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AR022930A2 - MICROCAPSULAS, DE TIPO RESERVORIO, QUE CONTIENEN POR LO MENOS UN PRINCIPIO ACTIVO MEDICAMENTOSO Y/O NUTRITIVO (PA) CON EXCLUSION DEL ACIDO ACETILSALICILICO (ASA), DESTINADAS A LA ADMINISTRACION POR VIA ORAL, SU UTILIZACIoN Y FORMA FARMACEUTICA QUE COMPRENDE A DICHAS MICROCAPSULAS. - Google Patents

MICROCAPSULAS, DE TIPO RESERVORIO, QUE CONTIENEN POR LO MENOS UN PRINCIPIO ACTIVO MEDICAMENTOSO Y/O NUTRITIVO (PA) CON EXCLUSION DEL ACIDO ACETILSALICILICO (ASA), DESTINADAS A LA ADMINISTRACION POR VIA ORAL, SU UTILIZACIoN Y FORMA FARMACEUTICA QUE COMPRENDE A DICHAS MICROCAPSULAS.

Info

Publication number
AR022930A2
AR022930A2 ARP000101126A ARP000101126A AR022930A2 AR 022930 A2 AR022930 A2 AR 022930A2 AR P000101126 A ARP000101126 A AR P000101126A AR P000101126 A ARP000101126 A AR P000101126A AR 022930 A2 AR022930 A2 AR 022930A2
Authority
AR
Argentina
Prior art keywords
microcapsules
medicinal
administration
reservory
asa
Prior art date
Application number
ARP000101126A
Other languages
English (en)
Original Assignee
Flamel Tech Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9468196&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR022930(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Flamel Tech Sa filed Critical Flamel Tech Sa
Publication of AR022930A2 publication Critical patent/AR022930A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5015Organic compounds, e.g. fats, sugars
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se proveen microcápsulas para la administracion oral de principios activos medicamentosos y/o nutritivos (PA), cuyos tamanos son inferiores o iguales a1.000 microm. Estas microcápsulas están compuestas por partículas que están recubiertas por unasub stancia de recubrimiento constituida por una mezcla de underivado polímero filmogeno, de un agente plastificante hidrofobo, de un agente tensioactivo y/o lubricante y de un polímero nitrogenado. Estas microcápsulasposeen la aptitud parapermanecer la rgo tiempo (por lo menos 5 horas) en el intestino delgado y para permitir, después de esta permanencia, la adsorcion del PAdurante un período superior al tiempo de tránsito natural en el intestino delgado. Asimismo se proveen susaplicaciones en medi cina y un sistema galénico,preferentemente en forma de comprimido, ventajosamente disgregable, de polvo o de cápsula gelatinosa que comprende a las microcápsulas.
ARP000101126A 1994-10-18 2000-03-15 MICROCAPSULAS, DE TIPO RESERVORIO, QUE CONTIENEN POR LO MENOS UN PRINCIPIO ACTIVO MEDICAMENTOSO Y/O NUTRITIVO (PA) CON EXCLUSION DEL ACIDO ACETILSALICILICO (ASA), DESTINADAS A LA ADMINISTRACION POR VIA ORAL, SU UTILIZACIoN Y FORMA FARMACEUTICA QUE COMPRENDE A DICHAS MICROCAPSULAS. AR022930A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9412759A FR2725623A1 (fr) 1994-10-18 1994-10-18 Microcapsules medicamenteuses et/ou nutritionnelles pour administration per os

Publications (1)

Publication Number Publication Date
AR022930A2 true AR022930A2 (es) 2002-09-04

Family

ID=9468196

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000101126A AR022930A2 (es) 1994-10-18 2000-03-15 MICROCAPSULAS, DE TIPO RESERVORIO, QUE CONTIENEN POR LO MENOS UN PRINCIPIO ACTIVO MEDICAMENTOSO Y/O NUTRITIVO (PA) CON EXCLUSION DEL ACIDO ACETILSALICILICO (ASA), DESTINADAS A LA ADMINISTRACION POR VIA ORAL, SU UTILIZACIoN Y FORMA FARMACEUTICA QUE COMPRENDE A DICHAS MICROCAPSULAS.

Country Status (14)

Country Link
US (1) US6022562A (es)
EP (1) EP0709087B1 (es)
JP (1) JP4053589B2 (es)
AR (1) AR022930A2 (es)
AT (1) ATE188117T1 (es)
AU (1) AU3807795A (es)
BR (2) BR9509286A (es)
CA (1) CA2160762C (es)
DE (1) DE69514192T2 (es)
ES (1) ES2140641T3 (es)
FR (1) FR2725623A1 (es)
IL (1) IL115646A (es)
WO (1) WO1996011675A2 (es)
ZA (1) ZA958762B (es)

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JP4053589B2 (ja) 2008-02-27
DE69514192D1 (de) 2000-02-03
ES2140641T3 (es) 2000-03-01
AU3807795A (en) 1996-05-06
EP0709087A1 (fr) 1996-05-01
WO1996011675A3 (fr) 1996-06-20
WO1996011675A2 (fr) 1996-04-25
IL115646A (en) 2000-07-16
US6022562A (en) 2000-02-08
FR2725623B1 (es) 1997-02-21
ZA958762B (en) 1996-05-09
FR2725623A1 (fr) 1996-04-19
CA2160762A1 (fr) 1996-04-19
BR9509286A (pt) 1997-10-14
JPH10509427A (ja) 1998-09-14
DE69514192T2 (de) 2000-07-13
ATE188117T1 (de) 2000-01-15
IL115646A0 (en) 1996-01-19
EP0709087B1 (fr) 1999-12-29
CA2160762C (fr) 2004-12-21
BRPI9509286B8 (pt) 2019-12-17

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