.000 abstract 3
- 125000004665 trialkylsilyl group Chemical group 0.000 abstract 3
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 abstract 2
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 2
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 2
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 2
- 230000009418 agronomic effect Effects 0.000 abstract 2
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 2
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 2
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 abstract 2
- 125000004995 haloalkylthio group Chemical group 0.000 abstract 2
- 125000001072 heteroaryl group Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 1
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 abstract 1
- 125000006656 (C2-C4) alkenyl group Chemical group 0.000 abstract 1
- 125000006650 (C2-C4) alkynyl group Chemical group 0.000 abstract 1
- 150000001204 N-oxides Chemical class 0.000 abstract 1
- -1 N-oxides salts Chemical class 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 244000000004 fungal plant pathogen Species 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Compuestos de la fórmula (1), inclusive todos los isómeros geométricos y estereoisómeros, N-óxidos sales adecuadas para uso agronómico de los mismos donde X y ya sea Y o Z son una cadena de unión de 3 o 4 átomos de longitud unida a átomos de C contiguos y se toman junto con dichos átomos de C para formar un anillo fenilo fusionado, un anillo carbocíclico o heterocíclico no aromático fusionado de 5 o 6 miembros que incluye opcionalmente uno o dos miembros del anillo seleccionados del grupo formado por C(=O), SO y S(O)2, o un anillo heteroaromático fusionado de 5 o 6 miembros, estando cada anillo opcionalmente fusionado con entre uno y tres sustituyentes seleccionados independientemente entre R7; y R1, R2, R5, R6, R7, n y p son como se definieron en la memoria descriptiva. También se describen composiciones que contienen los compuestos de la fórmula (1) y un método para controlar enfermedades en plantas causadas por patógenos fúngicos vegetales que comprende aplicar una cantidad eficaz de un compuesto de la fórmula (1). Reivindicación 1: Un compuesto, caracterizado porque se selecciona entre la fórmula (1) y N-óxidos y sales aceptables para uso agronómico del mismo donde: R1 y R2 son cada uno en forma independiente H, o alquilo C1-6; X y ya sea Y o Z son una cadena de unión de 3 o 4 átomos de longitud unida a átomos de C contiguos y se toman junto con dichos átomos de C para formar un anillo fenilo fusionado, un anillo carbocíclico o heterocíclico no aromático fusionado de 5 o 6 miembros que incluye opcionalmente 1 o 2 miembros del anillo seleccionados del grupo formado por C(=O), SO y S(O)2, o un anillo heteroaromático fusionado de 5 o 6 miembros, estando cada anillo opcionalmente fusionado con entre 1 y 3 sustituyentes seleccionados independientemente entre R7; cada R5 es en forma independiente alquilo C1-6, alquenilo C2-6, alquinilo C2-6, cicloalquilo C3-6, haloalquilo C1-6, haloalquenilo C2-6, haloalquinilo C2-6, halocicloalquilo C3-6, halógeno, CN, CO2H, CONH2, NO2, hidroxi, alcoxi C1-4, haloalcoxi C1-4, alquiltio C1-4, alquilsulfinilo C1-4, alquilsulfonilo C1-4, haloalquiltio C1-4, haloalquilsulfinilo C1-4, haloalquilsulfonilo C1-4, alquilamino C1-4, dialquilamino C2-8, cicloalquilamino C3-6, alquilcarbonilo C2-6, alcoxicarbonilo C2-6, alquilaminocarbonilo C2-6, dialquilaminocarbonilo C3-8 o trialquilsililo C3-6, cada R6 es en forma independiente C1-6 alquilo, C2-6 alquenilo, C2-6 alquinilo, C3-6 cicloalquilo, C1-6 haloalquilo, C2-6 haloalquenilo, C2-6 haloalquinilo, C3-6 halocicloalquilo, halógeno, CN, CO2H, CONH2, NO2, hidroxi, C1-4 alcoxi, C1-4 haloalcoxi, C1-4 alquiltio, C1-4 alquilsulfinilo, C1-4 alquilsulfonilo, C1-4 haloalquiltio, C1-4 haloalquilsulfinilo, C1-4 haloalquilsulfonilo, C1-4 alquilamino, C2-8 dialquilamino, C3-6 cicloalquilamino, C2-6 alquilcarbonilo, C2-6 alcoxicarbonilo, C2-6 alquilaminocarbonilo, C3-8 dialquilaminocarbonilo o C3-6 trialquilsililo; cada R7 es en forma independiente C1-4 alquilo, C2-4 alquenilo, C2-4 alquinilo, C3-6 cicloalquilo, C1-4 haloalquilo, C2-4 haloalquenilo, C2-4 haloalquinilo, C3-6 halocicloalquilo, halógeno, CN, NO2, C1-4 alcoxi, C1-4 haloalcoxi, C1-4 alquiltio, C1-4 alquilsulfinilo, C1-4 alquilsulfonilo, C1-4 alquilamino, C2-8 dialquilamino, C3-6 cicloalquilamino, C3-6 (alquil)cicloalquilamino, C2-4 alquilcarbonilo, C2-6 alcoxicarbonilo, C2-6 alquilaminocarbonilo. C3-8 dialquilaminocarbonilo o C3-6 trialquilsililo; m es 1, 2, 3, o 4; y p es 0, 1, o 2.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US36576702P | 2002-03-19 | 2002-03-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR039028A1 true AR039028A1 (es) | 2005-02-02 |
Family
ID=28454714
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP030100969A AR039028A1 (es) | 2002-03-19 | 2003-03-19 | Piridinil amidas biciclicas fusionadas y composiciones ventajosas de las mismas como fungicidas |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20050020644A1 (es) |
| EP (1) | EP1485372A2 (es) |
| JP (1) | JP2005526100A (es) |
| CN (1) | CN1642940A (es) |
| AR (1) | AR039028A1 (es) |
| AU (1) | AU2003216364A1 (es) |
| BR (1) | BR0308458A (es) |
| IL (1) | IL162892A0 (es) |
| MX (1) | MXPA04009002A (es) |
| PL (1) | PL372988A1 (es) |
| RU (1) | RU2004130832A (es) |
| TW (1) | TW200306159A (es) |
| WO (1) | WO2003080596A2 (es) |
| ZA (1) | ZA200405643B (es) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200407075A (en) * | 2002-03-19 | 2004-05-16 | Du Pont | Pyridinyl amides and advantageous compositions thereof for use as fungicides |
| US20090209589A1 (en) * | 2006-07-06 | 2009-08-20 | Bayer Cropscience Sa | N-[(pyridin-2-yl) methoxy] hetrocyclyl carboxamide derivatives and related compounds as fungicides |
| US7964732B2 (en) | 2006-11-17 | 2011-06-21 | Pfizer Inc. | Substituted bicyclocarboxyamide compounds |
| JP2009114178A (ja) * | 2007-10-15 | 2009-05-28 | Sumitomo Chemical Co Ltd | アミド化合物及びその植物病害防除用途 |
| JP2009120587A (ja) * | 2007-10-23 | 2009-06-04 | Sumitomo Chemical Co Ltd | アミド化合物及びその用途 |
| EP3632899A1 (en) | 2009-05-29 | 2020-04-08 | RaQualia Pharma Inc. | Aryl substituted carboxamide derivatives as calcium or sodium channel blockers |
| CN106478497B (zh) * | 2010-10-18 | 2020-05-08 | 拉夸里亚创药株式会社 | 作为ttx-s阻滞剂的芳胺衍生物 |
| WO2013003315A2 (en) * | 2011-06-26 | 2013-01-03 | President And Fellows Of Harvard College | Methods for preparing isoquinolines |
| BR112017023448A2 (pt) * | 2015-04-29 | 2018-07-31 | The State Of Israel, Ministry Of Agriculture & Rural Development, Agricultural Research Organization (Aro) (Volcani Center) | composições anti-fitopatogênicas |
| EP3681870B1 (en) * | 2017-09-13 | 2021-08-04 | Syngenta Participations AG | Microbiocidal quinoline (thio)carboxamide derivatives |
| US11185074B2 (en) * | 2017-09-13 | 2021-11-30 | Syngenta Participations Ag | Microbiocidal quinoline (thio)carboxamide derivatives |
| JP7150009B2 (ja) * | 2017-09-13 | 2022-10-07 | シンジェンタ パーティシペーションズ アーゲー | 殺微生物性キノリン（チオ）カルボキサミド誘導体 |
| WO2021063736A1 (en) * | 2019-10-02 | 2021-04-08 | Basf Se | Bicyclic pyridine derivatives |
| WO2022150962A1 (en) * | 2021-01-12 | 2022-07-21 | Westlake Pharmaceutical (Hangzhou) Co., Ltd. | Protease inhibitors, preparation, and uses thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2704256A1 (en) * | 1997-12-18 | 1999-07-01 | Basf Aktiengesellschaft | Fungicide mixtures based on pyridine carboxamides |
| GB9919588D0 (en) * | 1999-08-18 | 1999-10-20 | Hoechst Schering Agrevo Gmbh | Fungicidal compounds |
| WO2002022583A2 (en) * | 2000-09-18 | 2002-03-21 | E. I. Du Pont De Nemours And Company | Pyridinyl amides and imides for use as fungicides |
-
2003
- 2003-02-19 TW TW092103415A patent/TW200306159A/zh unknown
- 2003-02-20 MX MXPA04009002A patent/MXPA04009002A/es unknown
- 2003-02-20 AU AU2003216364A patent/AU2003216364A1/en not_active Abandoned
- 2003-02-20 PL PL03372988A patent/PL372988A1/xx not_active Application Discontinuation
- 2003-02-20 CN CN03806571.1A patent/CN1642940A/zh active Pending
- 2003-02-20 RU RU2004130832/04A patent/RU2004130832A/ru not_active Application Discontinuation
- 2003-02-20 EP EP03745079A patent/EP1485372A2/en not_active Withdrawn
- 2003-02-20 IL IL16289203A patent/IL162892A0/xx unknown
- 2003-02-20 BR BR0308458-2A patent/BR0308458A/pt not_active IP Right Cessation
- 2003-02-20 US US10/501,258 patent/US20050020644A1/en not_active Abandoned
- 2003-02-20 JP JP2003578350A patent/JP2005526100A/ja not_active Withdrawn
- 2003-02-20 WO PCT/US2003/005383 patent/WO2003080596A2/en not_active Ceased
- 2003-03-19 AR ARP030100969A patent/AR039028A1/es not_active Application Discontinuation
-
2004
- 2004-07-15 ZA ZA200405643A patent/ZA200405643B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL162892A0 (en) | 2005-11-20 |
| WO2003080596A3 (en) | 2004-04-01 |
| AU2003216364A1 (en) | 2003-10-08 |
| CN1642940A (zh) | 2005-07-20 |
| PL372988A1 (en) | 2005-08-08 |
| TW200306159A (en) | 2003-11-16 |
| BR0308458A (pt) | 2005-01-18 |
| WO2003080596A2 (en) | 2003-10-02 |
| EP1485372A2 (en) | 2004-12-15 |
| RU2004130832A (ru) | 2005-04-10 |
| US20050020644A1 (en) | 2005-01-27 |
| AU2003216364A8 (en) | 2003-10-08 |
| MXPA04009002A (es) | 2004-12-07 |
| ZA200405643B (en) | 2005-07-15 |
| JP2005526100A (ja) | 2005-09-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |