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AR036423A1 - Composicion farmaceutica. - Google Patents

Composicion farmaceutica.

Info

Publication number
AR036423A1
AR036423A1 ARP020103331A ARP020103331A AR036423A1 AR 036423 A1 AR036423 A1 AR 036423A1 AR P020103331 A ARP020103331 A AR P020103331A AR P020103331 A ARP020103331 A AR P020103331A AR 036423 A1 AR036423 A1 AR 036423A1
Authority
AR
Argentina
Prior art keywords
butyrobetaine
stimulation
pharmaceutical compositions
sexual activity
narcotized
Prior art date
Application number
ARP020103331A
Other languages
English (en)
Inventor
Ivars Kalvinsh
Maris Veveris
Anatolijs Birmans
Original Assignee
Anatolijs Birmans
Maris Veveris
Ivars Kalvinsh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anatolijs Birmans, Maris Veveris, Ivars Kalvinsh filed Critical Anatolijs Birmans
Publication of AR036423A1 publication Critical patent/AR036423A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/205Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Reproductive Health (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Utilización médica para la gamma-butirobetaína. Composiciones farmacéuticas que contienen gamma-butirobetaína o combinación de esta con 3-(2,2,2-trimetilhidrazinio) propionato o sildenafil para la aplicación oral, parenteral, subcutánea, transdérmica, tópica, sublingual, intrauretral, intranasal o rectal, útiles para la estimulación de la actividad y potencia sexuales en los mamíferos. Las composiciones cuando se aplican en forma oral durante 6 semanas a ratas macho no narcotizadas, aumentan en forma sustancial su actividad sexual, disminuyendo el tiempo de excitación, aumentando el número de copulaciones y los resultados de tentativas de monta. Cuando se aplica por ruta intracavernosa o intravenosa, dichas composiciones farmacéuticas aumentan la presión intracorporal y la duración de la erección, así como devuelve la erección reflectiva inducida por la estimulación en los animales narcotizados.
ARP020103331A 2001-09-07 2002-09-04 Composicion farmaceutica. AR036423A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
LVP-01-134A LV12979B (en) 2001-09-07 2001-09-07 Pharmaceutical composition

Publications (1)

Publication Number Publication Date
AR036423A1 true AR036423A1 (es) 2004-09-08

Family

ID=19735292

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP020103331A AR036423A1 (es) 2001-09-07 2002-09-04 Composicion farmaceutica.

Country Status (29)

Country Link
US (1) US20040242590A1 (es)
EP (1) EP1429753B1 (es)
JP (1) JP4382480B2 (es)
KR (1) KR100841035B1 (es)
CN (1) CN1275595C (es)
AR (1) AR036423A1 (es)
AT (1) ATE350029T1 (es)
AU (1) AU2002236340B2 (es)
BG (1) BG108673A (es)
CA (1) CA2459719C (es)
CU (1) CU23347B6 (es)
DE (1) DE60217369T2 (es)
DK (1) DK1429753T3 (es)
EA (1) EA006675B1 (es)
ES (1) ES2280505T3 (es)
HR (1) HRPK20040328B3 (es)
IL (2) IL160734A0 (es)
JO (1) JO2507B1 (es)
LV (1) LV12979B (es)
MA (1) MA27683A1 (es)
MX (1) MXPA04002050A (es)
MY (1) MY134074A (es)
NZ (1) NZ532178A (es)
PL (1) PL368758A1 (es)
PT (1) PT1429753E (es)
SI (1) SI1429753T1 (es)
TW (1) TWI224506B (es)
WO (1) WO2003022262A1 (es)
ZA (1) ZA200402702B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10325813B4 (de) 2003-06-06 2007-12-20 Universitätsklinikum Freiburg Prophylaxe und/oder Therapie bei der portalen Hypertonie
LV13450B (en) * 2004-08-24 2006-11-20 Grindeks As Novel medicinal use of meldonium and pharmaceutical compositions thereof
KR20080047375A (ko) 2005-07-29 2008-05-28 콘서트 파마슈티컬즈, 인크. 약제 화합물
WO2009095445A1 (en) * 2008-01-29 2009-08-06 Grindeks New second medical use of 3-(2,2,2-trimethylhydrazine)propionate dihydrate
CN101781302B (zh) * 2009-05-31 2013-07-10 段波 一种磷酸二酯酶抑制剂和异黄酮形成的加成物及其应用
RU2622757C1 (ru) * 2016-06-02 2017-06-19 федеральное государственное автономное образовательное учреждение высшего образования Первый Московский государственный медицинский университет имени И.М. Сеченова Министерства здравоохранения Российской Федерации (Сеченовский университет) Способ лечения эректильной дисфункции

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1198434B (it) * 1981-01-06 1988-12-21 Sigma Tau Ind Farmaceuti Composizione farmaceutica comprendente gamma butirrobetaina per il trattamento di sindromi da carenze di carnitina
LV11728B (en) * 1995-08-21 1997-08-20 Kalvins Ivars Pharmaceutical composition
LV11727B (en) * 1995-08-21 1997-08-20 Kalvins Ivars Pharmaceutical composition

Also Published As

Publication number Publication date
CA2459719C (en) 2010-07-06
DE60217369T2 (de) 2007-08-23
NZ532178A (en) 2007-05-31
CN1551764A (zh) 2004-12-01
HK1068003A1 (en) 2005-04-22
KR20040034704A (ko) 2004-04-28
MXPA04002050A (es) 2004-06-07
IL160734A0 (en) 2004-08-31
LV12979B (en) 2003-05-20
KR100841035B1 (ko) 2008-06-24
EP1429753B1 (en) 2007-01-03
ZA200402702B (en) 2005-05-11
SI1429753T1 (sl) 2007-06-30
EA006675B1 (ru) 2006-02-24
DE60217369D1 (de) 2007-02-15
ATE350029T1 (de) 2007-01-15
PT1429753E (pt) 2007-04-30
HRP20040328A2 (en) 2004-08-31
EP1429753A1 (en) 2004-06-23
WO2003022262A1 (en) 2003-03-20
HRPK20040328B3 (en) 2006-02-28
IL160734A (en) 2009-09-22
MA27683A1 (fr) 2006-01-02
US20040242590A1 (en) 2004-12-02
TWI224506B (en) 2004-12-01
CA2459719A1 (en) 2003-03-20
PL368758A1 (en) 2005-04-04
JO2507B1 (en) 2009-10-05
CN1275595C (zh) 2006-09-20
EA200400386A1 (ru) 2004-08-26
JP2005504071A (ja) 2005-02-10
AU2002236340B2 (en) 2008-06-12
DK1429753T3 (da) 2007-05-14
BG108673A (en) 2005-03-31
JP4382480B2 (ja) 2009-12-16
MY134074A (en) 2007-11-30
ES2280505T3 (es) 2007-09-16
CU23347B6 (es) 2009-02-20

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Legal Events

Date Code Title Description
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